JP2022051776A5 - - Google Patents
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- Publication number
- JP2022051776A5 JP2022051776A5 JP2022008665A JP2022008665A JP2022051776A5 JP 2022051776 A5 JP2022051776 A5 JP 2022051776A5 JP 2022008665 A JP2022008665 A JP 2022008665A JP 2022008665 A JP2022008665 A JP 2022008665A JP 2022051776 A5 JP2022051776 A5 JP 2022051776A5
- Authority
- JP
- Japan
- Prior art keywords
- excipient
- powder
- content
- mass
- parts
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 239000000546 pharmaceutical excipient Substances 0.000 claims description 7
- 239000001913 cellulose Substances 0.000 claims description 5
- 229920002678 cellulose Polymers 0.000 claims description 5
- 229920002472 Starch Polymers 0.000 claims description 3
- 239000008107 starch Substances 0.000 claims description 3
- 235000019698 starch Nutrition 0.000 claims description 3
- SERLAGPUMNYUCK-DCUALPFSSA-N 1-O-alpha-D-glucopyranosyl-D-mannitol Chemical compound OC[C@@H](O)[C@@H](O)[C@H](O)[C@H](O)CO[C@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O SERLAGPUMNYUCK-DCUALPFSSA-N 0.000 claims description 2
- OWEGMIWEEQEYGQ-UHFFFAOYSA-N 100676-05-9 Natural products OC1C(O)C(O)C(CO)OC1OCC1C(O)C(O)C(O)C(OC2C(OC(O)C(O)C2O)CO)O1 OWEGMIWEEQEYGQ-UHFFFAOYSA-N 0.000 claims description 2
- GUBGYTABKSRVRQ-XLOQQCSPSA-N Alpha-Lactose Chemical compound O[C@@H]1[C@@H](O)[C@@H](O)[C@@H](CO)O[C@H]1O[C@@H]1[C@@H](CO)O[C@H](O)[C@H](O)[C@H]1O GUBGYTABKSRVRQ-XLOQQCSPSA-N 0.000 claims description 2
- 229920002261 Corn starch Polymers 0.000 claims description 2
- GUBGYTABKSRVRQ-QKKXKWKRSA-N Lactose Natural products OC[C@H]1O[C@@H](O[C@H]2[C@H](O)[C@@H](O)C(O)O[C@@H]2CO)[C@H](O)[C@@H](O)[C@H]1O GUBGYTABKSRVRQ-QKKXKWKRSA-N 0.000 claims description 2
- GUBGYTABKSRVRQ-PICCSMPSSA-N Maltose Natural products O[C@@H]1[C@@H](O)[C@H](O)[C@@H](CO)O[C@@H]1O[C@@H]1[C@@H](CO)OC(O)[C@H](O)[C@H]1O GUBGYTABKSRVRQ-PICCSMPSSA-N 0.000 claims description 2
- GUBGYTABKSRVRQ-QUYVBRFLSA-N beta-maltose Chemical compound OC[C@H]1O[C@H](O[C@H]2[C@H](O)[C@@H](O)[C@H](O)O[C@@H]2CO)[C@H](O)[C@@H](O)[C@@H]1O GUBGYTABKSRVRQ-QUYVBRFLSA-N 0.000 claims description 2
- 239000008120 corn starch Substances 0.000 claims description 2
- 239000000905 isomalt Substances 0.000 claims description 2
- 235000010439 isomalt Nutrition 0.000 claims description 2
- HPIGCVXMBGOWTF-UHFFFAOYSA-N isomaltol Natural products CC(=O)C=1OC=CC=1O HPIGCVXMBGOWTF-UHFFFAOYSA-N 0.000 claims description 2
- 239000008101 lactose Substances 0.000 claims description 2
- 229940100486 rice starch Drugs 0.000 claims description 2
- 239000000843 powder Substances 0.000 claims 4
- 239000003795 chemical substances by application Substances 0.000 claims 1
- 239000000845 maltitol Substances 0.000 claims 1
- VQHSOMBJVWLPSR-WUJBLJFYSA-N maltitol Chemical compound OC[C@H](O)[C@@H](O)[C@@H]([C@H](O)CO)O[C@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O VQHSOMBJVWLPSR-WUJBLJFYSA-N 0.000 claims 1
- 235000010449 maltitol Nutrition 0.000 claims 1
- 229940035436 maltitol Drugs 0.000 claims 1
- 239000002994 raw material Substances 0.000 claims 1
- 240000003183 Manihot esculenta Species 0.000 description 1
- 235000016735 Manihot esculenta subsp esculenta Nutrition 0.000 description 1
- 241000278713 Theora Species 0.000 description 1
- 230000000052 comparative effect Effects 0.000 description 1
- -1 martitol Chemical compound 0.000 description 1
- 239000004848 polyfunctional curative Substances 0.000 description 1
- 229920001592 potato starch Polymers 0.000 description 1
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2016128150 | 2016-06-28 | ||
| JP2016128150 | 2016-06-28 | ||
| PCT/JP2017/023475 WO2018003762A1 (ja) | 2016-06-28 | 2017-06-27 | 賦形剤及び錠剤 |
