JP2021511299A5 - - Google Patents
Info
- Publication number
- JP2021511299A5 JP2021511299A5 JP2020538535A JP2020538535A JP2021511299A5 JP 2021511299 A5 JP2021511299 A5 JP 2021511299A5 JP 2020538535 A JP2020538535 A JP 2020538535A JP 2020538535 A JP2020538535 A JP 2020538535A JP 2021511299 A5 JP2021511299 A5 JP 2021511299A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- salt
- membered heteroaryl
- heteroaryl ring
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2023162922A JP7744955B2 (ja) | 2018-01-10 | 2023-09-26 | 可溶性グアニル酸シクラーゼ刺激剤を調製するための新規のプロセスおよび中間体 |
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862615678P | 2018-01-10 | 2018-01-10 | |
| US62/615,678 | 2018-01-10 | ||
| PCT/CN2018/076982 WO2019161534A1 (en) | 2018-02-22 | 2018-02-22 | Novel processes and intermediates for preparation of soluble guanylate cyclase stimulators |
| CNPCT/CN2018/076982 | 2018-02-22 | ||
| PCT/US2019/013060 WO2019140095A1 (en) | 2018-01-10 | 2019-01-10 | Novel processes and intermediates for the preparation of soluble guanylate cyclase stimulators |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023162922A Division JP7744955B2 (ja) | 2018-01-10 | 2023-09-26 | 可溶性グアニル酸シクラーゼ刺激剤を調製するための新規のプロセスおよび中間体 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021511299A JP2021511299A (ja) | 2021-05-06 |
| JP2021511299A5 true JP2021511299A5 (OSRAM) | 2022-01-19 |
| JP7357621B2 JP7357621B2 (ja) | 2023-10-06 |
Family
ID=65279655
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020538535A Active JP7357621B2 (ja) | 2018-01-10 | 2019-01-10 | 可溶性グアニル酸シクラーゼ刺激剤を調製するための新規のプロセスおよび中間体 |
| JP2023162922A Active JP7744955B2 (ja) | 2018-01-10 | 2023-09-26 | 可溶性グアニル酸シクラーゼ刺激剤を調製するための新規のプロセスおよび中間体 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023162922A Active JP7744955B2 (ja) | 2018-01-10 | 2023-09-26 | 可溶性グアニル酸シクラーゼ刺激剤を調製するための新規のプロセスおよび中間体 |
Country Status (16)
| Country | Link |
|---|---|
| US (5) | US11274096B2 (OSRAM) |
| EP (3) | EP4249469A3 (OSRAM) |
| JP (2) | JP7357621B2 (OSRAM) |
| KR (3) | KR20250048609A (OSRAM) |
| CN (3) | CN111902410B (OSRAM) |
| AU (3) | AU2019206560B2 (OSRAM) |
| CA (1) | CA3087943A1 (OSRAM) |
| CL (3) | CL2020001814A1 (OSRAM) |
| ES (1) | ES2963447T3 (OSRAM) |
| IL (3) | IL314714A (OSRAM) |
| JO (1) | JOP20200165A1 (OSRAM) |
| MA (2) | MA51565A (OSRAM) |
| MX (3) | MX2020007364A (OSRAM) |
| SG (1) | SG11202006311SA (OSRAM) |
| TW (2) | TWI888947B (OSRAM) |
| WO (1) | WO2019140095A1 (OSRAM) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2963563T3 (es) | 2016-07-07 | 2024-03-27 | Cyclerion Therapeutics Inc | Procesos novedosos para preparar estimuladores de guanilato ciclasa soluble |
| EP4249469A3 (en) | 2018-01-10 | 2023-12-27 | Cyclerion Therapeutics, Inc. | Novel processes and intermediates for the preparation of soluble guanylate cyclase stimulators |
| WO2024131860A1 (zh) * | 2022-12-21 | 2024-06-27 | 广东东阳光药业股份有限公司 | 氟取代的吲唑化合物的晶型及其用途 |
| AU2023412228A1 (en) * | 2022-12-21 | 2025-07-03 | Sunshine Lake Pharma Co., Ltd. | Crystal form of fluorine-substituted indazole compound and use thereof |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012003405A1 (en) * | 2010-06-30 | 2012-01-05 | Ironwood Pharmaceuticals, Inc. | Sgc stimulators |
| SI2970243T1 (sl) * | 2013-03-15 | 2020-04-30 | Cyclerion Therapeutics, Inc. | SGC stimulatorji |
| EP3094327A1 (en) * | 2014-01-13 | 2016-11-23 | Ironwood Pharmaceuticals, Inc. | USE OF sGC STIMULATORS FOR THE TREATMENT OF NEUROMUSCULAR DISORDERS |
