JP2023519824A5 - - Google Patents
Info
- Publication number
- JP2023519824A5 JP2023519824A5 JP2022556491A JP2022556491A JP2023519824A5 JP 2023519824 A5 JP2023519824 A5 JP 2023519824A5 JP 2022556491 A JP2022556491 A JP 2022556491A JP 2022556491 A JP2022556491 A JP 2022556491A JP 2023519824 A5 JP2023519824 A5 JP 2023519824A5
- Authority
- JP
- Japan
- Prior art keywords
- compound according
- optionally substituted
- alkyl
- cycloalkyl
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2025177542A JP2026009184A (ja) | 2020-04-03 | 2025-10-22 | 補体阻害剤としてのピロロピリミジンアミン |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202063004799P | 2020-04-03 | 2020-04-03 | |
| US63/004,799 | 2020-04-03 | ||
| PCT/US2021/025547 WO2021202977A1 (en) | 2020-04-03 | 2021-04-02 | Pyrrolopyrimidine amines as complement inhibitors |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025177542A Division JP2026009184A (ja) | 2020-04-03 | 2025-10-22 | 補体阻害剤としてのピロロピリミジンアミン |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023519824A JP2023519824A (ja) | 2023-05-15 |
| JP2023519824A5 true JP2023519824A5 (https=) | 2024-05-02 |
| JP7763772B2 JP7763772B2 (ja) | 2025-11-04 |
Family
ID=77929437
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022556491A Active JP7763772B2 (ja) | 2020-04-03 | 2021-04-02 | 補体阻害剤としてのピロロピリミジンアミン |
| JP2025177542A Pending JP2026009184A (ja) | 2020-04-03 | 2025-10-22 | 補体阻害剤としてのピロロピリミジンアミン |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025177542A Pending JP2026009184A (ja) | 2020-04-03 | 2025-10-22 | 補体阻害剤としてのピロロピリミジンアミン |
Country Status (25)
| Country | Link |
|---|---|
| US (1) | US20230159536A1 (https=) |
| EP (1) | EP4125914A4 (https=) |
| JP (2) | JP7763772B2 (https=) |
| KR (1) | KR20220163955A (https=) |
| CN (1) | CN115427044A (https=) |
| AR (1) | AR121715A1 (https=) |
| AU (1) | AU2021246098A1 (https=) |
| BR (1) | BR112022018067A2 (https=) |
| CA (1) | CA3176808A1 (https=) |
| CL (1) | CL2022002649A1 (https=) |
| CO (1) | CO2022015630A2 (https=) |
| CR (1) | CR20220553A (https=) |
| CU (1) | CU20220060A7 (https=) |
| DO (2) | DOP2022000211A (https=) |
| EC (1) | ECSP22085221A (https=) |
| GE (1) | GEP20257841B (https=) |
| IL (1) | IL296978A (https=) |
| JO (2) | JOP20220227A1 (https=) |
| MX (1) | MX2022012056A (https=) |
| PE (1) | PE20230601A1 (https=) |
| PY (1) | PY2126225A (https=) |
| TN (1) | TN2022000255A1 (https=) |
| TW (1) | TWI912303B (https=) |
| UY (1) | UY39150A (https=) |
| WO (1) | WO2021202977A1 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2023069301A1 (en) * | 2021-10-18 | 2023-04-27 | Alexion Pharmaceuticals, Inc. | Use of complement factor d inhibitor for treatment of lupus nephritis and immunoglobulin a nephropathy |
| WO2024008121A1 (zh) * | 2022-07-06 | 2024-01-11 | 南京明德新药研发有限公司 | 二氟取代的氮杂双环化合物及其应用 |
| JP2025530036A (ja) * | 2022-09-01 | 2025-09-10 | エフ． ホフマン－ラ ロシュ アーゲー | ビカシナビンの投与レジメン |
