JP2023510746A5 - - Google Patents

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Publication number
JP2023510746A5
JP2023510746A5 JP2022541815A JP2022541815A JP2023510746A5 JP 2023510746 A5 JP2023510746 A5 JP 2023510746A5 JP 2022541815 A JP2022541815 A JP 2022541815A JP 2022541815 A JP2022541815 A JP 2022541815A JP 2023510746 A5 JP2023510746 A5 JP 2023510746A5
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JP
Japan
Application number
JP2022541815A
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Japanese (ja)
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JPWO2021142247A5 (https=
JP2023510746A (ja
JP7706456B2 (ja
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Priority claimed from PCT/US2021/012683 external-priority patent/WO2021142247A1/en
Publication of JP2023510746A publication Critical patent/JP2023510746A/ja
Publication of JPWO2021142247A5 publication Critical patent/JPWO2021142247A5/ja
Publication of JP2023510746A5 publication Critical patent/JP2023510746A5/ja
Application granted granted Critical
Publication of JP7706456B2 publication Critical patent/JP7706456B2/ja
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JP2022541815A 2020-01-10 2021-01-08 Smarca2-vhl分解剤 Active JP7706456B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062959502P 2020-01-10 2020-01-10
US62/959,502 2020-01-10
PCT/US2021/012683 WO2021142247A1 (en) 2020-01-10 2021-01-08 Smarca2-vhl degraders

Publications (4)

Publication Number Publication Date
JP2023510746A JP2023510746A (ja) 2023-03-15
JPWO2021142247A5 JPWO2021142247A5 (https=) 2024-01-16
JP2023510746A5 true JP2023510746A5 (https=) 2024-01-16
JP7706456B2 JP7706456B2 (ja) 2025-07-11

Family

ID=74495106

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022541815A Active JP7706456B2 (ja) 2020-01-10 2021-01-08 Smarca2-vhl分解剤

Country Status (7)

Country Link
US (1) US20230091042A1 (https=)
EP (1) EP4087658A1 (https=)
JP (1) JP7706456B2 (https=)
AU (1) AU2021205326A1 (https=)
CA (1) CA3167166A1 (https=)
MX (1) MX2022008487A (https=)
WO (1) WO2021142247A1 (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2019140380A1 (en) 2018-01-12 2019-07-18 Kymera Therapeutics, Inc. Protein degraders and uses thereof
WO2020010227A1 (en) 2018-07-06 2020-01-09 Kymera Therapeutics, Inc. Protein degraders and uses thereof
WO2020251972A1 (en) 2019-06-10 2020-12-17 Kymera Therapeutics, Inc. Smarca degraders and uses thereof
WO2021133917A1 (en) 2019-12-23 2021-07-01 Kymera Therapeutics, Inc. Smarca inhibitors and uses thereof
BR112022012410A2 (pt) 2019-12-23 2022-08-30 Kymera Therapeutics Inc Degradadores smarca e usos dos mesmos
WO2022029617A1 (en) * 2020-08-04 2022-02-10 Aurigene Discovery Technologies Limited 6-substituted pyridazine compounds as smarca2 and/or smarca4 degraders
EP4259144A4 (en) * 2020-12-09 2025-08-20 Kymera Therapeutics Inc SMARCA DEGRADING AGENTS AND THEIR USES
US11993599B2 (en) 2021-08-09 2024-05-28 Genentech, Inc. Therapeutic compounds

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10519152B2 (en) * 2017-12-21 2019-12-31 Astrazeneca Ab Compounds and their use in treating cancer
US20190300521A1 (en) * 2018-04-01 2019-10-03 Arvinas Operations, Inc. Brm targeting compounds and associated methods of use
US12371426B2 (en) * 2018-04-26 2025-07-29 Aurigene Discovery Technologies Limited Pyridazine derivatives as SMARCA2/4 degraders
WO2019213005A1 (en) * 2018-04-30 2019-11-07 Dana-Farber Cancer Institute, Inc. Small molecule degraders of polybromo-1 (pbrm1)

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