JP2022511540A5 - - Google Patents

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Publication number
JP2022511540A5
JP2022511540A5 JP2021532155A JP2021532155A JP2022511540A5 JP 2022511540 A5 JP2022511540 A5 JP 2022511540A5 JP 2021532155 A JP2021532155 A JP 2021532155A JP 2021532155 A JP2021532155 A JP 2021532155A JP 2022511540 A5 JP2022511540 A5 JP 2022511540A5
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JP
Japan
Application number
JP2021532155A
Other languages
Japanese (ja)
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JP2022511540A (ja
JPWO2020124059A5 (https=
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Publication date
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Priority claimed from PCT/US2019/066413 external-priority patent/WO2020124059A1/en
Publication of JP2022511540A publication Critical patent/JP2022511540A/ja
Publication of JP2022511540A5 publication Critical patent/JP2022511540A5/ja
Publication of JPWO2020124059A5 publication Critical patent/JPWO2020124059A5/ja
Pending legal-status Critical Current

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JP2021532155A 2018-12-14 2019-12-14 Stingアゴニストとしての三環式化合物、ならびにその調製方法および医薬用途 Pending JP2022511540A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862779907P 2018-12-14 2018-12-14
US62/779,907 2018-12-14
PCT/US2019/066413 WO2020124059A1 (en) 2018-12-14 2019-12-14 Tricyclic compounds as sting agonists, and preparation methods and medicinal uses thereof

Publications (3)

Publication Number Publication Date
JP2022511540A JP2022511540A (ja) 2022-01-31
JP2022511540A5 true JP2022511540A5 (https=) 2022-12-19
JPWO2020124059A5 JPWO2020124059A5 (https=) 2022-12-19

Family

ID=71077552

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021532155A Pending JP2022511540A (ja) 2018-12-14 2019-12-14 Stingアゴニストとしての三環式化合物、ならびにその調製方法および医薬用途

Country Status (6)

Country Link
US (1) US20220056044A1 (https=)
EP (1) EP3873896A4 (https=)
JP (1) JP2022511540A (https=)
CN (1) CN113195473B (https=)
TW (1) TW202039508A (https=)
WO (1) WO2020124059A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111655682B (zh) * 2018-08-29 2024-05-31 杭州阿诺生物医药科技有限公司 一种高活性sting蛋白激动剂化合物
WO2021206158A1 (ja) 2020-04-10 2021-10-14 小野薬品工業株式会社 がん治療方法
CN119110800A (zh) * 2022-02-21 2024-12-10 健道生物医药有限公司 干扰素基因刺激因子(sting)调节剂及其组合物和方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2747678B1 (fr) * 1996-04-22 1998-05-22 Synthelabo Composes derives d'imidazobenzoxazine, leurs procedes de preparation et leurs utilisations en therapeutique
ECSP003637A (es) * 1999-08-31 2002-03-25 Agouron Pharma Inhibidores triciclicos de poli (adp-ribosa) polimerasas
KR20080035576A (ko) * 2005-08-05 2008-04-23 아스트라제네카 아베 트리사이클릭 벤즈이미다졸 및 대사체 글루타메이트 수용체조절제로서 이들의 용도
GB201220157D0 (en) * 2012-11-08 2012-12-26 Selvita Sa Substitute tricyclic benzimidazoles as kinase inhibitors
MX366703B (es) * 2013-03-15 2019-07-22 Incyte Holdings Corp Heterociclos tricíclicos como inhibidores de la proteína bet.
HRP20220936T1 (hr) * 2016-04-07 2022-10-28 Glaxosmithkline Intellectual Property Development Limited Heterociklički amidi korisni kao modulatori proteina
JP2021530442A (ja) * 2018-06-28 2021-11-11 ジエンス ヘンルイ メデイシンカンパニー リミテッドJiangsu Hengrui Medicine Co., Ltd. 縮合三環系複素環化合物およびその治療上の使用
CN111655682B (zh) * 2018-08-29 2024-05-31 杭州阿诺生物医药科技有限公司 一种高活性sting蛋白激动剂化合物

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