| JP2018525160A JP7020688B2 (ja) | 2016-06-28 | 2017-06-27 | 賦形剤及び錠剤 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018525160A Division JP7020688B2 (ja) | 2016-06-28 | 2017-06-27 | 賦形剤及び錠剤 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022051776A JP2022051776A (ja) | 2022-04-01 |
| JP2022051776A5 true JP2022051776A5 (cg-RX-API-DMAC7.html) | 2022-06-01 |
| JP7239119B2 JP7239119B2 (ja) | 2023-03-14 |
Family
ID=60785986
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018525160A Active JP7020688B2 (ja) | 2016-06-28 | 2017-06-27 | 賦形剤及び錠剤 |
| JP2022008665A Active JP7239119B2 (ja) | 2016-06-28 | 2022-01-24 | 賦形剤及び錠剤 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018525160A Active JP7020688B2 (ja) | 2016-06-28 | 2017-06-27 | 賦形剤及び錠剤 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20190201345A1 (cg-RX-API-DMAC7.html) |
| JP (2) | JP7020688B2 (cg-RX-API-DMAC7.html) |
| KR (1) | KR20190022709A (cg-RX-API-DMAC7.html) |
| CN (1) | CN109414051A (cg-RX-API-DMAC7.html) |
| WO (1) | WO2018003762A1 (cg-RX-API-DMAC7.html) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP4069203A1 (en) * | 2019-12-06 | 2022-10-12 | Synthon B.V. | Pharmaceutical composition comprising eltrombopag bis(monoethanolamine) |
| CN111035620B (zh) * | 2019-12-25 | 2021-08-27 | 广州莱可福生物科技有限公司 | 一种辅料组合物、植物甾醇复合营养素咀嚼片及其制备方法 |
| US20220015993A1 (en) * | 2020-07-14 | 2022-01-20 | Johnson & Johnson Consumer Inc. | Solid cleansing composition presenting controlled disintegration |
| CN113388341B (zh) * | 2021-06-17 | 2023-09-15 | 安徽精公检测检验中心有限公司 | 一种固体粘结剂及其制备方法和应用 |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK0979865T3 (da) | 1998-07-17 | 2002-08-19 | Procter & Gamble | Detergenttablet |
| CN1768741A (zh) * | 1999-05-21 | 2006-05-10 | 橘生药品工业株式会社 | 即释型口服用药物组合物 |
| JP4588818B2 (ja) * | 1999-09-16 | 2010-12-01 | 日本化学機械製造株式会社 | 錠剤用賦形剤及び錠剤 |
| KR100496749B1 (ko) * | 2000-07-05 | 2005-06-22 | 아사히 가세이 가부시키가이샤 | 셀룰로스 분말 |
| ATE454132T1 (de) * | 2003-01-21 | 2010-01-15 | Nippon Shinyaku Co Ltd | Rasch in der mundhöhle schmelzende tablette |
| JP5219508B2 (ja) * | 2005-05-18 | 2013-06-26 | 大日本住友製薬株式会社 | ドロキシドパを含有する安定な錠剤 |
| JP5120652B2 (ja) * | 2006-03-30 | 2013-01-16 | 日本臓器製薬株式会社 | 固形医薬製剤 |
| JP2008037853A (ja) * | 2006-08-01 | 2008-02-21 | Higuchi Shokai:Kk | イソマルトを含有する速崩壊性医薬品固形製剤 |
| EP2050448A4 (en) * | 2006-08-08 | 2012-01-04 | Kissei Pharmaceutical | Mouth-dropping tray with masked bitter taste and method of preparation |
| EP2062599A4 (en) * | 2006-09-14 | 2013-03-27 | Astellas Pharma Inc | ORAL DISSOLVING TABLET AND METHOD FOR THE PRODUCTION THEREOF |
| CA2715760C (en) * | 2008-02-21 | 2017-06-13 | Mitsubishi Tanabe Pharma Corporation | Solid preparation for oral administration of cariprazine hydrochloride |
| WO2010025796A1 (en) * | 2008-09-04 | 2010-03-11 | Cargill Incorporated | Tabletting of ervthritol |
| JP5637624B2 (ja) * | 2009-02-12 | 2014-12-10 | 富士化学工業株式会社 | 崩壊性粒子組成物及びそれを用いた速崩壊性圧縮成型物 |
| WO2012001977A1 (ja) * | 2010-06-29 | 2012-01-05 | 富士化学工業株式会社 | 崩壊性組成物及び易崩壊性圧縮成型物 |
| JO3753B1 (ar) * | 2011-10-14 | 2021-01-31 | Otsuka Pharma Co Ltd | قرص يتألف من 7-[4-(4-بينزو[بي]ثيوفين-4-ايل-ببرازين-1-1ايل)بوتكسيل]-1اتش-كوينولين-2-وان أو ملح منه |
| JPWO2017142001A1 (ja) * | 2016-02-16 | 2018-12-06 | テイカ製薬株式会社 | 口腔内速崩壊性錠剤用造粒物 |
-
2017
- 2017-06-27 KR KR1020197002187A patent/KR20190022709A/ko not_active Ceased
- 2017-06-27 US US16/314,219 patent/US20190201345A1/en not_active Abandoned
- 2017-06-27 JP JP2018525160A patent/JP7020688B2/ja active Active
- 2017-06-27 CN CN201780040620.XA patent/CN109414051A/zh active Pending
- 2017-06-27 WO PCT/JP2017/023475 patent/WO2018003762A1/ja not_active Ceased
-
2022
- 2022-01-24 JP JP2022008665A patent/JP7239119B2/ja active Active
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