JP2022500456A5 - - Google Patents

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Publication number
JP2022500456A5
JP2022500456A5 JP2021514419A JP2021514419A JP2022500456A5 JP 2022500456 A5 JP2022500456 A5 JP 2022500456A5 JP 2021514419 A JP2021514419 A JP 2021514419A JP 2021514419 A JP2021514419 A JP 2021514419A JP 2022500456 A5 JP2022500456 A5 JP 2022500456A5
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JP
Japan
Prior art keywords
crystal form
compound
cancer
chemical formula
group
Prior art date
Application number
JP2021514419A
Other languages
English (en)
Japanese (ja)
Other versions
JPWO2020053816A5 (https=
JP2022500456A (ja
JP7554030B2 (ja
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Priority claimed from PCT/IB2019/057720 external-priority patent/WO2020053816A1/en
Publication of JP2022500456A publication Critical patent/JP2022500456A/ja
Publication of JP2022500456A5 publication Critical patent/JP2022500456A5/ja
Publication of JPWO2020053816A5 publication Critical patent/JPWO2020053816A5/ja
Application granted granted Critical
Publication of JP7554030B2 publication Critical patent/JP7554030B2/ja
Active legal-status Critical Current
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JP2021514419A 2018-09-14 2019-09-12 キナゾリン化合物及びその塩酸塩の結晶形 Active JP7554030B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862731500P 2018-09-14 2018-09-14
US62/731,500 2018-09-14
PCT/IB2019/057720 WO2020053816A1 (en) 2018-09-14 2019-09-12 Crystalline forms of a quinazole compound and its hydrochloride salts

Publications (4)

Publication Number Publication Date
JP2022500456A JP2022500456A (ja) 2022-01-04
JP2022500456A5 true JP2022500456A5 (https=) 2022-09-22
JPWO2020053816A5 JPWO2020053816A5 (https=) 2022-09-22
JP7554030B2 JP7554030B2 (ja) 2024-09-19

Family

ID=69776732

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021513941A Pending JP2022500416A (ja) 2018-09-14 2019-09-12 がんを処置するためのキットおよび方法
JP2021514419A Active JP7554030B2 (ja) 2018-09-14 2019-09-12 キナゾリン化合物及びその塩酸塩の結晶形

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2021513941A Pending JP2022500416A (ja) 2018-09-14 2019-09-12 がんを処置するためのキットおよび方法

Country Status (17)

Country Link
US (2) US20220040180A1 (https=)
EP (2) EP3849557A4 (https=)
JP (2) JP2022500416A (https=)
KR (2) KR102802129B1 (https=)
CN (2) CN112770758A (https=)
AR (2) AR116669A1 (https=)
AU (2) AU2019337640A1 (https=)
BR (2) BR112021004527A2 (https=)
CA (2) CA3110369A1 (https=)
IL (2) IL281168A (https=)
MX (2) MX2021002875A (https=)
PH (2) PH12021550432A1 (https=)
PY (2) PY1976960A (https=)
SG (2) SG11202102006YA (https=)
TW (2) TW202027750A (https=)
UY (2) UY38374A (https=)
WO (2) WO2020056156A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112021004527A2 (pt) 2018-09-14 2021-06-08 Spectrum Pharmaceuticals, Inc. kits e métodos para tratamento contra câncer
JP2023503318A (ja) 2019-11-21 2023-01-27 ファルマ、マール、ソシエダード、アノニマ ルルビネクテジン製剤で小細胞肺がんを処置する方法
CN114642728A (zh) * 2021-06-02 2022-06-21 德琪(浙江)医药科技有限公司 mTOR抑制剂的制药用途及其药物组合物

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5069905B2 (ja) * 2003-01-21 2012-11-07 アプテュイト (ウエスト ラファイエット)、エルエルシー 新規な共結晶化
KR100735639B1 (ko) * 2004-12-29 2007-07-04 한미약품 주식회사 암세포 성장 억제 효과를 갖는 퀴나졸린 유도체 및 이의제조방법
MX2007010399A (es) * 2005-02-26 2007-09-25 Astrazeneca Ab Derivados de quinazolina en la forma de inhibidores de cinasa de tirosina.
CN101454302A (zh) * 2006-05-31 2009-06-10 艾博特公司 用作大麻素受体配位体的噻唑化合物及其用途
CA2659307A1 (en) 2006-07-28 2008-01-31 Synthon B.V. Crystalline erlotinib
US8349855B2 (en) * 2007-02-21 2013-01-08 Natco Pharma Limited Polymorphs of erlotinib hydrochloride and method of preparation
TWI377944B (en) 2007-06-05 2012-12-01 Hanmi Holdings Co Ltd Novel amide derivative for inhibiting the growth of cancer cells
KR101217526B1 (ko) * 2010-06-11 2013-01-02 한미사이언스 주식회사 아마이드 유도체 또는 이의 약학적으로 허용 가능한 염을 포함하는 약제학적 조성물
KR101317809B1 (ko) * 2011-06-07 2013-10-16 한미약품 주식회사 암세포의 성장을 억제하는 아마이드 유도체 및 비금속염 활택제를 포함하는 약학 조성물
KR101272613B1 (ko) * 2011-10-05 2013-06-10 한미사이언스 주식회사 1-(4-(4-(3,4-디클로로-2-플루오로페닐아미노)-7-메톡시퀴나졸린-6-일옥시)피페리딘-1-일)프로프-2-엔-1-온 염산염의 제조 방법 및 이에 사용되는 중간체
CN105209456B (zh) * 2013-03-06 2018-05-08 阿斯利康(瑞典)有限公司 表皮生长因子受体的活化突变形式的喹唑啉抑制剂
WO2015154725A1 (zh) * 2014-04-11 2015-10-15 四川海思科制药有限公司 喹唑啉衍生物及其制备方法和在医药上的应用
CN106588943B (zh) * 2015-10-19 2018-10-16 广东东阳光药业有限公司 一种egfr抑制剂的盐、晶型及其用途
US11672801B2 (en) * 2016-10-19 2023-06-13 United States Government As Represented By The Department Of Veterans Affairs Compositions and methods for treating cancer
MA46852A (fr) * 2016-11-17 2019-09-25 Univ Texas Composés à activité antitumorale contre des cellules cancéreuses porteuses de mutations egfr ou her2 exon 20
BR112021004527A2 (pt) 2018-09-14 2021-06-08 Spectrum Pharmaceuticals, Inc. kits e métodos para tratamento contra câncer

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