JP2022547558A5 - - Google Patents
Info
- Publication number
- JP2022547558A5 JP2022547558A5 JP2022515857A JP2022515857A JP2022547558A5 JP 2022547558 A5 JP2022547558 A5 JP 2022547558A5 JP 2022515857 A JP2022515857 A JP 2022515857A JP 2022515857 A JP2022515857 A JP 2022515857A JP 2022547558 A5 JP2022547558 A5 JP 2022547558A5
- Authority
- JP
- Japan
- Prior art keywords
- item
- approximately
- compound
- aqueous parenteral
- crystal morphology
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2025124956A JP2025137788A (ja) | 2019-09-11 | 2025-07-25 | 抗ウイルスプロドラッグ及びその医薬組成物 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962898679P | 2019-09-11 | 2019-09-11 | |
| US62/898,679 | 2019-09-11 | ||
| PCT/US2020/050511 WO2021050956A1 (en) | 2019-09-11 | 2020-09-11 | Antiviral prodrugs and pharmaceutical compositions thereof |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025124956A Division JP2025137788A (ja) | 2019-09-11 | 2025-07-25 | 抗ウイルスプロドラッグ及びその医薬組成物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022547558A JP2022547558A (ja) | 2022-11-14 |
| JP2022547558A5 true JP2022547558A5 (enExample) | 2024-03-19 |
| JP7719769B2 JP7719769B2 (ja) | 2025-08-06 |
Family
ID=74866690
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022515860A Active JP7703518B2 (ja) | 2019-09-11 | 2020-09-11 | 抗ウイルスプロドラッグ及びその製剤 |
| JP2022515857A Active JP7719769B2 (ja) | 2019-09-11 | 2020-09-11 | 抗ウイルスプロドラッグ及びその医薬組成物 |
| JP2025063311A Pending JP2025096427A (ja) | 2019-09-11 | 2025-04-07 | 抗ウイルスプロドラッグ及びその製剤 |
| JP2025124956A Pending JP2025137788A (ja) | 2019-09-11 | 2025-07-25 | 抗ウイルスプロドラッグ及びその医薬組成物 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022515860A Active JP7703518B2 (ja) | 2019-09-11 | 2020-09-11 | 抗ウイルスプロドラッグ及びその製剤 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025063311A Pending JP2025096427A (ja) | 2019-09-11 | 2025-04-07 | 抗ウイルスプロドラッグ及びその製剤 |
| JP2025124956A Pending JP2025137788A (ja) | 2019-09-11 | 2025-07-25 | 抗ウイルスプロドラッグ及びその医薬組成物 |
Country Status (18)
| Country | Link |
|---|---|
| US (3) | US20220323476A1 (enExample) |
| EP (2) | EP4028019A4 (enExample) |
| JP (4) | JP7703518B2 (enExample) |
| KR (2) | KR20220066303A (enExample) |
| CN (4) | CN114929236B (enExample) |
| AU (2) | AU2020346908B2 (enExample) |
| BR (2) | BR112022004424A2 (enExample) |
| CA (2) | CA3150418A1 (enExample) |
| CL (4) | CL2022000601A1 (enExample) |
| CO (2) | CO2022005128A2 (enExample) |
| CR (2) | CR20220110A (enExample) |
| DO (2) | DOP2022000056A (enExample) |
| IL (4) | IL290861B2 (enExample) |
| MX (4) | MX2022002897A (enExample) |
| PE (2) | PE20221036A1 (enExample) |
| PH (2) | PH12022550528A1 (enExample) |
| UA (1) | UA130229C2 (enExample) |
| WO (2) | WO2021050961A1 (enExample) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2019014247A1 (en) | 2017-07-11 | 2019-01-17 | Gilead Sciences, Inc. | COMPOSITIONS COMPRISING POLYMERASE RNA INHIBITOR AND CYCLODEXTRIN FOR THE TREATMENT OF VIRAL INFECTIONS |
