JP2022548690A5 - - Google Patents

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Publication number
JP2022548690A5
JP2022548690A5 JP2022517374A JP2022517374A JP2022548690A5 JP 2022548690 A5 JP2022548690 A5 JP 2022548690A5 JP 2022517374 A JP2022517374 A JP 2022517374A JP 2022517374 A JP2022517374 A JP 2022517374A JP 2022548690 A5 JP2022548690 A5 JP 2022548690A5
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JP
Japan
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JP2022517374A
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Japanese (ja)
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JP2022548690A (ja
JPWO2021055744A5 (https=
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Priority claimed from PCT/US2020/051486 external-priority patent/WO2021055744A1/en
Publication of JP2022548690A publication Critical patent/JP2022548690A/ja
Publication of JP2022548690A5 publication Critical patent/JP2022548690A5/ja
Publication of JPWO2021055744A5 publication Critical patent/JPWO2021055744A5/ja
Priority to JP2024193094A priority Critical patent/JP7781244B2/ja
Ceased legal-status Critical Current

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JP2022517374A 2019-09-20 2020-09-18 Parg阻害剤としての4-置換インドールおよびインダゾールスルホンアミド誘導体 Ceased JP2022548690A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024193094A JP7781244B2 (ja) 2019-09-20 2024-11-01 Parg阻害剤としての4-置換インドールおよびインダゾールスルホンアミド誘導体

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962903438P 2019-09-20 2019-09-20
US62/903,438 2019-09-20
PCT/US2020/051486 WO2021055744A1 (en) 2019-09-20 2020-09-18 4-substituted indole and indazole sulfonamido derivatives as parg inhibitors

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024193094A Division JP7781244B2 (ja) 2019-09-20 2024-11-01 Parg阻害剤としての4-置換インドールおよびインダゾールスルホンアミド誘導体

Publications (3)

Publication Number Publication Date
JP2022548690A JP2022548690A (ja) 2022-11-21
JP2022548690A5 true JP2022548690A5 (https=) 2023-09-20
JPWO2021055744A5 JPWO2021055744A5 (https=) 2023-09-20

Family

ID=72744866

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022517374A Ceased JP2022548690A (ja) 2019-09-20 2020-09-18 Parg阻害剤としての4-置換インドールおよびインダゾールスルホンアミド誘導体
JP2024193094A Active JP7781244B2 (ja) 2019-09-20 2024-11-01 Parg阻害剤としての4-置換インドールおよびインダゾールスルホンアミド誘導体

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JP2024193094A Active JP7781244B2 (ja) 2019-09-20 2024-11-01 Parg阻害剤としての4-置換インドールおよびインダゾールスルホンアミド誘導体

Country Status (12)

Country Link
US (1) US20220389003A1 (https=)
EP (1) EP4031249A1 (https=)
JP (2) JP2022548690A (https=)
KR (1) KR20220066922A (https=)
CN (1) CN114555593A (https=)
AU (1) AU2020348489A1 (https=)
BR (1) BR112022004624A2 (https=)
CA (1) CA3147493A1 (https=)
IL (1) IL291436A (https=)
MX (1) MX2022003276A (https=)
TW (1) TWI873187B (https=)
WO (1) WO2021055744A1 (https=)

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WO2024173514A1 (en) * 2023-02-14 2024-08-22 Ideaya Biosciences, Inc. Amide and ester-substituted imidazopyridine compounds
WO2024173524A1 (en) * 2023-02-14 2024-08-22 Ideaya Biosciences, Inc. Heteroaryl-substituted benzimidazole compounds
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WO2024209035A1 (en) 2023-04-05 2024-10-10 Forx Therapeutics Ag Parg inhibitory compounds
WO2024211506A1 (en) 2023-04-05 2024-10-10 Ideaya Biosciences, Inc. Combination therapy comprising a parg inhibitor and a topoisomerase inhibitor for treating cancer
TWI908044B (zh) * 2023-04-27 2025-12-11 大陸商北京丹擎醫藥科技有限公司 三環雜環衍生物及其組合物及其用途
CN119143747A (zh) * 2023-06-16 2024-12-17 上海璎黎药业有限公司 一种杂芳环结构化合物、其药物组合物及应用
WO2025046148A1 (en) 2023-09-01 2025-03-06 Forx Therapeutics Ag Novel parg inhibitors
TW202528308A (zh) * 2023-09-20 2025-07-16 美商愛德亞生物科學公司 Parg抑制劑
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WO2025072544A1 (en) * 2023-09-27 2025-04-03 Ideaya Biosciences, Inc. Sulfonamino indazole compounds as inhibitors of parg
CN119708015A (zh) * 2023-09-28 2025-03-28 杭州圣域生物医药科技有限公司 杂芳基化合物、其中间体、制备方法和应用
CN121889393A (zh) 2023-10-03 2026-04-17 福克斯治疗股份公司 Parg抑制化合物
CN119859145A (zh) * 2023-10-20 2025-04-22 上海璎黎药业有限公司 一种杂芳环磺酰胺结构化合物、其药物组合物及应用
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WO2025108225A1 (zh) * 2023-11-20 2025-05-30 上海复星医药(集团)股份有限公司 作为parg抑制剂的含氮三环衍生物
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WO2025133191A1 (en) * 2023-12-22 2025-06-26 Genecode Novel sulfonamides or sulfones and their use as neuroprotective and/or neurorestorative agents
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CN118459452B (zh) * 2024-07-10 2024-10-25 苏州国匡医药科技有限公司 一种多聚adp核糖水解酶抑制剂及其应用
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WO2026026739A1 (zh) * 2024-07-29 2026-02-05 海思科医药集团股份有限公司 一种磺酰胺化合物及其在医药上的应用
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