JP2022542072A5 - - Google Patents
Info
- Publication number
- JP2022542072A5 JP2022542072A5 JP2022504198A JP2022504198A JP2022542072A5 JP 2022542072 A5 JP2022542072 A5 JP 2022542072A5 JP 2022504198 A JP2022504198 A JP 2022504198A JP 2022504198 A JP2022504198 A JP 2022504198A JP 2022542072 A5 JP2022542072 A5 JP 2022542072A5
- Authority
- JP
- Japan
- Prior art keywords
- het
- hal
- atoms
- disubstituted
- unsubstituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2024212157A JP7730407B2 (ja) | 2019-07-24 | 2024-12-05 | ４－（イミダゾ［１，２－ａ］ピリジン－３－イル）－ピリミジン誘導体 |
| JP2025135307A JP2025186243A (ja) | 2019-07-24 | 2025-08-15 | ４－（イミダゾ［１，２－ａ］ピリジン－３－イル）－ピリミジン誘導体 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP19188031.9 | 2019-07-24 | ||
| EP19188031 | 2019-07-24 | ||
| PCT/EP2020/070616 WO2021013864A1 (en) | 2019-07-24 | 2020-07-22 | 4-(imidazo[1,2-a]pyridin-3-yl) -pyrimidine derivatives |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024212157A Division JP7730407B2 (ja) | 2019-07-24 | 2024-12-05 | ４－（イミダゾ［１，２－ａ］ピリジン－３－イル）－ピリミジン誘導体 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022542072A JP2022542072A (ja) | 2022-09-29 |
| JP2022542072A5 true JP2022542072A5 (https=) | 2023-07-31 |
| JP7601852B2 JP7601852B2 (ja) | 2024-12-17 |
Family
ID=67438678
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022504198A Active JP7601852B2 (ja) | 2019-07-24 | 2020-07-22 | ４－（イミダゾ［１，２－ａ］ピリジン－３－イル）－ピリミジン誘導体 |
| JP2024212157A Active JP7730407B2 (ja) | 2019-07-24 | 2024-12-05 | ４－（イミダゾ［１，２－ａ］ピリジン－３－イル）－ピリミジン誘導体 |
| JP2025135307A Pending JP2025186243A (ja) | 2019-07-24 | 2025-08-15 | ４－（イミダゾ［１，２－ａ］ピリジン－３－イル）－ピリミジン誘導体 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024212157A Active JP7730407B2 (ja) | 2019-07-24 | 2024-12-05 | ４－（イミダゾ［１，２－ａ］ピリジン－３－イル）－ピリミジン誘導体 |
| JP2025135307A Pending JP2025186243A (ja) | 2019-07-24 | 2025-08-15 | ４－（イミダゾ［１，２－ａ］ピリジン－３－イル）－ピリミジン誘導体 |
Country Status (13)
| Country | Link |
|---|---|
| US (2) | US20220267320A1 (https=) |
| EP (1) | EP4003992A1 (https=) |
| JP (3) | JP7601852B2 (https=) |
| KR (2) | KR20250174707A (https=) |
| CN (2) | CN118955500A (https=) |
| AR (1) | AR119461A1 (https=) |
| AU (2) | AU2020318710B2 (https=) |
| BR (1) | BR112022001158A2 (https=) |
| CA (1) | CA3148227A1 (https=) |
| IL (1) | IL289953B2 (https=) |
| MX (1) | MX2022000794A (https=) |
| TW (1) | TWI868186B (https=) |
| WO (1) | WO2021013864A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20240124450A1 (en) | 2022-09-21 | 2024-04-18 | Pfizer Inc. | Novel SIK Inhibitors |
| CN120379972A (zh) * | 2022-12-20 | 2025-07-25 | 深圳湾实验室 | 一种靶向usp1的小分子抑制剂及其应用 |
| WO2025248485A1 (en) | 2024-05-31 | 2025-12-04 | Idrx, Inc. | Pharmaceutical compositions and methods of use thereof |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20050014753A1 (en) | 2003-04-04 | 2005-01-20 | Irm Llc | Novel compounds and compositions as protein kinase inhibitors |
| US7977336B2 (en) | 2006-12-28 | 2011-07-12 | Banyu Pharmaceutical Co. Ltd | Aminopyrimidine derivatives as PLK1 inhibitors |
| US8124764B2 (en) * | 2008-07-14 | 2012-02-28 | Gilead Sciences, Inc. | Fused heterocyclyc inhibitor compounds |
| EP2430013B1 (en) * | 2009-05-13 | 2014-10-15 | Amgen Inc. | Heteroaryl compounds as pikk inhibitors |
| EP2338888A1 (en) | 2009-12-24 | 2011-06-29 | Almirall, S.A. | Imidazopyridine derivatives as JAK inhibitors |
| EA034866B1 (ru) | 2013-08-30 | 2020-03-31 | ПиТиСи ТЕРАПЬЮТИКС, ИНК. | Замещенные пиримидиновые ингибиторы bmi-1 |
-
2020
- 2020-07-22 BR BR112022001158A patent/BR112022001158A2/pt unknown
- 2020-07-22 IL IL289953A patent/IL289953B2/en unknown
- 2020-07-22 CA CA3148227A patent/CA3148227A1/en active Pending
- 2020-07-22 AU AU2020318710A patent/AU2020318710B2/en active Active
- 2020-07-22 WO PCT/EP2020/070616 patent/WO2021013864A1/en not_active Ceased
- 2020-07-22 KR KR1020257039581A patent/KR20250174707A/ko active Pending
- 2020-07-22 EP EP20750187.5A patent/EP4003992A1/en active Pending
- 2020-07-22 CN CN202411014632.3A patent/CN118955500A/zh active Pending
- 2020-07-22 US US17/597,729 patent/US20220267320A1/en active Pending
- 2020-07-22 MX MX2022000794A patent/MX2022000794A/es unknown
- 2020-07-22 JP JP2022504198A patent/JP7601852B2/ja active Active
- 2020-07-22 CN CN202080052946.6A patent/CN114174293B/zh active Active
- 2020-07-22 KR KR1020227005802A patent/KR102894509B1/ko active Active
- 2020-07-23 TW TW109124903A patent/TWI868186B/zh active
- 2020-07-23 AR ARP200102060A patent/AR119461A1/es unknown
-
2024
- 2024-12-05 JP JP2024212157A patent/JP7730407B2/ja active Active
-
2025
- 2025-08-15 JP JP2025135307A patent/JP2025186243A/ja active Pending
- 2025-10-30 US US19/373,991 patent/US20260109697A1/en active Pending
-
2026
- 2026-01-23 AU AU2026200481A patent/AU2026200481A1/en active Pending
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