| CA3146679A1 (en) * | 2019-07-27 | 2021-02-04 | Brii Biosciences, Inc. | Adenosine derivative and pharmaceutical composition comprising the same |
| KR20220066303A (ko) * | 2019-09-11 | 2022-05-24 | 더 스크립스 리서치 인스티튜트 | 항바이러스 전구약물 및 이의 약제학적 조성물 |
| JP7703538B2 (ja) * | 2019-12-09 | 2025-07-07 | ヴィーブ、ヘルスケア、カンパニー | カボテグラビルを含んでなる医薬組成物 |
| JP2023512656A (ja) | 2020-01-27 | 2023-03-28 | ギリアード サイエンシーズ, インコーポレイテッド | SARS CoV-2感染を治療するための方法 |
| KR20220153619A (ko) | 2020-03-12 | 2022-11-18 | 길리애드 사이언시즈, 인코포레이티드 | 1'-시아노 뉴클레오사이드의 제조 방법 |
| WO2021188959A1 (en) * | 2020-03-20 | 2021-09-23 | Gilead Sciences, Inc. | Prodrugs of 4'-c-substituted-2-halo-2'-deoxyadenosine nucleosides and methods of making and using the same |
| CA3172483A1 (en) | 2020-04-06 | 2021-10-14 | Scott Ellis | Inhalation formulations of 1'-cyano substituted carbanucleoside analogs |
| TW202203941A (zh) | 2020-05-29 | 2022-02-01 | 美商基利科學股份有限公司 | 瑞德西韋之治療方法 |
| PE20230618A1 (es) | 2020-06-24 | 2023-04-14 | Gilead Sciences Inc | Analogos de nucleosido de 1'-ciano y usos de los mismos |
| IL300453A (en) | 2020-08-27 | 2023-04-01 | Gilead Sciences Inc | COMPOSITIONS AND METHODS FOR THE TREATMENT OF VIRAL INFECTIONS |
| EP4281083A4 (en) | 2021-01-25 | 2025-01-01 | Brii Biosciences, Inc. | COMBINATION THERAPY FOR HIV WITH ADENOSINE DERIVATIVE AND CAPSID INHIBITORS |
| EP4281081A4 (en) | 2021-01-25 | 2025-05-14 | Brii Biosciences, Inc. | ADENOSINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION THEREOF |
| MX2023010797A (es) * | 2021-03-16 | 2023-09-27 | Scripps Research Inst | Profarmacos antivirales de entecavir (etv) y formulaciones de los mismos. |
| KR20240154647A (ko) | 2022-03-02 | 2024-10-25 | 길리애드 사이언시즈, 인코포레이티드 | 바이러스성 감염 치료를 위한 화합물 및 방법 |
| US12357577B1 (en) | 2024-02-02 | 2025-07-15 | Gilead Sciences, Inc. | Pharmaceutical formulations and uses thereof |
| CN121358747A (zh) | 2023-06-27 | 2026-01-16 | 吉利德科学公司 | 核苷逆转录酶易位抑制剂的固体形式 |
| CN121419986A (zh) * | 2023-06-27 | 2026-01-27 | 吉利德科学公司 | 用于制备抗病毒前药的方法和中间体 |
| FI20245041A1 (en) | 2024-01-17 | 2025-07-18 | Metso Finland Oy | Precipitation of calcium compounds in liquid extraction systems |
Family Cites Families (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5283067A (en) | 1987-01-30 | 1994-02-01 | Ciba-Geigy Corporation | Parenteral suspensions |
| US5192749A (en) | 1990-05-21 | 1993-03-09 | Syntex (U.S.A.) Inc. | 4'-substituted nucleosides |
| FR2694693B1 (fr) * | 1992-07-28 | 1994-10-28 | Abrax Bio Labs Sa | Composition pharmaceutique à base de flavopéréirine et son utilisation dans un traitement contre le virus VIH. |
| ATE250622T1 (de) | 1999-05-12 | 2003-10-15 | Yamasa Corp | 4'-c-ethynyl-pyrimidine nukleoside |
| US6576619B2 (en) * | 1999-05-24 | 2003-06-10 | Cv Therapeutics, Inc. | Orally active A1 adenosine receptor agonists |
| US6875751B2 (en) | 2000-06-15 | 2005-04-05 | Idenix Pharmaceuticals, Inc. | 3′-prodrugs of 2′-deoxy-β-L-nucleosides |
