JP2020512373A5 - - Google Patents

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Publication number
JP2020512373A5
JP2020512373A5 JP2019553478A JP2019553478A JP2020512373A5 JP 2020512373 A5 JP2020512373 A5 JP 2020512373A5 JP 2019553478 A JP2019553478 A JP 2019553478A JP 2019553478 A JP2019553478 A JP 2019553478A JP 2020512373 A5 JP2020512373 A5 JP 2020512373A5
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JP
Japan
Prior art keywords
alkyl
amine
phenyl
compound
benzodiazole
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2019553478A
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English (en)
Japanese (ja)
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JP7674811B2 (ja
JP2020512373A (ja
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Publication date
Priority claimed from GBGB1705263.0A external-priority patent/GB201705263D0/en
Application filed filed Critical
Publication of JP2020512373A publication Critical patent/JP2020512373A/ja
Publication of JP2020512373A5 publication Critical patent/JP2020512373A5/ja
Priority to JP2022082769A priority Critical patent/JP7589191B2/ja
Priority to JP2024107135A priority patent/JP2024153639A/ja
Application granted granted Critical
Publication of JP7674811B2 publication Critical patent/JP7674811B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2019553478A 2017-03-31 2018-04-03 新規の阻害剤 Active JP7674811B2 (ja)

Priority Applications (2)

Application Number Priority Date Filing Date Title
JP2022082769A JP7589191B2 (ja) 2017-03-31 2022-05-20 新規の阻害剤
JP2024107135A JP2024153639A (ja) 2017-03-31 2024-07-03 新規の阻害剤

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB1705263.0 2017-03-31
GBGB1705263.0A GB201705263D0 (en) 2017-03-31 2017-03-31 Novel inhibitors
PCT/EP2018/058391 WO2018178384A1 (en) 2017-03-31 2018-04-03 Novel inhibitors

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2022082769A Division JP7589191B2 (ja) 2017-03-31 2022-05-20 新規の阻害剤

Publications (3)

Publication Number Publication Date
JP2020512373A JP2020512373A (ja) 2020-04-23
JP2020512373A5 true JP2020512373A5 (enExample) 2021-05-20
JP7674811B2 JP7674811B2 (ja) 2025-05-12

Family

ID=58682483

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2019553478A Active JP7674811B2 (ja) 2017-03-31 2018-04-03 新規の阻害剤
JP2022082769A Active JP7589191B2 (ja) 2017-03-31 2022-05-20 新規の阻害剤
JP2024107135A Pending JP2024153639A (ja) 2017-03-31 2024-07-03 新規の阻害剤

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2022082769A Active JP7589191B2 (ja) 2017-03-31 2022-05-20 新規の阻害剤
JP2024107135A Pending JP2024153639A (ja) 2017-03-31 2024-07-03 新規の阻害剤

Country Status (14)

Country Link
US (3) US11339152B2 (enExample)
EP (1) EP3601269A1 (enExample)
JP (3) JP7674811B2 (enExample)
KR (2) KR102737532B1 (enExample)
CN (2) CN110719910B (enExample)
AU (2) AU2018246382C1 (enExample)
CA (2) CA3221839A1 (enExample)
EA (1) EA201992120A1 (enExample)
GB (1) GB201705263D0 (enExample)
IL (3) IL297534A (enExample)
MX (2) MX2019011544A (enExample)
NZ (1) NZ792694A (enExample)
WO (1) WO2018178384A1 (enExample)
ZA (1) ZA201905811B (enExample)

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CN114560817B (zh) * 2022-04-25 2022-10-25 北京大学第三医院(北京大学第三临床医学院) 一种用于抑制纤维化的小分子药物及其应用
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IL319523A (en) 2022-09-13 2025-05-01 Augmedics Ltd Augmented reality glasses for image-guided medical intervention
WO2024131742A1 (zh) * 2022-12-20 2024-06-27 深圳湾实验室 一种靶向usp1的小分子抑制剂及其应用
CN120359213A (zh) 2022-12-22 2025-07-22 勃林格殷格翰国际有限公司 作为谷氨酰胺酰肽环转移酶和谷氨酰胺酰肽环转移酶样蛋白的抑制剂的苯基哌啶衍生物
EP4680333A1 (en) 2023-03-13 2026-01-21 Boehringer Ingelheim International GmbH Phenylpiperidine derivatives as inhibitors of glutaminyl-peptide cyclotransferase and glutaminyl-peptide cyclotransferase like protein
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