JP2023513731A5 - - Google Patents

Info

Publication number
JP2023513731A5
JP2023513731A5 JP2022548818A JP2022548818A JP2023513731A5 JP 2023513731 A5 JP2023513731 A5 JP 2023513731A5 JP 2022548818 A JP2022548818 A JP 2022548818A JP 2022548818 A JP2022548818 A JP 2022548818A JP 2023513731 A5 JP2023513731 A5 JP 2023513731A5
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022548818A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023513731A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/018137 external-priority patent/WO2021163676A1/en
Publication of JP2023513731A publication Critical patent/JP2023513731A/ja
Publication of JP2023513731A5 publication Critical patent/JP2023513731A5/ja
Pending legal-status Critical Current

Links

JP2022548818A 2020-02-16 2021-02-16 キラルベンゾジアゼピノン誘導体の調製方法 Pending JP2023513731A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062977316P 2020-02-16 2020-02-16
US62/977,316 2020-02-16
PCT/US2021/018137 WO2021163676A1 (en) 2020-02-16 2021-02-16 Methods of preparing chiral benzodiazepinone derivatives

Publications (2)

Publication Number Publication Date
JP2023513731A JP2023513731A (ja) 2023-04-03
JP2023513731A5 true JP2023513731A5 (https=) 2024-02-22

Family

ID=77291712

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022548818A Pending JP2023513731A (ja) 2020-02-16 2021-02-16 キラルベンゾジアゼピノン誘導体の調製方法

Country Status (11)

Country Link
US (2) US12503449B2 (https=)
EP (1) EP4107148A4 (https=)
JP (1) JP2023513731A (https=)
KR (1) KR20220143094A (https=)
CN (1) CN115103836A (https=)
AU (1) AU2021218456A1 (https=)
BR (1) BR112022016249A2 (https=)
CA (1) CA3171651A1 (https=)
IL (1) IL295572A (https=)
MX (1) MX2022010079A (https=)
WO (1) WO2021163676A1 (https=)

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0253571B1 (en) * 1986-07-14 1989-08-23 Merck & Co. Inc. Process for resolution and race mization of amines with acidic alpha-hydrogens
NL9000386A (nl) * 1990-02-16 1991-09-16 Stamicarbon Werkwijze voor de bereiding van optisch aktief aminozuuramide.
JPH0751555B2 (ja) 1992-04-15 1995-06-05 キヤノン株式会社 ジイモニウム塩化合物
BRPI0520554A2 (pt) * 2005-09-19 2009-06-13 Arrow Therapeutics Ltd uso de uma benzodiazepina ou um sal farmaceuticamente aceitável do mesmo, método para tratar ou prevenir uma infecção por hcv em um paciente, derivado de benzodiazepina ou um sal famaceuticamente aceitável do mesmo, e, composição farmacêutica
WO2010073253A1 (en) 2008-12-22 2010-07-01 Natco Pharma Limited Method for preparing an optically active frovatriptan
WO2013148554A1 (en) * 2012-03-30 2013-10-03 Merck Sharp & Dohme Corp. Process for preparing fluoroleucine alkyl esters
CN105308030A (zh) * 2012-09-21 2016-02-03 百时美施贵宝公司 烷基、氟烷基-1,4-苯并二氮杂*酮化合物
EP2897942B1 (en) 2012-09-21 2016-08-31 Bristol-Myers Squibb Company Fluoroalkyl and fluorocycloalkyl 1,4-benzodiazepinone compounds as notch inhibitors
WO2014047392A1 (en) 2012-09-21 2014-03-27 Bristol-Myers Squibb Company Fluoroalkyl-1,4-benzodiazepinone compounds
TWI614238B (zh) * 2012-09-21 2018-02-11 必治妥美雅史谷比公司 雙(氟烷基)-1,4-苯并二氮呯酮化合物及其前藥
JP6687596B2 (ja) 2015-02-17 2020-04-22 アモーレパシフィック コーポレーションAmorepacific Corporation N−[4−(1−アミノエチル)−フェニル]−スルホンアミド誘導体のキラル分割方法
CN105439939B (zh) 2015-11-12 2018-12-04 四川恒康科技发展有限公司 一种(S)-N-Boc-3-羟基哌啶的合成方法

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