JP2022500456A5 - - Google Patents

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Publication number
JP2022500456A5
JP2022500456A5 JP2021514419A JP2021514419A JP2022500456A5 JP 2022500456 A5 JP2022500456 A5 JP 2022500456A5 JP 2021514419 A JP2021514419 A JP 2021514419A JP 2021514419 A JP2021514419 A JP 2021514419A JP 2022500456 A5 JP2022500456 A5 JP 2022500456A5
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JP
Japan
Prior art keywords
crystal form
compound
cancer
chemical formula
group
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021514419A
Other languages
English (en)
Japanese (ja)
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JP7554030B2 (ja
JP2022500456A (ja
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Application filed filed Critical
Priority claimed from PCT/IB2019/057720 external-priority patent/WO2020053816A1/en
Publication of JP2022500456A publication Critical patent/JP2022500456A/ja
Publication of JP2022500456A5 publication Critical patent/JP2022500456A5/ja
Application granted granted Critical
Publication of JP7554030B2 publication Critical patent/JP7554030B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2021514419A 2018-09-14 2019-09-12 キナゾリン化合物及びその塩酸塩の結晶形 Active JP7554030B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862731500P 2018-09-14 2018-09-14
US62/731,500 2018-09-14
PCT/IB2019/057720 WO2020053816A1 (en) 2018-09-14 2019-09-12 Crystalline forms of a quinazole compound and its hydrochloride salts

Publications (3)

Publication Number Publication Date
JP2022500456A JP2022500456A (ja) 2022-01-04
JP2022500456A5 true JP2022500456A5 (enExample) 2022-09-22
JP7554030B2 JP7554030B2 (ja) 2024-09-19

Family

ID=69776732

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021514419A Active JP7554030B2 (ja) 2018-09-14 2019-09-12 キナゾリン化合物及びその塩酸塩の結晶形
JP2021513941A Pending JP2022500416A (ja) 2018-09-14 2019-09-12 がんを処置するためのキットおよび方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2021513941A Pending JP2022500416A (ja) 2018-09-14 2019-09-12 がんを処置するためのキットおよび方法

Country Status (17)

Country Link
US (2) US20220040180A1 (enExample)
EP (2) EP3849964A4 (enExample)
JP (2) JP7554030B2 (enExample)
KR (2) KR20210061371A (enExample)
CN (2) CN112823153A (enExample)
AR (2) AR116669A1 (enExample)
AU (2) AU2019337640A1 (enExample)
BR (2) BR112021004527A2 (enExample)
CA (2) CA3110369A1 (enExample)
IL (2) IL281168A (enExample)
MX (2) MX2021002876A (enExample)
PH (2) PH12021550432A1 (enExample)
PY (2) PY1976960A (enExample)
SG (2) SG11202102006YA (enExample)
TW (2) TW202027750A (enExample)
UY (2) UY38374A (enExample)
WO (2) WO2020056156A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112021004527A2 (pt) 2018-09-14 2021-06-08 Spectrum Pharmaceuticals, Inc. kits e métodos para tratamento contra câncer
PE20252386A1 (es) 2019-11-21 2025-10-10 Pharma Mar Sa Metodo de tratamiento del cancer de pulmon de celulas pequenas con formulaciones de lurbinectedina
CN114642728A (zh) * 2021-06-02 2022-06-21 德琪(浙江)医药科技有限公司 mTOR抑制剂的制药用途及其药物组合物

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1596869B1 (en) * 2003-01-21 2014-06-04 New Form Pharmaceuticals Inc. Novel cocrystallization
KR100735639B1 (ko) * 2004-12-29 2007-07-04 한미약품 주식회사 암세포 성장 억제 효과를 갖는 퀴나졸린 유도체 및 이의제조방법
KR20070107151A (ko) * 2005-02-26 2007-11-06 아스트라제네카 아베 티로신 키나제 억제제로서의 퀴나졸린 유도체
CN101454302A (zh) * 2006-05-31 2009-06-10 艾博特公司 用作大麻素受体配位体的噻唑化合物及其用途
CA2659307A1 (en) 2006-07-28 2008-01-31 Synthon B.V. Crystalline erlotinib
ES2573931T3 (es) * 2007-02-21 2016-06-13 Natco Pharma Limited Nuevos polimorfismos de clorhidrato de erlotinib y método de preparación
TWI377944B (en) * 2007-06-05 2012-12-01 Hanmi Holdings Co Ltd Novel amide derivative for inhibiting the growth of cancer cells
KR101217526B1 (ko) 2010-06-11 2013-01-02 한미사이언스 주식회사 아마이드 유도체 또는 이의 약학적으로 허용 가능한 염을 포함하는 약제학적 조성물
KR101317809B1 (ko) * 2011-06-07 2013-10-16 한미약품 주식회사 암세포의 성장을 억제하는 아마이드 유도체 및 비금속염 활택제를 포함하는 약학 조성물
KR101272613B1 (ko) 2011-10-05 2013-06-10 한미사이언스 주식회사 1-(4-(4-(3,4-디클로로-2-플루오로페닐아미노)-7-메톡시퀴나졸린-6-일옥시)피페리딘-1-일)프로프-2-엔-1-온 염산염의 제조 방법 및 이에 사용되는 중간체
EP2964638B1 (en) * 2013-03-06 2017-08-09 Astrazeneca AB Quinazoline inhibitors of activating mutant forms of epidermal growth factor receptor
CN106068262B (zh) * 2014-04-11 2019-10-29 海思科医药集团股份有限公司 喹唑啉衍生物及其制备方法和在医药上的应用
US10308658B2 (en) * 2015-10-19 2019-06-04 Sunshine Lake Pharma Co., Ltd. Salt of EGFR inhibitor, crystalline form and uses thereof
US11672801B2 (en) * 2016-10-19 2023-06-13 United States Government As Represented By The Department Of Veterans Affairs Compositions and methods for treating cancer
KR102771603B1 (ko) 2016-11-17 2025-02-24 더 보드 오브 리젠츠 오브 더 유니버시티 오브 텍사스 시스템 Egfr 또는 her2 엑손 20 돌연변이를 갖는 암 세포에 대한 항종양 활성을 갖는 화합물
BR112021004527A2 (pt) 2018-09-14 2021-06-08 Spectrum Pharmaceuticals, Inc. kits e métodos para tratamento contra câncer

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