JP2023510971A5 - - Google Patents
Info
- Publication number
- JP2023510971A5 JP2023510971A5 JP2022544123A JP2022544123A JP2023510971A5 JP 2023510971 A5 JP2023510971 A5 JP 2023510971A5 JP 2022544123 A JP2022544123 A JP 2022544123A JP 2022544123 A JP2022544123 A JP 2022544123A JP 2023510971 A5 JP2023510971 A5 JP 2023510971A5
- Authority
- JP
- Japan
- Prior art keywords
- carbonyl
- carboxamide
- methylimidazole
- chloro
- phenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN2020073830 | 2020-01-22 | ||
| CNPCT/CN2020/073830 | 2020-01-22 | ||
| PCT/EP2021/051095 WO2021148420A1 (en) | 2020-01-22 | 2021-01-20 | Novel heterocyclic compounds |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023510971A JP2023510971A (ja) | 2023-03-15 |
| JP2023510971A5 true JP2023510971A5 (https=) | 2024-01-22 |
| JP7715715B2 JP7715715B2 (ja) | 2025-07-30 |
Family
ID=74418400
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022544123A Active JP7715715B2 (ja) | 2020-01-22 | 2021-01-20 | 新規複素環式化合物 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20220396565A1 (https=) |
| EP (1) | EP4093734A1 (https=) |
| JP (1) | JP7715715B2 (https=) |
| CN (1) | CN114981259B (https=) |
| WO (1) | WO2021148420A1 (https=) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP4211116B1 (en) * | 2020-09-07 | 2024-08-07 | F. Hoffmann-La Roche AG | Novel heterocyclic antibiotics |
| JP2024506021A (ja) * | 2021-02-07 | 2024-02-08 | エフ. ホフマン-ラ ロシュ アーゲー | 新規ヘテロアリール置換イミダゾール誘導体 |
| CN117715892A (zh) * | 2021-07-06 | 2024-03-15 | 豪夫迈·罗氏有限公司 | 用于治疗细菌感染的季铵阳离子取代化合物 |
| JP2024525793A (ja) * | 2021-07-15 | 2024-07-12 | エフ. ホフマン-ラ ロシュ アーゲー | イミダゾール誘導体及びその抗生物質としての使用 |
| JP2025508473A (ja) * | 2022-02-25 | 2025-03-26 | エフ. ホフマン-ラ ロシュ アーゲー | 両性イオン性抗菌化合物 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6849660B1 (en) * | 2000-08-01 | 2005-02-01 | Isis Pharmaceuticals, Inc. | Antimicrobial biaryl compounds |
| GB201406956D0 (en) * | 2014-04-17 | 2014-06-04 | Univ Nottingham | Compounds |
| AU2016347456B2 (en) | 2015-10-27 | 2018-12-13 | F. Hoffmann-La Roche Ag | Peptide macrocycles against acinetobacter baumannii |
| CA3068305A1 (en) * | 2017-06-29 | 2019-01-03 | Rigel Pharmaceuticals, Inc. | Kinase inhibitors and methods for making and using |
| US10471045B2 (en) * | 2017-07-21 | 2019-11-12 | The University Of Hong Kong | Compounds and methods for the treatment of microbial infections |
| US11505573B2 (en) | 2018-03-28 | 2022-11-22 | Hoffmann-La Roche Inc. | Peptide macrocycles against Acinetobacter baumannii |
| US11819532B2 (en) | 2018-04-23 | 2023-11-21 | Hoffmann-La Roche Inc. | Peptide macrocycles against Acinetobacter baumannii |
| CN113164771A (zh) * | 2018-12-17 | 2021-07-23 | 豪夫迈·罗氏有限公司 | 咪唑并吡嗪衍生物作为抗菌剂 |
| WO2020182648A1 (en) * | 2019-03-08 | 2020-09-17 | F. Hoffmann-La Roche Ag | Novel imidazole-pyrazole derivatives |
-
2021
- 2021-01-20 CN CN202180010360.8A patent/CN114981259B/zh active Active
- 2021-01-20 JP JP2022544123A patent/JP7715715B2/ja active Active
- 2021-01-20 EP EP21702384.5A patent/EP4093734A1/en active Pending
- 2021-01-20 WO PCT/EP2021/051095 patent/WO2021148420A1/en not_active Ceased
-
2022
- 2022-07-20 US US17/869,755 patent/US20220396565A1/en active Pending
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