JP2023159197A5 - - Google Patents

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JP2023159197A5
JP2023159197A5 JP2023129305A JP2023129305A JP2023159197A5 JP 2023159197 A5 JP2023159197 A5 JP 2023159197A5 JP 2023129305 A JP2023129305 A JP 2023129305A JP 2023129305 A JP2023129305 A JP 2023129305A JP 2023159197 A5 JP2023159197 A5 JP 2023159197A5
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JP7651203B2 (ja
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JP2023129305A 2018-04-20 2023-08-08 ボロン酸誘導体およびその治療的使用 Active JP7651203B2 (ja)

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JP2025035562A JP2025083398A (ja) 2018-04-20 2025-03-06 ボロン酸誘導体およびその治療的使用

Applications Claiming Priority (4)

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US201862660729P 2018-04-20 2018-04-20
US62/660,729 2018-04-20
PCT/US2019/027844 WO2019204419A1 (en) 2018-04-20 2019-04-17 Boronic acid derivatives and therapeutic uses thereof
JP2020557178A JP7329260B2 (ja) 2018-04-20 2019-04-17 ボロン酸誘導体およびその治療的使用

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JP2023159197A JP2023159197A (ja) 2023-10-31
JP2023159197A5 true JP2023159197A5 (https=) 2023-11-24
JP7651203B2 JP7651203B2 (ja) 2025-03-26

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JP2020557178A Active JP7329260B2 (ja) 2018-04-20 2019-04-17 ボロン酸誘導体およびその治療的使用
JP2023129305A Active JP7651203B2 (ja) 2018-04-20 2023-08-08 ボロン酸誘導体およびその治療的使用
JP2025035562A Pending JP2025083398A (ja) 2018-04-20 2025-03-06 ボロン酸誘導体およびその治療的使用

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US (2) US12016868B2 (https=)
EP (1) EP3781576B1 (https=)
JP (3) JP7329260B2 (https=)
CN (1) CN112424209A (https=)
AU (1) AU2019256351B2 (https=)
CA (1) CA3097127A1 (https=)
TW (1) TW201945005A (https=)
WO (1) WO2019204419A1 (https=)
ZA (1) ZA202006377B (https=)

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CN113880871B (zh) * 2020-10-16 2022-08-23 中国科学院兰州化学物理研究所 一种饱和单硼类化合物的制备方法
CN117377470A (zh) 2021-03-08 2024-01-09 伊莱利利公司 美维达林和其他d1正向别构调节剂在幻觉和痴呆相关精神病的治疗中的用途
EP4304577A1 (en) 2021-03-09 2024-01-17 Eli Lilly And Co. Use of mevidalen and other d1 positive allosteric modulators for slowing of parkinson's disease progression
TW202404610A (zh) * 2022-06-24 2024-02-01 大陸商瑞石生物醫藥有限公司 一種硼酸酯衍生物的結晶、其製備方法及用途
US20250099495A1 (en) * 2023-09-22 2025-03-27 City University Of Hong Kong Methods of inhibiting klebsiella pneumoniae carbapenemase-2
WO2025119216A1 (zh) * 2023-12-04 2025-06-12 珠海联邦制药股份有限公司 硼酸类β-内酰胺酶抑制剂及其制备方法和应用
CN119119096B (zh) * 2024-09-09 2025-09-16 郑州药领医药科技有限公司 一种4-((4,4,5,5-四甲基-1,3,2-二氧硼杂环戊烷-2-基)甲基)哌啶-1-甲酸叔丁酯的合成方法

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