JP2023519666A5 - - Google Patents
Info
- Publication number
- JP2023519666A5 JP2023519666A5 JP2022555137A JP2022555137A JP2023519666A5 JP 2023519666 A5 JP2023519666 A5 JP 2023519666A5 JP 2022555137 A JP2022555137 A JP 2022555137A JP 2022555137 A JP2022555137 A JP 2022555137A JP 2023519666 A5 JP2023519666 A5 JP 2023519666A5
- Authority
- JP
- Japan
- Prior art keywords
- pyridine
- carboxamide
- trifluoromethyl
- pyrazole
- fluoro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB2003668.7A GB202003668D0 (en) | 2020-03-13 | 2020-03-13 | GPR52 Modulator compounds |
| GB2003668.7 | 2020-03-13 | ||
| PCT/GB2021/050638 WO2021181122A1 (en) | 2020-03-13 | 2021-03-15 | Gpr52 modulator compounds |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023519666A JP2023519666A (ja) | 2023-05-12 |
| JP2023519666A5 true JP2023519666A5 (https=) | 2024-03-27 |
| JP7492597B2 JP7492597B2 (ja) | 2024-05-29 |
Family
ID=70453676
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022555137A Active JP7492597B2 (ja) | 2020-03-13 | 2021-03-15 | Ｇｐｒ５２モジュレーター化合物 |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US20240254101A1 (https=) |
| EP (1) | EP4117784B1 (https=) |
| JP (1) | JP7492597B2 (https=) |
| KR (1) | KR20220152296A (https=) |
| CN (1) | CN115515681B (https=) |
| AU (1) | AU2021235257A1 (https=) |
| BR (1) | BR112022018287A2 (https=) |
| CA (1) | CA3175429A1 (https=) |
| DK (1) | DK4117784T3 (https=) |
| ES (1) | ES2992600T3 (https=) |
| FI (1) | FI4117784T3 (https=) |
| GB (1) | GB202003668D0 (https=) |
| HR (1) | HRP20241375T1 (https=) |
| HU (1) | HUE068758T2 (https=) |
| IL (1) | IL296413B2 (https=) |
| LT (1) | LT4117784T (https=) |
| MX (1) | MX2022011333A (https=) |
| PL (1) | PL4117784T3 (https=) |
| PT (1) | PT4117784T (https=) |
| RS (1) | RS66063B1 (https=) |
| SI (1) | SI4117784T1 (https=) |
| SM (1) | SMT202400402T1 (https=) |
| WO (1) | WO2021181122A1 (https=) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW202206413A (zh) | 2020-04-22 | 2022-02-16 | 美商紐羅克里生物科學有限公司 | Gpr52調節劑及其使用方法 |
| EP4330232A1 (en) * | 2021-04-26 | 2024-03-06 | Neurocrine Biosciences, Inc. | Gpr52 modulators and methods of use |
| GB202113186D0 (en) | 2021-09-15 | 2021-10-27 | Heptares Therapeutics Ltd | GPR52 Modulator compounds |
| WO2024091541A1 (en) * | 2022-10-26 | 2024-05-02 | Neurocrine Biosciences, Inc. | Compounds and compositions as gpr52 modulators |
| JP2026508053A (ja) * | 2022-10-26 | 2026-03-10 | ニューロクライン バイオサイエンシーズ，インコーポレイテッド | Ｇｐｒ５２モジュレーターとしての化合物および組成物 |
| WO2024091542A1 (en) * | 2022-10-26 | 2024-05-02 | Neurocrine Biosciences, Inc. | Compounds and compositions as gpr52 modulators |
| WO2025252061A1 (zh) * | 2024-06-04 | 2025-12-11 | 海思科医药集团股份有限公司 | 一种gpr52激动剂及其在医药上的应用 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005037797A1 (en) * | 2003-10-21 | 2005-04-28 | Pharmacia Corporation | Substituted pyrazole urea compounds for the treatment of inflammation |
| WO2009107391A1 (ja) | 2008-02-27 | 2009-09-03 | 武田薬品工業株式会社 | ６員芳香環含有化合物 |
| WO2011078360A1 (ja) | 2009-12-24 | 2011-06-30 | 武田薬品工業株式会社 | アミド化合物 |
| EP2530078A1 (en) | 2010-01-27 | 2012-12-05 | Takeda Pharmaceutical Company Limited | Thiazole derivative |
| KR20180004193A (ko) * | 2015-04-29 | 2018-01-10 | 아레나 파마슈티칼스, 인크. | Gpr52와 관련된 장애의 치료 또는 예방을 위한 gpr52 조절제로서 1-헤테로아릴-인돌린-4-카르복스아미드 |
| JP7394747B2 (ja) * | 2017-09-13 | 2023-12-08 | ノバルティス アーゲー | ジフェニル誘導体及びその使用 |
-
2020
- 2020-03-13 GB GBGB2003668.7A patent/GB202003668D0/en not_active Ceased
-
2021
- 2021-03-15 HR HRP20241375TT patent/HRP20241375T1/hr unknown
- 2021-03-15 ES ES21713103T patent/ES2992600T3/es active Active
- 2021-03-15 EP EP21713103.6A patent/EP4117784B1/en active Active
- 2021-03-15 SI SI202130212T patent/SI4117784T1/sl unknown
- 2021-03-15 US US17/909,792 patent/US20240254101A1/en active Pending
- 2021-03-15 RS RS20241089A patent/RS66063B1/sr unknown
- 2021-03-15 AU AU2021235257A patent/AU2021235257A1/en active Pending
- 2021-03-15 IL IL296413A patent/IL296413B2/en unknown
- 2021-03-15 WO PCT/GB2021/050638 patent/WO2021181122A1/en not_active Ceased
- 2021-03-15 LT LTEPPCT/GB2021/050638T patent/LT4117784T/lt unknown
- 2021-03-15 DK DK21713103.6T patent/DK4117784T3/da active
- 2021-03-15 PT PT217131036T patent/PT4117784T/pt unknown
- 2021-03-15 CA CA3175429A patent/CA3175429A1/en active Pending
- 2021-03-15 SM SM20240402T patent/SMT202400402T1/it unknown
- 2021-03-15 MX MX2022011333A patent/MX2022011333A/es unknown
- 2021-03-15 PL PL21713103.6T patent/PL4117784T3/pl unknown
- 2021-03-15 KR KR1020227035100A patent/KR20220152296A/ko active Pending
- 2021-03-15 HU HUE21713103A patent/HUE068758T2/hu unknown
- 2021-03-15 BR BR112022018287A patent/BR112022018287A2/pt unknown
- 2021-03-15 FI FIEP21713103.6T patent/FI4117784T3/fi active
- 2021-03-15 CN CN202180033813.9A patent/CN115515681B/zh active Active
- 2021-03-15 JP JP2022555137A patent/JP7492597B2/ja active Active
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