JP2021138710A5 - - Google Patents

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Publication number
JP2021138710A5
JP2021138710A5 JP2021081095A JP2021081095A JP2021138710A5 JP 2021138710 A5 JP2021138710 A5 JP 2021138710A5 JP 2021081095 A JP2021081095 A JP 2021081095A JP 2021081095 A JP2021081095 A JP 2021081095A JP 2021138710 A5 JP2021138710 A5 JP 2021138710A5
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JP
Japan
Prior art keywords
drug
eye diseases
diabetic
rpe
pvr
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Pending
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JP2021081095A
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English (en)
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JP2021138710A (ja
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Priority claimed from JP2019517058A external-priority patent/JP2019531296A/ja
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Publication of JP2021138710A publication Critical patent/JP2021138710A/ja
Publication of JP2021138710A5 publication Critical patent/JP2021138710A5/ja
Priority to JP2023100597A priority Critical patent/JP2023116748A/ja
Pending legal-status Critical Current

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Claims (2)

  1. 有効量の、式I:
    Figure 2021138710
    で示される化合物を含む、網膜色素上皮(RPE)細胞の傷害を逆転させ、眼血流を向上させることにより眼疾患を処置するための医薬であって、
    眼疾患が、増殖性硝子体網膜症(PVR)、ブドウ膜炎、加齢黄斑変性症(AMD)の初期事象、糖尿病網膜症(DR)および糖尿病黄斑浮腫(DME)からなる群より選択される、医薬。
  2. 該医薬が1日1〜3回経口投与され、式Iで示される化合物の量が、各経口投与において0.5〜50mgである、請求項1に記載の医薬。
JP2021081095A 2016-09-29 2021-05-12 眼疾患の処置方法 Pending JP2021138710A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023100597A JP2023116748A (ja) 2016-09-29 2023-06-20 眼疾患の処置方法

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662401725P 2016-09-29 2016-09-29
US62/401,725 2016-09-29
JP2019517058A JP2019531296A (ja) 2016-09-29 2017-09-29 眼疾患の処置方法

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JP2019517058A Division JP2019531296A (ja) 2016-09-29 2017-09-29 眼疾患の処置方法

Related Child Applications (1)

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JP2023100597A Division JP2023116748A (ja) 2016-09-29 2023-06-20 眼疾患の処置方法

Publications (2)

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JP2021138710A JP2021138710A (ja) 2021-09-16
JP2021138710A5 true JP2021138710A5 (ja) 2021-12-23

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ID=61688114

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JP2019517058A Withdrawn JP2019531296A (ja) 2016-09-29 2017-09-29 眼疾患の処置方法
JP2021081095A Pending JP2021138710A (ja) 2016-09-29 2021-05-12 眼疾患の処置方法
JP2023100597A Pending JP2023116748A (ja) 2016-09-29 2023-06-20 眼疾患の処置方法

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JP2019517058A Withdrawn JP2019531296A (ja) 2016-09-29 2017-09-29 眼疾患の処置方法

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JP2023100597A Pending JP2023116748A (ja) 2016-09-29 2023-06-20 眼疾患の処置方法

Country Status (8)

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US (1) US11045435B2 (ja)
EP (1) EP3518913A4 (ja)
JP (3) JP2019531296A (ja)
KR (1) KR102341446B1 (ja)
CN (1) CN109789115A (ja)
CA (1) CA3038845C (ja)
TW (1) TWI765917B (ja)
WO (1) WO2018059543A1 (ja)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN110585196B (zh) * 2018-06-13 2022-11-04 郭涛 一种治疗及预防眼科疾病的药物及其应用

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20060074100A1 (en) * 2002-11-12 2006-04-06 Klimko Peter G Histone deacetylase inhibitors for the treatment of ocular neovascular or edematous disorders and diseases
US20050074497A1 (en) * 2003-04-09 2005-04-07 Schultz Clyde L. Hydrogels used to deliver medicaments to the eye for the treatment of posterior segment diseases
JP4873904B2 (ja) * 2005-08-22 2012-02-08 国立大学法人弘前大学 眼血管血流障害改善剤
CN101646460A (zh) 2007-03-28 2010-02-10 参天制药株式会社 含有具有组蛋白脱乙酰化酶抑制作用的化合物作为有效成分的降眼压剂
CA2630174A1 (en) * 2007-05-02 2008-11-02 Mitchell Alan Winnik Loading quantum dots into thermo-responsive microgels by reversible transfer from organic solvents to water
US20110014294A1 (en) 2008-03-03 2011-01-20 Pharmalight Inc. Stimulation of ocular retrobulbar blood flow using ocular irritants
NZ591820A (en) * 2008-08-27 2012-12-21 Leo Pharma As Pyridine derivatives as vegfr-2 receptor and protein tyrosine kinase inhibitors
ES2473792T3 (es) * 2009-04-03 2014-07-07 Naturewise Biotech & Medicals Corporation Compuestos cin�micos y derivados de los mismos para la inhibición de la histona desacetilasa
US7994357B2 (en) * 2009-04-03 2011-08-09 Naturewise Biotech & Medicals Corporation Cinamic compounds and derivatives therefrom for the inhibition of histone deacetylase
EP2277387B1 (en) * 2009-07-22 2016-10-19 NatureWise Biotech & Medicals Corporation New use of histone deacetylase inhibitors in changing mrjp3 protein in royal jelly
KR102165421B1 (ko) * 2011-05-09 2020-10-14 알레그로 파마슈티칼스, 인코포레이티드. 인테그린 수용체 길항물질 및 이의 사용 방법
CA2946086A1 (en) * 2014-04-17 2015-10-22 Teraclon Idf, S.L. Recombinant monoclonal antibodies vnar neutralizing the vascular endothelial growth factor (vegf)
US9956254B2 (en) * 2015-02-26 2018-05-01 Naturewise Biotech & Medicals Corporation Extract of taiwanese propolis for treating ocular diseases

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