JP2022524151A5 - - Google Patents

Info

Publication number
JP2022524151A5
JP2022524151A5 JP2021553777A JP2021553777A JP2022524151A5 JP 2022524151 A5 JP2022524151 A5 JP 2022524151A5 JP 2021553777 A JP2021553777 A JP 2021553777A JP 2021553777 A JP2021553777 A JP 2021553777A JP 2022524151 A5 JP2022524151 A5 JP 2022524151A5
Authority
JP
Japan
Prior art keywords
optionally substituted
alkyl
heterocycloalkyl
cycloalkyl
heteroaryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021553777A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022524151A (ja
JP7670618B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/022272 external-priority patent/WO2020185999A1/en
Publication of JP2022524151A publication Critical patent/JP2022524151A/ja
Publication of JP2022524151A5 publication Critical patent/JP2022524151A5/ja
Priority to JP2024203544A priority Critical patent/JP2025037920A/ja
Application granted granted Critical
Publication of JP7670618B2 publication Critical patent/JP7670618B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2021553777A 2019-03-14 2020-03-12 環状ペプチド抗生物質 Active JP7670618B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024203544A JP2025037920A (ja) 2019-03-14 2024-11-21 環状ペプチド抗生物質

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN2019078189 2019-03-14
CNPCT/CN2019/078189 2019-03-14
PCT/US2020/022272 WO2020185999A1 (en) 2019-03-14 2020-03-12 Cyclic peptide antibiotics

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024203544A Division JP2025037920A (ja) 2019-03-14 2024-11-21 環状ペプチド抗生物質

Publications (3)

Publication Number Publication Date
JP2022524151A JP2022524151A (ja) 2022-04-27
JP2022524151A5 true JP2022524151A5 (https=) 2023-03-22
JP7670618B2 JP7670618B2 (ja) 2025-04-30

Family

ID=70190176

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021553777A Active JP7670618B2 (ja) 2019-03-14 2020-03-12 環状ペプチド抗生物質
JP2024203544A Pending JP2025037920A (ja) 2019-03-14 2024-11-21 環状ペプチド抗生物質

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2024203544A Pending JP2025037920A (ja) 2019-03-14 2024-11-21 環状ペプチド抗生物質

Country Status (5)

Country Link
US (1) US12358951B2 (https=)
EP (1) EP3938377A1 (https=)
JP (2) JP7670618B2 (https=)
CN (1) CN113710687A (https=)
WO (1) WO2020185999A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7670618B2 (ja) * 2019-03-14 2025-04-30 エフ・ホフマン-ラ・ロシュ・アクチェンゲゼルシャフト 環状ペプチド抗生物質
WO2022009212A1 (en) * 2020-07-09 2022-01-13 Technion Research And Development Foundation Ltd. TYROSINE, TRYPTOPHAN AND PHENYLALANINE AS mTOR AGONISTS MEDIATING PROTEASOME DYNAMICS, COMPOSITIONS, METHODS AND USES THEREOF IN THERAPY, AND PROGNOSTIC METHODS FOR DRUG-RESISTANCE
CN118307583A (zh) * 2024-04-03 2024-07-09 上海科技大学 β氨基酯、聚β氨基酯化合物及其制备方法及应用

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS594990B2 (ja) 1977-05-13 1984-02-02 三共株式会社 抗生物質グロボマイシン
JPS5547644A (en) 1978-10-02 1980-04-04 Meiji Seika Kaisha Ltd New antibiotics sf-1902 a2, a3, a4 and a5 and their preparation
US5384309A (en) 1989-07-17 1995-01-24 Genentech, Inc. Cyclized peptides and their use as platelet aggregation inhibitors
US10787490B2 (en) 2015-07-15 2020-09-29 Protaganist Therapeutics, Inc. Peptide inhibitors of interleukin-23 receptor and their use to treat inflammatory diseases
US11072616B2 (en) 2015-11-11 2021-07-27 Universite De Montreal Cyclic peptides targeting alpha-4-beta-7 integrin
JP2020533374A (ja) 2017-09-15 2020-11-19 エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft 環状ペプチド抗生物質
JP7670618B2 (ja) * 2019-03-14 2025-04-30 エフ・ホフマン-ラ・ロシュ・アクチェンゲゼルシャフト 環状ペプチド抗生物質

Similar Documents

Publication Publication Date Title
RU2013104951A (ru) Циклические бороновые кислотно-эфирные производные и их использование в терапии
JP2023159197A5 (https=)
JP2022524151A5 (https=)
JP2022137011A5 (https=)
JP2021522167A5 (https=)
RU2016146581A (ru) Макроциклические антибиотики широкого спектра действия
JP2019527196A5 (https=)
CA2504448A1 (en) Transcription factor modulating compounds and methods of use thereof
FI3986419T3 (fi) Boorihappojohdannaisia ja niiden terapeuttisia käyttöjä
JP2017517567A5 (https=)
JP2023518418A5 (https=)
JP2016501864A5 (https=)
RU2018122505A (ru) Макроциклические антибиотики широкого спектра действия
RU2016107436A (ru) Линейные пептидные антибиотики
ES2985626T3 (es) Sales y polimorfos de derivados cíclicos de éster de ácido borónico y usos terapéuticos de los mismos
RU2686740C2 (ru) Ингибиторы бета-лактамазы
SI2344129T1 (en) AEROSOL FLUOROKINOLONAL FORMULATIONS FOR IMPROVED PHARMACOKINETICS
JP2016528257A5 (https=)
RU2018122498A (ru) Макроциклические антибиотики широкого спектра действия
JP2020510044A5 (https=)
RU2012111458A (ru) Применение левофлоксацина в форме аэрозоля для лечения муковисцидоза
JP2020507564A5 (https=)
WO2011101710A1 (en) Efflux pump inhibitors
CN113015532B (zh) 包含β-内酰胺酶抑制剂的组合式组合物
JP2009541332A5 (https=)