JP2023518774A5 - - Google Patents
Info
- Publication number
- JP2023518774A5 JP2023518774A5 JP2022556468A JP2022556468A JP2023518774A5 JP 2023518774 A5 JP2023518774 A5 JP 2023518774A5 JP 2022556468 A JP2022556468 A JP 2022556468A JP 2022556468 A JP2022556468 A JP 2022556468A JP 2023518774 A5 JP2023518774 A5 JP 2023518774A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- alkoxy
- halogenated
- membered
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN202010183457 | 2020-03-16 | ||
| CN202010183457.6 | 2020-03-16 | ||
| CN202011279917 | 2020-11-16 | ||
| CN202011279917.1 | 2020-11-16 | ||
| PCT/CN2021/081126 WO2021185256A1 (zh) | 2020-03-16 | 2021-03-16 | 取代的嘧啶或吡啶胺衍生物、其组合物及医药上的用途 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023518774A JP2023518774A (ja) | 2023-05-08 |
| JP2023518774A5 true JP2023518774A5 (https=) | 2024-06-24 |
| JP7654008B2 JP7654008B2 (ja) | 2025-03-31 |
Family
ID=77770127
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022556468A Active JP7654008B2 (ja) | 2020-03-16 | 2021-03-16 | 置換ピリミジンまたはピリジルアミン誘導体、その組成物及び医薬的使用 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20230145793A1 (https=) |
| EP (1) | EP4122927A4 (https=) |
| JP (1) | JP7654008B2 (https=) |
| KR (1) | KR20220147124A (https=) |
| CN (2) | CN118373808A (https=) |
| AU (1) | AU2021239135B2 (https=) |
| CA (1) | CA3171774C (https=) |
| WO (1) | WO2021185256A1 (https=) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2022007376A (es) | 2019-12-20 | 2022-09-02 | Tenaya Therapeutics Inc | Fluoroalqull-oxadiazoles y sus usos. |
| WO2022166796A1 (zh) * | 2021-02-05 | 2022-08-11 | 上海齐鲁制药研究中心有限公司 | 嘧啶或吡啶并杂环类腺苷受体抑制剂及其制备方法和用途 |
| US20240252502A1 (en) | 2021-05-04 | 2024-08-01 | Tenaya Therapeutics, Inc. | Hdac6 inhibitors for treatment of metabolic disease and hfpef |
| EP4337202A4 (en) | 2021-06-18 | 2025-04-02 | Aligos Therapeutics, Inc. | METHODS AND COMPOSITIONS FOR TARGETING PD-L1 |
| WO2023040876A1 (zh) * | 2021-09-15 | 2023-03-23 | 上海海雁医药科技有限公司 | 氮杂芳环类化合物及其药学上可接受的盐的多晶型物、药物组合物和应用 |
| AU2022347682B2 (en) * | 2021-09-15 | 2025-08-28 | Shanghai Haiyan Pharmaceutical Technology Co., Ltd. | Polymorph and application of pyrimidine derivative and pharmaceutically acceptable salt thereof |
| CN116063292A (zh) * | 2021-10-29 | 2023-05-05 | 山东晶源生物医药有限公司 | 一种含氮化合物、其中间体、其组合物、其制备方法及其应用 |
| EP4448512A4 (en) | 2021-12-16 | 2025-11-19 | Aligos Therapeutics Inc | METHODS AND COMPOSITIONS FOR TARGETING PD-L1 |
| JP2025512384A (ja) | 2022-04-13 | 2025-04-17 | ギリアード サイエンシーズ, インコーポレイテッド | Trop-2発現がんを治療するための併用療法 |
| JP2024005443A (ja) * | 2022-06-30 | 2024-01-17 | ユニマテック株式会社 | 塩素化された含フッ素ピリミジン化合物の製造方法 |
| JP2024005442A (ja) * | 2022-06-30 | 2024-01-17 | ユニマテック株式会社 | 塩素化された含フッ素ピリミジン化合物の製造方法 |
| WO2025137640A1 (en) | 2023-12-22 | 2025-06-26 | Gilead Sciences, Inc. | Azaspiro wrn inhibitors |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI330183B (https=) * | 2001-10-22 | 2010-09-11 | Eisai R&D Man Co Ltd | |
| JP2005298449A (ja) * | 2004-04-15 | 2005-10-27 | Astellas Pharma Inc | 4−アミノピリミジン誘導体 |
| AR070127A1 (es) * | 2008-01-11 | 2010-03-17 | Novartis Ag | Pirrolo - pirimidinas y pirrolo -piridinas |
| ES2365960B1 (es) * | 2010-03-31 | 2012-06-04 | Palobiofarma, S.L | Nuevos antagonistas de los receptores de adenosina. |
| WO2013124246A1 (de) * | 2012-02-22 | 2013-08-29 | Bayer Intellectual Property Gmbh | Herbizid wirksame 4-dialkoxymethyl-2-phenylpyrimidine |
| WO2015091531A1 (en) * | 2013-12-19 | 2015-06-25 | Almirall, S.A. | Imidazolopyrimidin-2-yl derivatives as jak inhibitors |
| WO2017088755A1 (en) * | 2015-11-23 | 2017-06-01 | Suzhou Yunxuan Yiyao Keji Youxian Gongsi | Aminopyrimidine heterocyclic compound with adenosine receptor antagonistic activity |
| HUE064141T2 (hu) * | 2017-01-20 | 2024-02-28 | Arcus Biosciences Inc | Azolopirimidin rákkal összefüggõ rendellenességek kezelésére |
| CN109651358B (zh) * | 2017-10-11 | 2023-04-07 | 上海迪诺医药科技有限公司 | 4-氨基吡啶衍生物、其药物组合物、制备方法及应用 |
-
2021
- 2021-03-16 JP JP2022556468A patent/JP7654008B2/ja active Active
- 2021-03-16 EP EP21770539.1A patent/EP4122927A4/en active Pending
- 2021-03-16 CN CN202410486071.0A patent/CN118373808A/zh active Pending
- 2021-03-16 WO PCT/CN2021/081126 patent/WO2021185256A1/zh not_active Ceased
- 2021-03-16 AU AU2021239135A patent/AU2021239135B2/en active Active
- 2021-03-16 US US17/911,192 patent/US20230145793A1/en active Pending
- 2021-03-16 KR KR1020227033700A patent/KR20220147124A/ko active Pending
- 2021-03-16 CN CN202180001773.XA patent/CN113748110B/zh active Active
- 2021-03-16 CA CA3171774A patent/CA3171774C/en active Active
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