| CA2502109C (en) * | 2004-03-24 | 2010-02-23 | Yamasa Corporation | 4'-c-substituted-2-haloadenosine derivative |
| EA200800932A1 (ru) | 2005-09-26 | 2008-10-30 | Фармассет, Инк. | Модифицированные 4`-нуклеозиды в качестве противовирусных агентов |
| CN100532388C (zh) | 2007-07-16 | 2009-08-26 | 郑州大学 | 2’-氟-4’-取代-核苷类似物、其制备方法及应用 |
| US20090274686A1 (en) | 2008-05-02 | 2009-11-05 | Yat Sun Or | Nucleoside phosphonate derivatives |
| NZ593649A (en) | 2008-12-23 | 2013-11-29 | Gilead Pharmasset Llc | Nucleoside analogs |
| WO2013090420A2 (en) | 2011-12-12 | 2013-06-20 | Catabasis Pharmaceuticals, Inc. | Fatty acid antiviral conjugates and their uses |
| WO2015143712A1 (en) | 2014-03-28 | 2015-10-01 | Merck Sharp & Dohme Corp. | 4'-substituted nucleoside reverse transcriptase inhibitors |
| CA3182565A1 (en) | 2015-03-06 | 2016-09-15 | Atea Pharmaceuticals, Inc. | .beta.-d-2'-deoxy-2'-.alpha.-fluoro-2'-.beta.-c-substituted-2-modified-n6-substituted purine nucleotides for hcv treatment |
| MX391226B (es) | 2015-09-23 | 2025-03-21 | Merck Sharp & Dohme Llc | Inhibidores de transcriptasa inversa de nucleosido 4'-substituido y preparaciones de los mismos. |
| US10745428B2 (en) * | 2015-12-10 | 2020-08-18 | Idenix Pharmaceuticals Llc | Antiviral phosphodiamide prodrugs of tenofovir |
| FR3053281B1 (fr) | 2016-06-30 | 2020-03-27 | Banque De France | Procede de fabrication d'un document de securite presentant un signe de securite a contraste de brillance |
| US10185393B2 (en) | 2017-04-03 | 2019-01-22 | Facebook Technologies, Llc | Waveguide display with spatially switchable grating |
| PT3706762T (pt) * | 2017-12-07 | 2024-12-05 | Univ Emory | N4-hidroxicitidina e derivados e utilizações antivirais relacionadas com os mesmos |
| US20190185508A1 (en) | 2017-12-15 | 2019-06-20 | Merck Sharp & Dohme Corp. | Deuterated nucleoside reverse transcriptase inhibitors |
| EP3762396A1 (en) | 2018-03-07 | 2021-01-13 | GlaxoSmithKline Intellectual Property (No.2) Limited | Compounds useful in hiv therapy |
| AU2019317810A1 (en) | 2018-08-09 | 2021-02-25 | Glaxosmithkline Intellectual Property (No.2) Limited | Compounds useful in HIV therapy |
| US11572595B2 (en) * | 2018-12-31 | 2023-02-07 | Roche Molecular Systems, Inc. | Non-replicative transduction particles with one or more non-native tail fibers and transduction particle-based reporter systems |
| CN113811360A (zh) | 2019-03-06 | 2021-12-17 | 葛兰素史密斯克莱知识产权(第2 号)有限公司 | 用于hiv治疗的化合物 |
| CA3146679A1 (en) | 2019-07-27 | 2021-02-04 | Brii Biosciences, Inc. | Adenosine derivative and pharmaceutical composition comprising the same |
| KR20220066303A (ko) | 2019-09-11 | 2022-05-24 | 더 스크립스 리서치 인스티튜트 | 항바이러스 전구약물 및 이의 약제학적 조성물 |
| CN121358747A (zh) | 2023-06-27 | 2026-01-16 | 吉利德科学公司 | 核苷逆转录酶易位抑制剂的固体形式 |
| CN121419986A (zh) | 2023-06-27 | 2026-01-27 | 吉利德科学公司 | 用于制备抗病毒前药的方法和中间体 |
-
2020
- 2020-09-11 KR KR1020227011982A patent/KR20220066303A/ko active Pending
- 2020-09-11 IL IL290861A patent/IL290861B2/en unknown
