JP2021519285A5 - - Google Patents

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Publication number
JP2021519285A5
JP2021519285A5 JP2020551481A JP2020551481A JP2021519285A5 JP 2021519285 A5 JP2021519285 A5 JP 2021519285A5 JP 2020551481 A JP2020551481 A JP 2020551481A JP 2020551481 A JP2020551481 A JP 2020551481A JP 2021519285 A5 JP2021519285 A5 JP 2021519285A5
Authority
JP
Japan
Prior art keywords
cancer
combination
pharmaceuticals
fluorophenyl
fluoro
Prior art date
Application number
JP2020551481A
Other languages
English (en)
Japanese (ja)
Other versions
JPWO2019186488A5 (https=
JP2021519285A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2019/052601 external-priority patent/WO2019186488A1/en
Publication of JP2021519285A publication Critical patent/JP2021519285A/ja
Publication of JPWO2019186488A5 publication Critical patent/JPWO2019186488A5/ja
Publication of JP2021519285A5 publication Critical patent/JP2021519285A5/ja
Pending legal-status Critical Current

Links

JP2020551481A 2018-03-30 2019-03-29 ダブラフェニブ、トラメチニブ及びerk阻害剤を含む医薬品の三重の組合せ Pending JP2021519285A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862650744P 2018-03-30 2018-03-30
US62/650,744 2018-03-30
PCT/IB2019/052601 WO2019186488A1 (en) 2018-03-30 2019-03-29 A triple pharmaceutical combination comprising dabrafenib, trametinib and an erk inhibitor

Publications (3)

Publication Number Publication Date
JP2021519285A JP2021519285A (ja) 2021-08-10
JPWO2019186488A5 JPWO2019186488A5 (https=) 2022-04-06
JP2021519285A5 true JP2021519285A5 (https=) 2022-04-06

Family

ID=66397350

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020551481A Pending JP2021519285A (ja) 2018-03-30 2019-03-29 ダブラフェニブ、トラメチニブ及びerk阻害剤を含む医薬品の三重の組合せ

Country Status (13)

Country Link
US (1) US20210121460A1 (https=)
EP (1) EP3773586A1 (https=)
JP (1) JP2021519285A (https=)
KR (1) KR20200138303A (https=)
CN (1) CN111936141A (https=)
AU (1) AU2019246719B2 (https=)
BR (1) BR112020019577A2 (https=)
CA (1) CA3094780A1 (https=)
CL (1) CL2020002505A1 (https=)
IL (1) IL277380A (https=)
MX (1) MX2020010231A (https=)
RU (1) RU2020135055A (https=)
WO (1) WO2019186488A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021171261A1 (en) * 2020-02-28 2021-09-02 Novartis Ag A triple pharmaceutical combination comprising dabrafenib, an erk inhibitor and a shp2 inhibitor
EP4110341A2 (en) * 2020-02-28 2023-01-04 Novartis AG A triple pharmaceutical combination comprising dabrafenib, an erk inhibitor and a raf inhibitor

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2005252110B2 (en) 2004-06-11 2008-09-04 Shionogi & Co., Ltd. 5-amino-2,4,7-trioxo-3,4,7,8-tetrahydro-2H-pyrido[2,3-D] pyrimidine derivatives and related compounds for the treatment of cancer
UA103319C2 (en) 2008-05-06 2013-10-10 Глаксосмитклайн Ллк Thiazole- and oxazole-benzene sulfonamide compounds
AU2014342338B2 (en) * 2013-11-01 2016-12-01 Novartis Ag Aminoheteroaryl benzamides as kinase inhibitors
CN108368171A (zh) * 2015-07-10 2018-08-03 根马布股份公司 用于癌症治疗的axl特异性抗体-药物缀合物
AU2017329090B9 (en) * 2016-09-19 2019-09-05 Novartis Ag Therapeutic combinations comprising a RAF inhibitor and a ERK inhibitor

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