JP2022529061A5 - - Google Patents

Info

Publication number
JP2022529061A5
JP2022529061A5 JP2021561927A JP2021561927A JP2022529061A5 JP 2022529061 A5 JP2022529061 A5 JP 2022529061A5 JP 2021561927 A JP2021561927 A JP 2021561927A JP 2021561927 A JP2021561927 A JP 2021561927A JP 2022529061 A5 JP2022529061 A5 JP 2022529061A5
Authority
JP
Japan
Prior art keywords
compound according
alkyl
hydroxyl
pharmaceutically acceptable
pharmaceutical composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021561927A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022529061A (ja
JP7555959B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CN2020/085338 external-priority patent/WO2020211839A1/en
Publication of JP2022529061A publication Critical patent/JP2022529061A/ja
Publication of JP2022529061A5 publication Critical patent/JP2022529061A5/ja
Application granted granted Critical
Publication of JP7555959B2 publication Critical patent/JP7555959B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2021561927A 2019-04-19 2020-04-17 Jak1選択的キナーゼ阻害剤 Active JP7555959B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CNPCT/CN2019/083376 2019-04-19
CN2019083376 2019-04-19
PCT/CN2020/085338 WO2020211839A1 (en) 2019-04-19 2020-04-17 Jak1 selective kinase inhibitor

Publications (3)

Publication Number Publication Date
JP2022529061A JP2022529061A (ja) 2022-06-16
JP2022529061A5 true JP2022529061A5 (https=) 2024-07-08
JP7555959B2 JP7555959B2 (ja) 2024-09-25

Family

ID=72837031

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021561927A Active JP7555959B2 (ja) 2019-04-19 2020-04-17 Jak1選択的キナーゼ阻害剤

Country Status (15)

Country Link
US (1) US12606544B2 (https=)
EP (1) EP3956322B1 (https=)
JP (1) JP7555959B2 (https=)
KR (1) KR20220003537A (https=)
CN (1) CN113710664B (https=)
AR (1) AR118729A1 (https=)
AU (1) AU2020258619C1 (https=)
BR (1) BR112021020964A2 (https=)
CA (1) CA3134174A1 (https=)
DK (1) DK3956322T3 (https=)
ES (1) ES3031576T3 (https=)
MX (1) MX2021012749A (https=)
PT (1) PT3956322T (https=)
TW (1) TWI910107B (https=)
WO (1) WO2020211839A1 (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022111499A1 (zh) * 2020-11-26 2022-06-02 深圳铂立健医药有限公司 一种酰胺化合物、药物组合物及其应用
CN114380806B (zh) * 2022-03-24 2022-06-10 中国药科大学 2-氨基-4-吲哚基嘧啶类化合物及其制备方法与应用
US12240836B2 (en) * 2022-07-05 2025-03-04 Dong-A St Co., Ltd. Compounds as GCN2 inhibitors, pharmaceutical compositions and uses thereof
EP4554931A1 (en) * 2022-07-12 2025-05-21 Adama Makhteshim Ltd. Process for preparing substituted benzamides
CN115260128B (zh) * 2022-09-21 2022-12-09 苏州凯瑞医药科技有限公司 一种新型jak抑制剂关键中间体的制备方法
GB202403369D0 (en) 2024-03-08 2024-04-24 Astrazeneca Ab Process and intermediates for the production of a jak1 inhibitor

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9198900B2 (en) * 2011-11-10 2015-12-01 Los Angeles Biomedical Research Institute At Harbor-Ucla Medical Center Treatment of peritoneal injury using JAK inhibitors
JP6767491B2 (ja) 2015-09-25 2020-10-14 ディザル(ジァンスー)ファーマシューティカル・カンパニー・リミテッド Jakを阻害するための化合物及び方法
ES2938648T3 (es) * 2017-01-17 2023-04-13 Astrazeneca Ab Inhibidores selectivos de JAK1
CA3113732C (en) * 2018-09-21 2023-07-11 Shanghai Ennovabio Pharmaceuticals Co., Ltd. Aromatic heterocyclic compound with kinase inhibitory activity

Similar Documents

Publication Publication Date Title
JP2022529061A5 (https=)
JP6434416B2 (ja) PDE4阻害剤とPI3δ阻害剤または二重PI3δ−γキナーゼ阻害剤とを含有する薬学的組成物
CN114072396A (zh) 作为dna-pk抑制剂的喹啉和噌啉衍生物
JP2014505107A5 (https=)
US20150018396A1 (en) Prevention and treatment of respiratory infection with peroxisome proliferator activator receptor delta agonist
JP2019509276A5 (https=)
JP2010524932A5 (https=)
JP2008531714A (ja) 不安障害の治療用及び/又は予防用の医薬組成物
RU2017105470A (ru) Способы лечения парамиксовирусов
JP2005509024A5 (https=)
CN104024217B (zh) 用于治疗或预防与内分泌功能障碍相关的症状的三环含氨基化合物
JP2019505529A5 (https=)
JP2008538741A (ja) 鬱病の治療用及び/又は予防用の医薬組成物
JP2017504635A5 (https=)
RU2009123525A (ru) ПРОИЗВОДНЫЕ 5-СУЛЬФАНИЛМЕТИЛ[1,2,4}ТРИАЗОЛ[1,5-а]ПИРИМИДИН-7-ОЛА В КАЧЕСТВЕ АНТАГОНИСТОВ CXCR2
JP2023512664A5 (https=)
JP2018522861A5 (https=)
RU2015146417A (ru) Пероральная фармацевтическая композиция для профилактики или лечения синдрома "сухого глаза", содержащая ребамипид или его предшественник
RU2014119711A (ru) Трициклические соединения, композиции, содержащие указанные соединения, и их применения
WO2016101898A1 (zh) 3-[(苯并[d][1,3]二氧戊环-4-基)-氧基]-3-芳基丙胺类化合物及其应用
JP2007518798A5 (https=)
CA2567797A1 (en) Peptidic vasopressin receptor agonists
JP2020510061A5 (https=)
DK1634595T3 (da) N-Phenylbenzamidderivater som medikamenter til behandling af kronisk obstruktiv lungesygdom (KOL)
JP2006524677A5 (https=)