| US11945818B1 (en) | 2023-09-06 | 2024-04-02 | King Faisal University | Pyrrolo[3,2-c]quinoline compounds as CK2 inhibitors |
| US11964981B1 (en) | 2023-09-18 | 2024-04-23 | King Faisal University | Substituted pyrimido[4,5-b]indoles as CK2 inhibitors |
| WO2025217212A1 (en) * | 2024-04-09 | 2025-10-16 | The Regents Of The University Of California | Mac1 inhibitors and uses thereof |
Family Cites Families (29)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4559157A (en) | 1983-04-21 | 1985-12-17 | Creative Products Resource Associates, Ltd. | Cosmetic applicator useful for skin moisturizing |
| LU84979A1 (fr) | 1983-08-30 | 1985-04-24 | Oreal | Composition cosmetique ou pharmaceutique sous forme aqueuse ou anhydre dont la phase grasse contient un polyether oligomere et polyethers oligomeres nouveaux |
| LU86084A1 (fr) | 1985-09-20 | 1987-04-02 | Faco Sa | Apparei de massage electrique |
| US5102417A (en) | 1985-11-07 | 1992-04-07 | Expandable Grafts Partnership | Expandable intraluminal graft, and method and apparatus for implanting an expandable intraluminal graft |
| US4800882A (en) | 1987-03-13 | 1989-01-31 | Cook Incorporated | Endovascular stent and delivery system |
| US4820508A (en) | 1987-06-23 | 1989-04-11 | Neutrogena Corporation | Skin protective composition |
| US4886062A (en) | 1987-10-19 | 1989-12-12 | Medtronic, Inc. | Intravascular radially expandable stent and method of implant |
| US4992478A (en) | 1988-04-04 | 1991-02-12 | Warner-Lambert Company | Antiinflammatory skin moisturizing composition and method of preparing same |
| US4938949A (en) | 1988-09-12 | 1990-07-03 | University Of New York | Treatment of damaged bone marrow and dosage units therefor |
| WO1990013332A1 (en) | 1989-05-11 | 1990-11-15 | Cedars-Sinai Medical Center | Stent with sustained drug delivery |
| DE69110787T2 (de) | 1990-02-28 | 1996-04-04 | Medtronic, Inc., Minneapolis, Minn. | Intraluminale prothese mit wirkstoffeluierung. |
| US5429634A (en) | 1993-09-09 | 1995-07-04 | Pdt Systems | Biogenic implant for drug delivery and method |
| US5419760A (en) | 1993-01-08 | 1995-05-30 | Pdt Systems, Inc. | Medicament dispensing stent for prevention of restenosis of a blood vessel |
| US6774278B1 (en) | 1995-06-07 | 2004-08-10 | Cook Incorporated | Coated implantable medical device |
| IL123986A (en) * | 1997-04-24 | 2011-10-31 | Organon Nv | Medicinal compounds |
| JPH11292840A (ja) * | 1998-04-06 | 1999-10-26 | Soyaku Gijutsu Kenkyusho:Kk | ノルスタチン誘導体又はその塩 |
| EP1144373B1 (en) | 1999-01-13 | 2005-10-19 | Genentech, Inc. | Serine protease inhibitors |
| US6770729B2 (en) | 2002-09-30 | 2004-08-03 | Medtronic Minimed, Inc. | Polymer compositions containing bioactive agents and methods for their use |
| PT2661433T (pt) | 2011-01-04 | 2017-10-24 | Novartis Ag | Compostos de indole ou seus análogos úteis para o tratamento da degeneração macular relacionada com a idade (amd) |
| CN104379579B (zh) | 2012-06-28 | 2017-03-08 | 诺华股份有限公司 | 吡咯烷衍生物及其作为补体途径调节剂的用途 |
