JP2023518543A5 - - Google Patents

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Publication number
JP2023518543A5
JP2023518543A5 JP2022556248A JP2022556248A JP2023518543A5 JP 2023518543 A5 JP2023518543 A5 JP 2023518543A5 JP 2022556248 A JP2022556248 A JP 2022556248A JP 2022556248 A JP2022556248 A JP 2022556248A JP 2023518543 A5 JP2023518543 A5 JP 2023518543A5
Authority
JP
Japan
Prior art keywords
alkyl
group
optionally substituted
halogen
independently
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022556248A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023518543A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/023228 external-priority patent/WO2021188944A1/en
Publication of JP2023518543A publication Critical patent/JP2023518543A/ja
Publication of JP2023518543A5 publication Critical patent/JP2023518543A5/ja
Pending legal-status Critical Current

Links

JP2022556248A 2020-03-20 2021-03-19 Phd阻害剤化合物、組成物、及びそれらの使用 Pending JP2023518543A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062992616P 2020-03-20 2020-03-20
US62/992,616 2020-03-20
PCT/US2021/023228 WO2021188944A1 (en) 2020-03-20 2021-03-19 Phd inhibitor compounds, compositions, and their use

Publications (2)

Publication Number Publication Date
JP2023518543A JP2023518543A (ja) 2023-05-02
JP2023518543A5 true JP2023518543A5 (https=) 2024-05-29

Family

ID=75478265

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022556248A Pending JP2023518543A (ja) 2020-03-20 2021-03-19 Phd阻害剤化合物、組成物、及びそれらの使用

Country Status (6)

Country Link
US (1) US20230212138A1 (https=)
EP (1) EP4121424A1 (https=)
JP (1) JP2023518543A (https=)
CN (2) CN120004851A (https=)
AR (1) AR121626A1 (https=)
WO (1) WO2021188944A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11713298B2 (en) 2018-05-09 2023-08-01 Akebia Therapeutics, Inc. Process for preparing 2-[[5-(3-chlorophenyl)-3-hydroxypyridine-2-carbonyl]amino]acetic acid
WO2021117767A1 (ja) 2019-12-10 2021-06-17 田辺三菱製薬株式会社 含窒素ヘテロアリールカルボキサミド酢酸誘導体の製造方法
EP4447963A1 (en) * 2021-12-17 2024-10-23 Akebia Therapeutics Inc. Selective phd1 inhibitor compounds, compositions, and methods of use
CN118745146B (zh) * 2024-06-24 2025-09-23 上海坦泰生物科技有限公司 一种5-氟-2-肼基吡啶二盐酸盐的制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4663327A (en) * 1984-05-23 1987-05-05 Bayer Aktiengesellschaft 1-heteroaryl-4-aryl-pyrazolin-5-ones
DE3443308A1 (de) * 1984-11-28 1986-05-28 Bayer Ag, 5090 Leverkusen 1-heteroaryl-4-aryl-pyrazolin-5-one zur verwendung als arzneimittel
DE102005019712A1 (de) * 2005-04-28 2006-11-09 Bayer Healthcare Ag Dipyridyl-dihydropyrazolone und ihre Verwendung
DE102006050516A1 (de) * 2006-10-26 2008-04-30 Bayer Healthcare Ag Substituierte Dihydropyrazolone und ihre Verwendung
DE102006050512A1 (de) * 2006-10-26 2008-04-30 Bayer Healthcare Ag Substituierte heterocyclische Verbindungen und ihre Verwendung
DE102006050515A1 (de) * 2006-10-26 2008-04-30 Bayer Healthcare Ag Substituierte Dipyridiyl-dihydropyrazolone und ihre Verwendung
DE102007044032A1 (de) * 2007-09-14 2009-03-19 Bayer Healthcare Ag Substituierte heterocyclische Verbindungen und ihre Verwendung
WO2010005851A1 (en) * 2008-07-08 2010-01-14 Xenon Pharmaceuticals Inc. Combination therapy for treating iron disorders
CA2894399A1 (en) * 2012-12-06 2014-06-12 Quanticel Pharmaceuticals, Inc. Histone demethylase inhibitors
EA031647B1 (ru) * 2013-03-29 2019-02-28 Такеда Фармасьютикал Компани Лимитед 6-(5-гидрокси-1h-пиразол-1-ил)никотинамидные ингибиторы phd

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