JP2022537358A - エクトヌクレオチダーゼ阻害剤およびその使用方法 - Google Patents
エクトヌクレオチダーゼ阻害剤およびその使用方法 Download PDFInfo
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- JP2022537358A JP2022537358A JP2021575365A JP2021575365A JP2022537358A JP 2022537358 A JP2022537358 A JP 2022537358A JP 2021575365 A JP2021575365 A JP 2021575365A JP 2021575365 A JP2021575365 A JP 2021575365A JP 2022537358 A JP2022537358 A JP 2022537358A
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- amino
- cancer
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- chloro
- alkyl
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- A61K31/7076—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
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- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
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Landscapes
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| JP6657182B2 (ja) * | 2014-04-25 | 2020-03-04 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 癌治療用のｃｄ７３阻害剤としてのプリン誘導体 |
| WO2018049145A1 (en) * | 2016-09-09 | 2018-03-15 | Calithera Biosciences, Inc. | Ectonucleotidase inhibitors and methods of use thereof |
| CN110402249A (zh) * | 2016-12-22 | 2019-11-01 | 卡利泰拉生物科技公司 | 外核苷酸酶抑制剂及其使用方法 |
| CN112888696B (zh) * | 2018-06-21 | 2024-04-16 | 德琪医疗有限公司 | 外核苷酸酶抑制剂及其使用方法 |
-
2020
- 2020-06-18 AU AU2020294724A patent/AU2020294724A1/en not_active Abandoned
- 2020-06-18 JP JP2021575365A patent/JP2022537358A/ja not_active Withdrawn
- 2020-06-18 US US17/620,508 patent/US20220363709A1/en not_active Abandoned
- 2020-06-18 WO PCT/US2020/038395 patent/WO2020257429A1/en not_active Ceased
- 2020-06-18 CN CN202080045115.6A patent/CN114008048A/zh active Pending
- 2020-06-18 CA CA3143496A patent/CA3143496A1/en active Pending
- 2020-06-18 KR KR1020227001589A patent/KR20220024629A/ko not_active Withdrawn
- 2020-06-18 EP EP20826073.7A patent/EP3986894A4/en not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| KR20220024629A (ko) | 2022-03-03 |
| CN114008048A (zh) | 2022-02-01 |
| EP3986894A1 (en) | 2022-04-27 |
| EP3986894A4 (en) | 2023-08-09 |
| CA3143496A1 (en) | 2020-12-24 |
| US20220363709A1 (en) | 2022-11-17 |
| WO2020257429A1 (en) | 2020-12-24 |
| AU2020294724A1 (en) | 2022-01-20 |
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