JP2022513089A5 - - Google Patents

Info

Publication number
JP2022513089A5
JP2022513089A5 JP2021527849A JP2021527849A JP2022513089A5 JP 2022513089 A5 JP2022513089 A5 JP 2022513089A5 JP 2021527849 A JP2021527849 A JP 2021527849A JP 2021527849 A JP2021527849 A JP 2021527849A JP 2022513089 A5 JP2022513089 A5 JP 2022513089A5
Authority
JP
Japan
Prior art keywords
alkyl
pharmaceutical composition
composition according
hydrogen
cycloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021527849A
Other languages
English (en)
Japanese (ja)
Other versions
JP7576799B2 (ja
JP2022513089A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/000065 external-priority patent/WO2020106303A1/en
Publication of JP2022513089A publication Critical patent/JP2022513089A/ja
Publication of JP2022513089A5 publication Critical patent/JP2022513089A5/ja
Application granted granted Critical
Publication of JP7576799B2 publication Critical patent/JP7576799B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2021527849A 2018-11-20 2019-11-20 皮膚癌の処置のためのアリールアニリンおよびヘテロアリールアニリン化合物 Active JP7576799B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862769879P 2018-11-20 2018-11-20
US62/769,879 2018-11-20
PCT/US2019/000065 WO2020106303A1 (en) 2018-11-20 2019-11-20 Aryl-aniline and heteroaryl-aniline compounds for treatment of skin cancers

Publications (3)

Publication Number Publication Date
JP2022513089A JP2022513089A (ja) 2022-02-07
JP2022513089A5 true JP2022513089A5 (https=) 2023-09-11
JP7576799B2 JP7576799B2 (ja) 2024-11-01

Family

ID=70773565

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021527849A Active JP7576799B2 (ja) 2018-11-20 2019-11-20 皮膚癌の処置のためのアリールアニリンおよびヘテロアリールアニリン化合物

Country Status (8)

Country Link
US (2) US20220087989A1 (https=)
EP (2) EP3883553A4 (https=)
JP (1) JP7576799B2 (https=)
CN (2) CN113660931B (https=)
AU (1) AU2019383310B2 (https=)
CA (1) CA3120351A1 (https=)
MA (1) MA55143A (https=)
WO (1) WO2020106303A1 (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2020106308A1 (en) 2018-11-20 2020-05-28 Nflection Therapeutics, Inc. Naphthyridinone-aniline compounds for treatment of dermal disorders
WO2020106306A1 (en) 2018-11-20 2020-05-28 Nflection Therapeutics, Inc. Cyanoaryl-aniline compounds for treatment of dermal disorders
WO2020106305A1 (en) * 2018-11-20 2020-05-28 Nflection Therapeutics, Inc. Thienyl-aniline compounds for treatment of dermal disorders
EP4281055A4 (en) * 2021-01-21 2025-06-18 NFlection Therapeutics, Inc. CRYSTALLINE FORMS OF A PYRROLOPYRIDINANILINE COMPOUND
IL312977A (en) 2021-11-23 2024-07-01 Nflection Therapeutics Inc Formulations of pyrrolopyridine-aniline compounds
WO2023096935A1 (en) * 2021-11-23 2023-06-01 Nflection Therapeutics, Inc. Formulations of pyrrolopyridine-aniline compounds
TW202342018A (zh) 2022-03-04 2023-11-01 美商奇奈特生物製藥公司 Mek激酶抑制劑
EP4493169A4 (en) * 2022-03-17 2026-03-04 Springworks Therapeutics Inc Fluorinated phenylamine compounds and pharmaceutical compositions

