JP2020529988A5 - - Google Patents

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JP2020529988A5
JP2020529988A5 JP2020505233A JP2020505233A JP2020529988A5 JP 2020529988 A5 JP2020529988 A5 JP 2020529988A5 JP 2020505233 A JP2020505233 A JP 2020505233A JP 2020505233 A JP2020505233 A JP 2020505233A JP 2020529988 A5 JP2020529988 A5 JP 2020529988A5
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Japan
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JP2020505233A
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Japanese (ja)
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JP2020529988A (ja
JP7498108B2 (ja
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Priority claimed from PCT/US2018/045175 external-priority patent/WO2019028357A1/en
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JP2020505233A 2017-08-03 2018-08-03 医学的障害の予防および治療のための化合物およびその使用 Active JP7498108B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762540860P 2017-08-03 2017-08-03
US62/540,860 2017-08-03
PCT/US2018/045175 WO2019028357A1 (en) 2017-08-03 2018-08-03 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF MEDICAL DISORDERS AND USES THEREOF

Publications (3)

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JP2020529988A JP2020529988A (ja) 2020-10-15
JP2020529988A5 true JP2020529988A5 (https=) 2021-09-09
JP7498108B2 JP7498108B2 (ja) 2024-06-11

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JP2020505233A Active JP7498108B2 (ja) 2017-08-03 2018-08-03 医学的障害の予防および治療のための化合物およびその使用

Country Status (12)

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US (3) US11583530B2 (https=)
EP (1) EP3661502A4 (https=)
JP (1) JP7498108B2 (https=)
KR (1) KR102692840B1 (https=)
CN (1) CN111032039B (https=)
AU (1) AU2018309085B2 (https=)
BR (1) BR112020001698A2 (https=)
CA (1) CA3069745A1 (https=)
IL (1) IL272097B2 (https=)
MX (1) MX2020001256A (https=)
WO (1) WO2019028357A1 (https=)
ZA (1) ZA202000375B (https=)

Families Citing this family (9)

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Publication number Priority date Publication date Assignee Title
TWI744300B (zh) * 2016-03-23 2021-11-01 里爾中央醫學中心 改良性熱處理的血小板顆粒裂解液在製備用於治療神經系統疾病的組合物的用途
AU2018308088B2 (en) 2017-07-25 2025-05-29 Truebinding, Inc. Treating cancer by blocking the interaction of TIM-3 and its ligand
EP3661502A4 (en) 2017-08-03 2020-12-02 Galectin Sciences, LLC COMPOUNDS FOR THE PREVENTION AND TREATMENT OF MEDICAL CONDITIONS AND THEIR USES
AU2020214796A1 (en) 2019-01-30 2021-07-29 Truebinding, Inc. Anti-Gal3 antibodies and uses thereof
WO2021242776A2 (en) 2020-05-26 2021-12-02 Truebinding, Inc. Methods of treating inflammatory diseases by blocking galectin-3
WO2022261113A2 (en) * 2021-06-08 2022-12-15 Truebinding, Inc. Anti-gal3 antibodies and methods of use for insulin resistance
CN113476442A (zh) * 2021-07-28 2021-10-08 上海交通大学医学院附属第九人民医院 化合物gb-0139在治疗心肌梗死后心肌过度纤维化的药物中的应用
GB2631509A (en) * 2023-07-04 2025-01-08 Univ Liverpool Compositions
GB2631507A (en) * 2023-07-04 2025-01-08 Univ Liverpool Compositions

Family Cites Families (15)

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Publication number Priority date Publication date Assignee Title
AT377586B (de) * 1981-06-30 1985-04-10 Erba Farmitalia Verfahren zur herstellung von substituierten pyrrolo-(2,1-b)-chinazolinen und pyrido(2,1-b)chinazolinen
ES8501397A1 (es) * 1982-08-05 1984-11-16 Erba Farmitalia "procedimiento para preparar derivados de quinazolina"
SE0100172D0 (sv) * 2001-01-22 2001-01-22 Ulf Nilsson New inhibitors against galectins
BR0206844A (pt) 2001-01-31 2005-07-12 Synaptic Pharma Corp Uso de antagonistas do receptor gal3 para o tratamento de depressão e/ou ansiedade e compostos usados em tais métodos
US20030078271A1 (en) 2001-01-31 2003-04-24 Blackburn Thomas P. Use of GAL3 receptor antagonists for the treatment of depression and/or anxiety and compounds useful in such methods
ES2278197T3 (es) * 2002-07-09 2007-08-01 Actelion Pharmaceuticals Ltd. Derivados de 7,8,9,10-tetrahidro-6h-azepino, 6,7,8,9-tetrahidro-pirido y 2,3-dihidro-2h-pirrolo(1,2-b)-quinazolinona.
US7220775B2 (en) 2002-08-07 2007-05-22 H. Lundbeck A/S Compound useful for the treatment of neuropathic pain
DE10304141B4 (de) * 2003-02-03 2006-03-09 Hf Arzneimittelforschung Gmbh Verfahren zur Herstellung von Chinazolin-Alkaloiden
WO2012158913A2 (en) * 2011-05-17 2012-11-22 Discoverybiomed Inc. Treating protein folding disorders with small molecule cftr correctors
RU2606635C2 (ru) * 2011-07-13 2017-01-10 Сантен Фармасьютикал Ко., Лтд. Новое соединение, проявляющее ингибиторную активность в отношении parp
WO2016004093A2 (en) 2014-07-01 2016-01-07 Stealth Biotherapeutics Corp Therapeutic compositions including galectin-3 inhibitors and uses thereof
JP6904906B2 (ja) * 2015-01-30 2021-07-21 ガレクト・バイオテック・エイビイ ガレクチンの新規なガラクトシド阻害剤
CN105272986A (zh) * 2015-06-15 2016-01-27 厦门医学高等专科学校 一种可抑制乙酰胆碱酯酶活性的化合物或其制备方法和应用
CN106220631B (zh) * 2016-07-26 2019-02-05 中山大学 一种7位氟取代Isaindigotone衍生物及其制备方法和在制备抗癌药物中的应用
EP3661502A4 (en) 2017-08-03 2020-12-02 Galectin Sciences, LLC COMPOUNDS FOR THE PREVENTION AND TREATMENT OF MEDICAL CONDITIONS AND THEIR USES

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