| AR106018A1 (es) | 2015-08-26 | 2017-12-06 | Achillion Pharmaceuticals Inc | Compuestos de arilo, heteroarilo y heterocíclicos para el tratamiento de trastornos médicos |
| WO2017035348A1 (en) | 2015-08-26 | 2017-03-02 | Achillion Pharmaceuticals, Inc. | Alkyne compounds for treatment of medical disorders |
| AR105809A1 (es) * | 2015-08-26 | 2017-11-08 | Achillion Pharmaceuticals Inc | Compuestos para el tratamiento de trastornos médicos |
| AR105808A1 (es) | 2015-08-26 | 2017-11-08 | Achillion Pharmaceuticals Inc | Compuestos de amida para el tratamiento de trastornos médicos |
| US10385097B2 (en) | 2015-08-26 | 2019-08-20 | Achillion Pharmaceuticals, Inc. | Ether compounds for treatment of medical disorders |
| TWI747873B (zh) | 2016-02-01 | 2021-12-01 | 美商百歐克斯製藥公司 | 苯并吡唑化合物及其類似物 |
| CN110603252A (zh) | 2017-03-01 | 2019-12-20 | 艾其林医药公司 | 用于治疗医学障碍的芳基、杂芳基和杂环药物化合物 |
| WO2018229543A2 (en) | 2017-06-14 | 2018-12-20 | Lifesci Pharmaceuticals, Inc. | Therapeutic inhibitory compounds |
| TWI873092B (zh) | 2018-04-06 | 2025-02-21 | 美商百歐克斯製藥公司 | 取代的苯并呋喃、苯并吡咯、苯并噻吩及結構相關的補體抑制劑 |
-
2021
- 2021-03-31 AR ARP210100817A patent/AR121715A1/es unknown
- 2021-04-01 TW TW110112139A patent/TWI912303B/zh active
- 2021-04-02 BR BR112022018067A patent/BR112022018067A2/pt unknown
- 2021-04-02 GE GEAP202116073A patent/GEP20257841B/en unknown
- 2021-04-02 KR KR1020227033595A patent/KR20220163955A/ko active Pending
- 2021-04-02 JP JP2022556491A patent/JP7763772B2/ja active Active
- 2021-04-02 PE PE2022002121A patent/PE20230601A1/es unknown
- 2021-04-02 CN CN202180025930.0A patent/CN115427044A/zh active Pending
- 2021-04-02 AU AU2021246098A patent/AU2021246098A1/en active Pending
- 2021-04-02 TN TNP/2022/000255A patent/TN2022000255A1/en unknown
- 2021-04-02 MX MX2022012056A patent/MX2022012056A/es unknown
- 2021-04-02 JO JOP/2022/0227A patent/JOP20220227A1/ar unknown
- 2021-04-02 EP EP21781014.2A patent/EP4125914A4/en active Pending
- 2021-04-02 CR CR20220553A patent/CR20220553A/es unknown
- 2021-04-02 CU CU2022000060A patent/CU20220060A7/es unknown
- 2021-04-02 CA CA3176808A patent/CA3176808A1/en active Pending
- 2021-04-02 WO PCT/US2021/025547 patent/WO2021202977A1/en not_active Ceased
- 2021-04-02 US US17/915,179 patent/US20230159536A1/en active Pending
- 2021-04-02 IL IL296978A patent/IL296978A/en unknown
- 2021-04-05 PY PY202102126225A patent/PY2126225A/es unknown
- 2021-04-05 UY UY0001039150A patent/UY39150A/es unknown
-
2022
- 2022-09-22 JO JOJO/P/2022/0228A patent/JOP20220228A1/ar unknown
- 2022-09-28 DO DO2022000211A patent/DOP2022000211A/es unknown
- 2022-09-28 CL CL2022002649A patent/CL2022002649A1/es unknown
- 2022-10-31 CO CONC2022/0015630A patent/CO2022015630A2/es unknown
- 2022-11-02 EC ECSENADI202285221A patent/ECSP22085221A/es unknown
-
2025
- 2025-02-26 DO DO2025000044A patent/DOP2025000044A/es unknown
- 2025-10-22 JP JP2025177542A patent/JP2026009184A/ja active Pending
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