Family Cites Families (50)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3536809A (en) 1969-02-17 1970-10-27 Alza Corp Medication method
US3598123A (en) 1969-04-01 1971-08-10 Alza Corp Bandage for administering drugs
US3845770A (en) 1972-06-05 1974-11-05 Alza Corp Osmatic dispensing device for releasing beneficial agent
US3916899A (en) 1973-04-25 1975-11-04 Alza Corp Osmotic dispensing device with maximum and minimum sizes for the passageway
US4008719A (en) 1976-02-02 1977-02-22 Alza Corporation Osmotic system having laminar arrangement for programming delivery of active agent
HU196714B (en) 1984-10-04 1989-01-30 Monsanto Co Process for producing non-aqueous composition comprising somatotropin
IE58110B1 (en) 1984-10-30 1993-07-14 Elan Corp Plc Controlled release powder and process for its preparation
US5073543A (en) 1988-07-21 1991-12-17 G. D. Searle & Co. Controlled release formulations of trophic factors in ganglioside-lipsome vehicle
IT1229203B (it) 1989-03-22 1991-07-25 Bioresearch Spa Impiego di acido 5 metiltetraidrofolico, di acido 5 formiltetraidrofolico e dei loro sali farmaceuticamente accettabili per la preparazione di composizioni farmaceutiche in forma a rilascio controllato attive nella terapia dei disturbi mentali organici e composizioni farmaceutiche relative.
PH30995A (en) 1989-07-07 1997-12-23 Novartis Inc Sustained release formulations of water soluble peptides.
US5120548A (en) 1989-11-07 1992-06-09 Merck & Co., Inc. Swelling modulated polymeric drug delivery device
US5733566A (en) 1990-05-15 1998-03-31 Alkermes Controlled Therapeutics Inc. Ii Controlled release of antiparasitic agents in animals
US5580578A (en) 1992-01-27 1996-12-03 Euro-Celtique, S.A. Controlled release formulations coated with aqueous dispersions of acrylic polymers
TW333456B (en) 1992-12-07 1998-06-11 Takeda Pharm Ind Co Ltd A pharmaceutical composition of sustained-release preparation the invention relates to a pharmaceutical composition of sustained-release preparation which comprises a physiologically active peptide.
US5591767A (en) 1993-01-25 1997-01-07 Pharmetrix Corporation Liquid reservoir transdermal patch for the administration of ketorolac
US6087324A (en) 1993-06-24 2000-07-11 Takeda Chemical Industries, Ltd. Sustained-release preparation
IT1270594B (it) 1994-07-07 1997-05-07 Recordati Chem Pharm Composizione farmaceutica a rilascio controllato di moguisteina in sospensione liquida
AU6242096A (en) 1995-06-27 1997-01-30 Takeda Chemical Industries Ltd. Method of producing sustained-release preparation
TW448055B (en) 1995-09-04 2001-08-01 Takeda Chemical Industries Ltd Method of production of sustained-release preparation
JP2909418B2 (ja) 1995-09-18 1999-06-23 株式会社資生堂 薬物の遅延放出型マイクロスフイア
US5980945A (en) 1996-01-16 1999-11-09 Societe De Conseils De Recherches Et D'applications Scientifique S.A. Sustained release drug formulations
US6264970B1 (en) 1996-06-26 2001-07-24 Takeda Chemical Industries, Ltd. Sustained-release preparation
US6419961B1 (en) 1996-08-29 2002-07-16 Takeda Chemical Industries, Ltd. Sustained release microcapsules of a bioactive substance and a biodegradable polymer
CA2217134A1 (en) 1996-10-09 1998-04-09 Sumitomo Pharmaceuticals Co., Ltd. Sustained release formulation
PT839525E (pt) 1996-10-31 2004-10-29 Takeda Chemical Industries Ltd Preparacao de libertacao prolongada
WO1998027980A2 (en) 1996-12-20 1998-07-02 Takeda Chemical Industries, Ltd. Method of producing a sustained-release preparation
US5891474A (en) 1997-01-29 1999-04-06 Poli Industria Chimica, S.P.A. Time-specific controlled release dosage formulations and method of preparing same
BR9810385A (pt) * 1997-07-01 2000-09-05 Warner Lambert Co Derivados de ácido benzóico 2-(4-bromo ou 4-iodo fenilamino) e sua utilização como inibidores de mek
NZ501276A (en) 1997-07-01 2000-10-27 Warner Lambert Co 4-bromo or 4-iodo phenylamino benzhydroxamic acid derivatives and their use as MEK inhibitors in treating proliferative disorders
US6613358B2 (en) 1998-03-18 2003-09-02 Theodore W. Randolph Sustained-release composition including amorphous polymer
KR19990085365A (ko) 1998-05-16 1999-12-06 허영섭 지속적으로 약물 조절방출이 가능한 생분해성 고분자 미립구 및그 제조방법
DE69926914T2 (de) * 1999-01-13 2006-06-29 Warner-Lambert Co. Llc 1-heterozyklus-substituierte diarylaminen
US6248363B1 (en) 1999-11-23 2001-06-19 Lipocine, Inc. Solid carriers for improved delivery of active ingredients in pharmaceutical compositions
JP5710855B2 (ja) 2005-02-02 2015-04-30 ネクスジェニクス・ファーマシューティカルズ,リミテッド・ライアビリティ・カンパニー 神経線維腫の局所治療
SI1934174T1 (sl) 2005-10-07 2011-08-31 Exelixis Inc Inhibitorji MEK in postopki za njihovo uporabo
GB0601962D0 (en) * 2006-01-31 2006-03-15 Ucb Sa Therapeutic agents
US7772233B2 (en) * 2006-04-19 2010-08-10 Merck Serono, S.A. Arylamino N-heteroaryl compounds as MEK inhibitors
GB0616214D0 (en) * 2006-08-15 2006-09-27 Ucb Sa Therapeutic Agents
CN101528231A (zh) * 2006-08-16 2009-09-09 埃克塞利希斯股份有限公司 在癌症的治疗中使用pi3k和mek调控剂
EP2089359A2 (en) 2006-10-31 2009-08-19 Takeda Pharmaceutical Company Limited Mapk/erk kinase inhibitors
US20090082328A1 (en) * 2007-05-11 2009-03-26 Bayer Schering Pharma Aktiengesellschaft Substituted phenylamino-benzene derivatives useful for treating hyper-proliferative disorders and diseases associated with mitogen extracellular kinase activity
US20080312307A1 (en) 2007-05-25 2008-12-18 Takeda Pharmaceutical Company Limited Mapk/erk kinase inhibitors
GB0714384D0 (en) * 2007-07-23 2007-09-05 Ucb Pharma Sa theraputic agents
GB0801081D0 (en) * 2008-01-21 2008-02-27 Ucb Pharma Sa Therapeutic agents
JP7237941B2 (ja) * 2017-05-19 2023-03-13 エヌフレクション セラピューティクス インコーポレイテッド 皮膚障害の処置用の融合複素環式芳香族アニリン化合物
PT3624796T (pt) * 2017-05-19 2025-06-02 Nflection Therapeutics Inc Compostos de pirrolopiridina-anilina para tratamento de distúrbios dérmicos
CN112334496B (zh) * 2018-06-01 2023-12-22 陶氏环球技术有限责任公司 用于产生聚乙烯的齐格勒-纳塔催化剂
WO2020106304A1 (en) * 2018-11-20 2020-05-28 Nflection Therapeutics, Inc. Topical formulations
WO2020106305A1 (en) * 2018-11-20 2020-05-28 Nflection Therapeutics, Inc. Thienyl-aniline compounds for treatment of dermal disorders
EP4233834A3 (en) * 2018-11-20 2023-10-25 NFlection Therapeutics, Inc. Aryl-aniline and heteroaryl-aniline compounds for treatment of birthmarks

