JP2022537358A5 - - Google Patents

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Publication number
JP2022537358A5
JP2022537358A5 JP2021575365A JP2021575365A JP2022537358A5 JP 2022537358 A5 JP2022537358 A5 JP 2022537358A5 JP 2021575365 A JP2021575365 A JP 2021575365A JP 2021575365 A JP2021575365 A JP 2021575365A JP 2022537358 A5 JP2022537358 A5 JP 2022537358A5
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JP
Japan
Prior art keywords
cancer
compound according
amino
compound
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2021575365A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022537358A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/038395 external-priority patent/WO2020257429A1/en
Publication of JP2022537358A publication Critical patent/JP2022537358A/ja
Publication of JP2022537358A5 publication Critical patent/JP2022537358A5/ja
Withdrawn legal-status Critical Current

Links

JP2021575365A 2019-06-20 2020-06-18 エクトヌクレオチダーゼ阻害剤およびその使用方法 Withdrawn JP2022537358A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962864031P 2019-06-20 2019-06-20
US62/864,031 2019-06-20
PCT/US2020/038395 WO2020257429A1 (en) 2019-06-20 2020-06-18 Ectonucleotidase inhibitors and methods of use thereof

Publications (2)

Publication Number Publication Date
JP2022537358A JP2022537358A (ja) 2022-08-25
JP2022537358A5 true JP2022537358A5 (enExample) 2023-06-14

Family

ID=74040909

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021575365A Withdrawn JP2022537358A (ja) 2019-06-20 2020-06-18 エクトヌクレオチダーゼ阻害剤およびその使用方法

Country Status (8)

Country Link
US (1) US20220363709A1 (enExample)
EP (1) EP3986894A4 (enExample)
JP (1) JP2022537358A (enExample)
KR (1) KR20220024629A (enExample)
CN (1) CN114008048A (enExample)
AU (1) AU2020294724A1 (enExample)
CA (1) CA3143496A1 (enExample)
WO (1) WO2020257429A1 (enExample)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2018208980A1 (en) 2017-05-10 2018-11-15 Oric Pharmaceuticals, Inc. Cd73 inhibitors
US11377469B2 (en) 2017-11-03 2022-07-05 Oric Pharmaceuticals, Inc. CD73 inhibitors
IL304348B2 (en) 2018-04-30 2024-08-01 Oric Pharmaceuticals Inc CD73 inhibitors
SG11202012001YA (en) 2018-06-21 2021-01-28 Calithera Biosciences Inc Ectonucleotidase inhibitors and methods of use thereof
JP7557522B2 (ja) 2019-07-16 2024-09-27 オリック ファーマシューティカルズ,インク. Cd73阻害剤
PL4051688T3 (pl) 2019-10-30 2025-09-22 Oric Pharmaceuticals, Inc. Inhibitory cd73
JP2025512384A (ja) 2022-04-13 2025-04-17 ギリアード サイエンシーズ, インコーポレイテッド Trop-2発現がんを治療するための併用療法
KR102775989B1 (ko) * 2022-11-01 2025-03-04 윤주호 콜치신과 메트포르민을 유효성분으로 하는 퇴행성 신경계 질환의 예방 또는 치료용 조성물
WO2025137640A1 (en) 2023-12-22 2025-06-26 Gilead Sciences, Inc. Azaspiro wrn inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW528755B (en) * 1996-12-24 2003-04-21 Glaxo Group Ltd 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives
MA39986A (fr) * 2014-04-25 2017-03-01 Vitae Pharmaceuticals Inc Dérivés de purine en tant qu'inhibiteurs de cd73 pour le traitement du cancer
EP3510040A4 (en) * 2016-09-09 2020-06-03 Calithera Biosciences, Inc. EKTONUCLEOTIDASE INHIBITORS AND METHOD FOR USE THEREOF
KR102638592B1 (ko) * 2016-12-22 2024-02-19 안텐진 테라퓨틱스 리미티드 엑토뉴클레오티다제 억제제 및 이의 용도
SG11202012001YA (en) * 2018-06-21 2021-01-28 Calithera Biosciences Inc Ectonucleotidase inhibitors and methods of use thereof

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