JP2022537358A5 - - Google Patents

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Publication number
JP2022537358A5
JP2022537358A5 JP2021575365A JP2021575365A JP2022537358A5 JP 2022537358 A5 JP2022537358 A5 JP 2022537358A5 JP 2021575365 A JP2021575365 A JP 2021575365A JP 2021575365 A JP2021575365 A JP 2021575365A JP 2022537358 A5 JP2022537358 A5 JP 2022537358A5
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JP
Japan
Prior art keywords
cancer
compound according
amino
compound
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2021575365A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022537358A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/038395 external-priority patent/WO2020257429A1/en
Publication of JP2022537358A publication Critical patent/JP2022537358A/ja
Publication of JP2022537358A5 publication Critical patent/JP2022537358A5/ja
Withdrawn legal-status Critical Current

Links

JP2021575365A 2019-06-20 2020-06-18 エクトヌクレオチダーゼ阻害剤およびその使用方法 Withdrawn JP2022537358A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962864031P 2019-06-20 2019-06-20
US62/864,031 2019-06-20
PCT/US2020/038395 WO2020257429A1 (en) 2019-06-20 2020-06-18 Ectonucleotidase inhibitors and methods of use thereof

Publications (2)

Publication Number Publication Date
JP2022537358A JP2022537358A (ja) 2022-08-25
JP2022537358A5 true JP2022537358A5 (enExample) 2023-06-14

Family

ID=74040909

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021575365A Withdrawn JP2022537358A (ja) 2019-06-20 2020-06-18 エクトヌクレオチダーゼ阻害剤およびその使用方法

Country Status (8)

Country Link
US (1) US20220363709A1 (enExample)
EP (1) EP3986894A4 (enExample)
JP (1) JP2022537358A (enExample)
KR (1) KR20220024629A (enExample)
CN (1) CN114008048A (enExample)
AU (1) AU2020294724A1 (enExample)
CA (1) CA3143496A1 (enExample)
WO (1) WO2020257429A1 (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11129841B2 (en) 2017-05-10 2021-09-28 Oric Pharmaceuticals, Inc. CD73 inhibitors
US11377469B2 (en) 2017-11-03 2022-07-05 Oric Pharmaceuticals, Inc. CD73 inhibitors
CA3098493A1 (en) 2018-04-30 2019-11-07 Oric Pharmaceuticals, Inc. Cd73 inhibitors
KR102902754B1 (ko) 2018-06-21 2025-12-19 안텐진 테라퓨틱스 리미티드 엑토뉴클레오티다제 저해제 및 이의 사용 방법
US12544391B2 (en) 2019-07-16 2026-02-10 Oric Pharmaceuticals, Inc. CD73 inhibitors
CN116854758A (zh) 2019-10-30 2023-10-10 欧瑞克制药公司 Cd73抑制剂
AU2023252914A1 (en) 2022-04-13 2024-10-17 Arcus Biosciences, Inc. Combination therapy for treating trop-2 expressing cancers
KR102775989B1 (ko) * 2022-11-01 2025-03-04 윤주호 콜치신과 메트포르민을 유효성분으로 하는 퇴행성 신경계 질환의 예방 또는 치료용 조성물
US20250230168A1 (en) 2023-12-22 2025-07-17 Gilead Sciences, Inc. Azaspiro wrn inhibitors
CN118001265A (zh) * 2024-03-14 2024-05-10 哈尔滨医科大学附属第一医院 苏拉明在制备减轻心肌梗死后心肌纤维化产品中的应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW528755B (en) * 1996-12-24 2003-04-21 Glaxo Group Ltd 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives
EP3134411B1 (en) * 2014-04-25 2021-06-30 Boehringer Ingelheim International GmbH Purine derivatives as cd73 inhibitors for the treatment of cancer
CN110234656B (zh) * 2016-09-09 2023-02-28 卡利泰拉生物科技公司 外核苷酸酶抑制剂及其使用方法
KR102638592B1 (ko) * 2016-12-22 2024-02-19 안텐진 테라퓨틱스 리미티드 엑토뉴클레오티다제 억제제 및 이의 용도
KR102902754B1 (ko) * 2018-06-21 2025-12-19 안텐진 테라퓨틱스 리미티드 엑토뉴클레오티다제 저해제 및 이의 사용 방법

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