Similar Documents

Publication Publication Date Title
JP2022513089A5 (https=)
JP2022511127A5 (https=)
PH12022550611A1 (en) Brd9 bifunctional degraders and their methods of use
WO2022222994A1 (zh) 一种核苷类化合物及其在治疗猫传染性腹膜炎中的应用
MX2025011899A (es) Compuestos de pirido[4,3-d]pirimidina
CN111263586B (zh) 乙型肝炎抗病毒剂
CN103664899B (zh) 杂芳基取代的二氢嘧啶类化合物及其在药物中的应用
RU2017117413A (ru) Пролекарства карбидопа и l-dopa и их применение для лечения болезни паркинсона
HK1250032A1 (zh) 作为sting调节剂的环状嘌呤二核苷酸
WO2017066227A1 (en) Compounds useful as immunomodulators
WO2016134223A3 (en) Fluorinated tetrahydronaphthyridinyl nonanoic acid derivatives and uses thereof
MX2010007374A (es) Nuevos derivados de c-21-ceto lupano, preparacion y uso de los mismos.
RU2009144538A (ru) Новые циклические пептидные соединения
JP2017513824A5 (https=)
JP2022510586A5 (https=)
JP2017200931A (ja) スルフォラファンの単離及び精製
JP2017518360A5 (https=)
MX2024014315A (es) Compuestos amido heteroaromaticos utiles en el tratamiento de enfermedades hepaticas
JP2022511730A5 (https=)
CA3170031A1 (en) Nicotinamide mononucleotide derivatives for the treatment of arrhythmia
CN104530127B (zh) 一种淫羊藿苷衍生物及其使用方法和用途
RU2017140078A (ru) Косметический способ и его терапевтическое применение для уменьшения объема жировой ткани
JP2013525290A5 (https=)
WO2025049521A3 (en) Aryl ether analogs as inhibitors of the menin-mll interaction
EP2276464A2 (en) Combinations of antiviral agents and other compounds