| JP2017527605A (ja) * | 2014-09-17 | 2017-09-21 | アイアンウッド ファーマシューティカルズ インコーポレイテッド | ｓＧＣ刺激剤 |
| CA2959757A1 (en) | 2014-09-17 | 2016-03-24 | Ironwood Pharmaceuticals, Inc. | Pyrazole derivatives as sgc stimulators |
| EA201891315A1 (ru) * | 2015-11-30 | 2018-12-28 | Айронвуд Фармасьютикалз, Инк. | Твердые дисперсии, содержащие стимулятор sgc |
| SG10202100168XA (en) | 2016-07-07 | 2021-02-25 | Cyclerion Therapeutics Inc | Novel processes for preparation of soluble guanylate cyclase stimulators |
| ES2963563T3 (es) | 2016-07-07 | 2024-03-27 | Cyclerion Therapeutics Inc | Procesos novedosos para preparar estimuladores de guanilato ciclasa soluble |
| EP4249469A3 (en) | 2018-01-10 | 2023-12-27 | Cyclerion Therapeutics, Inc. | Novel processes and intermediates for the preparation of soluble guanylate cyclase stimulators |
-
2019
- 2019-01-10 EP EP23187776.2A patent/EP4249469A3/en active Pending
- 2019-01-10 KR KR1020257010603A patent/KR20250048609A/ko active Pending
- 2019-01-10 CN CN201980017700.2A patent/CN111902410B/zh active Active
- 2019-01-10 AU AU2019206560A patent/AU2019206560B2/en active Active
- 2019-01-10 JO JOP/2020/0165A patent/JOP20200165A1/ar unknown
- 2019-01-10 IL IL314714A patent/IL314714A/en unknown
- 2019-01-10 MA MA051565A patent/MA51565A/fr unknown
- 2019-01-10 CN CN202410363184.1A patent/CN118221665A/zh active Pending
- 2019-01-10 KR KR1020207022640A patent/KR102739727B1/ko active Active
- 2019-01-10 US US16/961,109 patent/US11274096B2/en active Active
- 2019-01-10 MX MX2020007364A patent/MX2020007364A/es unknown
- 2019-01-10 CN CN202410363182.2A patent/CN118184645A/zh active Pending
- 2019-01-10 EP EP19703440.8A patent/EP3737679B1/en active Active
- 2019-01-10 MA MA71753A patent/MA71753A/fr unknown
- 2019-01-10 IL IL275748A patent/IL275748B2/en unknown
- 2019-01-10 SG SG11202006311SA patent/SG11202006311SA/en unknown
- 2019-01-10 WO PCT/US2019/013060 patent/WO2019140095A1/en not_active Ceased
- 2019-01-10 KR KR1020247039985A patent/KR20250002720A/ko active Pending
- 2019-01-10 ES ES19703440T patent/ES2963447T3/es active Active
- 2019-01-10 CA CA3087943A patent/CA3087943A1/en active Pending
- 2019-01-10 JP JP2020538535A patent/JP7357621B2/ja active Active
- 2019-01-10 IL IL319883A patent/IL319883A/en unknown
- 2019-01-10 TW TW112138274A patent/TWI888947B/zh active
- 2019-01-10 TW TW108101044A patent/TWI821237B/zh active
- 2019-01-10 EP EP25174051.0A patent/EP4570797A3/en active Pending
-
2020
- 2020-07-07 CL CL2020001814A patent/CL2020001814A1/es unknown
- 2020-07-13 MX MX2023000045A patent/MX2023000045A/es unknown
- 2020-07-13 MX MX2023000044A patent/MX2023000044A/es unknown
-
2021
- 2021-10-08 US US17/497,352 patent/US11708361B2/en active Active
-
2022
- 2022-04-08 CL CL2022000904A patent/CL2022000904A1/es unknown
- 2022-04-08 CL CL2022000907A patent/CL2022000907A1/es unknown
-
2023
- 2023-04-28 US US18/140,966 patent/US12030874B2/en active Active
- 2023-09-26 JP JP2023162922A patent/JP7744955B2/ja active Active
- 2023-11-22 AU AU2023270260A patent/AU2023270260B2/en active Active
-
2024
- 2024-05-22 US US18/671,182 patent/US12275724B2/en active Active
-
2025
- 2025-03-31 AU AU2025202281A patent/AU2025202281A1/en active Pending
- 2025-04-11 US US19/176,742 patent/US20250361228A1/en active Pending
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