- 2020-09-11 CR CR20220110A patent/CR20220110A/es unknown
- 2020-09-11 IL IL319709A patent/IL319709A/en unknown
- 2020-09-11 WO PCT/US2020/050519 patent/WO2021050961A1/en not_active Ceased
- 2020-09-11 WO PCT/US2020/050511 patent/WO2021050956A1/en not_active Ceased
- 2020-09-11 CN CN202080075497.7A patent/CN114929236B/zh active Active
- 2020-09-11 BR BR112022004424A patent/BR112022004424A2/pt unknown
- 2020-09-11 CN CN202410626114.0A patent/CN118580291A/zh active Pending
- 2020-09-11 JP JP2022515860A patent/JP7703518B2/ja active Active
- 2020-09-11 AU AU2020346908A patent/AU2020346908B2/en active Active
- 2020-09-11 EP EP20862704.2A patent/EP4028019A4/en active Pending
- 2020-09-11 MX MX2022002897A patent/MX2022002897A/es unknown
- 2020-09-11 EP EP20862707.5A patent/EP4028020A4/en active Pending
- 2020-09-11 PE PE2022000382A patent/PE20221036A1/es unknown
- 2020-09-11 US US17/642,552 patent/US20220323476A1/en not_active Abandoned
- 2020-09-11 CR CR20220109A patent/CR20220109A/es unknown
- 2020-09-11 JP JP2022515857A patent/JP7719769B2/ja active Active
- 2020-09-11 IL IL290919A patent/IL290919B2/en unknown
- 2020-09-11 PH PH1/2022/550528A patent/PH12022550528A1/en unknown
- 2020-09-11 UA UAA202201150A patent/UA130229C2/uk unknown
- 2020-09-11 PE PE2022000389A patent/PE20221037A1/es unknown
- 2020-09-11 AU AU2020346907A patent/AU2020346907A1/en active Pending
- 2020-09-11 IL IL320979A patent/IL320979B1/en unknown
- 2020-09-11 KR KR1020227011981A patent/KR20220066302A/ko active Pending
- 2020-09-11 BR BR112022004417A patent/BR112022004417A2/pt unknown
- 2020-09-11 PH PH1/2022/550527A patent/PH12022550527A1/en unknown
- 2020-09-11 CN CN202411383875.4A patent/CN119462802A/zh active Pending
- 2020-09-11 US US17/642,559 patent/US12569510B2/en active Active
- 2020-09-11 CN CN202080077922.6A patent/CN114793421B/zh active Active
- 2020-09-11 MX MX2022002899A patent/MX2022002899A/es unknown
- 2020-09-11 CA CA3150418A patent/CA3150418A1/en active Pending
- 2020-09-11 CA CA3150467A patent/CA3150467A1/en active Pending
-
2022
- 2022-03-09 MX MX2025011432A patent/MX2025011432A/es unknown
- 2022-03-09 MX MX2025014404A patent/MX2025014404A/es unknown
- 2022-03-10 DO DO2022000056A patent/DOP2022000056A/es unknown
- 2022-03-10 DO DO2022000055A patent/DOP2022000055A/es unknown
- 2022-03-10 CL CL2022000601A patent/CL2022000601A1/es unknown
- 2022-03-10 CL CL2022000587A patent/CL2022000587A1/es unknown
- 2022-04-25 CO CONC2022/0005128A patent/CO2022005128A2/es unknown
- 2022-06-22 CO CONC2022/0004681A patent/CO2022004681A2/es unknown
-
2023
- 2023-08-15 US US18/233,959 patent/US20230390318A1/en not_active Abandoned
-
2024
- 2024-10-23 CL CL2024003241A patent/CL2024003241A1/es unknown
-
2025
- 2025-04-07 JP JP2025063311A patent/JP2025096427A/ja active Pending
- 2025-07-25 JP JP2025124956A patent/JP2025137788A/ja active Pending
- 2025-12-02 CL CL2025003801A patent/CL2025003801A1/es unknown
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