JP2021535159A5 - - Google Patents

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Publication number
JP2021535159A5
JP2021535159A5 JP2021510960A JP2021510960A JP2021535159A5 JP 2021535159 A5 JP2021535159 A5 JP 2021535159A5 JP 2021510960 A JP2021510960 A JP 2021510960A JP 2021510960 A JP2021510960 A JP 2021510960A JP 2021535159 A5 JP2021535159 A5 JP 2021535159A5
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JP
Japan
Prior art keywords
compound
formula
alkyl
group
haloalkyl
Prior art date
Application number
JP2021510960A
Other languages
English (en)
Japanese (ja)
Other versions
JP7583710B2 (ja
JP2021535159A (ja
JPWO2020046991A5 (https=
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Publication date
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Priority claimed from PCT/US2019/048408 external-priority patent/WO2020046991A1/en
Publication of JP2021535159A publication Critical patent/JP2021535159A/ja
Publication of JP2021535159A5 publication Critical patent/JP2021535159A5/ja
Publication of JPWO2020046991A5 publication Critical patent/JPWO2020046991A5/ja
Priority to JP2024192796A priority Critical patent/JP2025016676A/ja
Application granted granted Critical
Publication of JP7583710B2 publication Critical patent/JP7583710B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2021510960A 2018-08-27 2019-08-27 スパイン形成のためのファシン結合化合物 Active JP7583710B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024192796A JP2025016676A (ja) 2018-08-27 2024-11-01 スパイン形成のためのファシン結合化合物

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201862723381P 2018-08-27 2018-08-27
US62/723,381 2018-08-27
US201862726904P 2018-09-04 2018-09-04
US62/726,904 2018-09-04
US201862785435P 2018-12-27 2018-12-27
US62/785,435 2018-12-27
PCT/US2019/048408 WO2020046991A1 (en) 2018-08-27 2019-08-27 Fascin binding compounds for spinogenesis

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024192796A Division JP2025016676A (ja) 2018-08-27 2024-11-01 スパイン形成のためのファシン結合化合物

Publications (4)

Publication Number Publication Date
JP2021535159A JP2021535159A (ja) 2021-12-16
JP2021535159A5 true JP2021535159A5 (https=) 2022-08-25
JPWO2020046991A5 JPWO2020046991A5 (https=) 2022-08-25
JP7583710B2 JP7583710B2 (ja) 2024-11-14

Family

ID=69644570

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021510960A Active JP7583710B2 (ja) 2018-08-27 2019-08-27 スパイン形成のためのファシン結合化合物
JP2024192796A Pending JP2025016676A (ja) 2018-08-27 2024-11-01 スパイン形成のためのファシン結合化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2024192796A Pending JP2025016676A (ja) 2018-08-27 2024-11-01 スパイン形成のためのファシン結合化合物

Country Status (7)

Country Link
US (2) US20210330646A1 (https=)
EP (1) EP3843846A4 (https=)
JP (2) JP7583710B2 (https=)
CN (1) CN112912141B (https=)
AU (1) AU2019329835B2 (https=)
CA (1) CA3110877A1 (https=)
WO (1) WO2020046991A1 (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2018312558B2 (en) 2017-08-02 2022-09-29 Spinogenix, Inc. Benzothiazole and related compounds
HUE072464T2 (hu) 2019-01-31 2025-11-28 Spinogenix Inc Spinogenézis egy promoterének szilárd formái
CA3189027A1 (en) 2020-07-11 2022-01-20 Pfizer Inc. Antiviral heteroaryl ketone derivatives
US11351149B2 (en) 2020-09-03 2022-06-07 Pfizer Inc. Nitrile-containing antiviral compounds
EP4294391A4 (en) * 2021-02-22 2024-12-18 Spinogenix, Inc. METHODS OF TREATING SPINAL CORD INJURY OR DAMAGE
JP2024510632A (ja) * 2021-03-23 2024-03-08 スピノジェニックス, インコーポレイテッド スパイン形成のためのある特定のファスシン結合化合物
WO2024211310A1 (en) * 2023-04-03 2024-10-10 Spinogenix, Inc. Methods of dosing spinogenic compounds
CN121773104A (zh) * 2023-06-30 2026-03-31 北京双鹤润创科技有限公司 肌成束蛋白抑制剂
WO2025184576A1 (en) * 2024-02-29 2025-09-04 Spinogenix, Inc. Methods for prevention and treatment of depression

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3845770A (en) 1972-06-05 1974-11-05 Alza Corp Osmatic dispensing device for releasing beneficial agent
US4326525A (en) 1980-10-14 1982-04-27 Alza Corporation Osmotic device that improves delivery properties of agent in situ
US5364620A (en) 1983-12-22 1994-11-15 Elan Corporation, Plc Controlled absorption diltiazem formulation for once daily administration
US5023252A (en) 1985-12-04 1991-06-11 Conrex Pharmaceutical Corporation Transdermal and trans-membrane delivery of drugs
US4992445A (en) 1987-06-12 1991-02-12 American Cyanamid Co. Transdermal delivery of pharmaceuticals
US5001139A (en) 1987-06-12 1991-03-19 American Cyanamid Company Enchancers for the transdermal flux of nivadipine
US4902514A (en) 1988-07-21 1990-02-20 Alza Corporation Dosage form for administering nilvadipine for treating cardiovascular symptoms
AU2012239977B9 (en) 2011-04-07 2016-11-17 Sloan-Kettering Institute For Cancer Research Migrastatins and uses thereof
WO2013013240A2 (en) 2011-07-21 2013-01-24 Theracrine, Inc. Macrocyclic compounds and related compositons and methods of use
EP2755974A1 (en) * 2011-09-14 2014-07-23 Proximagen Limited New enzyme inhibitor compounds
CA3139033A1 (en) 2012-08-22 2014-02-27 Cornell University Methods for inhibiting fascin
CN111349087B (zh) * 2014-02-20 2023-07-14 康奈尔大学 用于抑制肌成束蛋白的化合物和方法
CA3010445A1 (en) 2016-01-05 2017-07-13 The Regents Of The University Of California Benzothiazole amphiphiles
TWI586367B (zh) 2016-03-28 2017-06-11 蔡懷楨 磷酸甘油酯激酶增加神經突生長及/或治療神經性疾病的用途
AU2018312558B2 (en) 2017-08-02 2022-09-29 Spinogenix, Inc. Benzothiazole and related compounds

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