JP2020503277A5 - - Google Patents
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- JP2020503277A5 JP2020503277A5 JP2019529623A JP2019529623A JP2020503277A5 JP 2020503277 A5 JP2020503277 A5 JP 2020503277A5 JP 2019529623 A JP2019529623 A JP 2019529623A JP 2019529623 A JP2019529623 A JP 2019529623A JP 2020503277 A5 JP2020503277 A5 JP 2020503277A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- haloalkyl
- salt
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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- 150000001875 compounds Chemical class 0.000 claims description 85
- 150000003839 salts Chemical class 0.000 claims description 30
- 125000001188 haloalkyl group Chemical group 0.000 claims description 25
- 229910052736 halogen Inorganic materials 0.000 claims description 24
- 150000002367 halogens Chemical class 0.000 claims description 23
- 125000004122 cyclic group Chemical group 0.000 claims description 20
- 238000000034 method Methods 0.000 claims description 19
- 125000003545 alkoxy group Chemical group 0.000 claims description 12
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 12
- 125000004434 sulfur atom Chemical group 0.000 claims description 10
- 239000000203 mixture Substances 0.000 claims description 9
- QGZKDVFQNNGYKY-UHFFFAOYSA-N Ammonia Chemical compound N QGZKDVFQNNGYKY-UHFFFAOYSA-N 0.000 claims description 8
- 241000607479 Yersinia pestis Species 0.000 claims description 8
- 125000000753 cycloalkyl group Chemical group 0.000 claims description 8
- 125000004186 cyclopropylmethyl group Chemical group [H]C([H])(*)C1([H])C([H])([H])C1([H])[H] 0.000 claims description 8
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims description 8
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims description 8
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims description 8
- 125000004123 n-propyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])* 0.000 claims description 8
- 125000004430 oxygen atom Chemical group O* 0.000 claims description 8
- 239000000463 material Substances 0.000 claims description 6
- 230000001850 reproductive effect Effects 0.000 claims description 6
- 229910052717 sulfur Inorganic materials 0.000 claims description 6
- 101100025412 Arabidopsis thaliana XI-A gene Proteins 0.000 claims description 4
- BAVYZALUXZFZLV-UHFFFAOYSA-N Methylamine Chemical compound NC BAVYZALUXZFZLV-UHFFFAOYSA-N 0.000 claims description 4
- 239000002253 acid Substances 0.000 claims description 4
- 229910021529 ammonia Inorganic materials 0.000 claims description 4
- 150000003863 ammonium salts Chemical class 0.000 claims description 4
- 125000004093 cyano group Chemical group *C#N 0.000 claims description 4
- 229910052760 oxygen Inorganic materials 0.000 claims description 4
- 125000004076 pyridyl group Chemical group 0.000 claims description 4
- 125000001424 substituent group Chemical group 0.000 claims description 4
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims description 3
- 125000004770 (C1-C4) haloalkylsulfanyl group Chemical group 0.000 claims description 2
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 claims description 2
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 claims description 2
- 150000001204 N-oxides Chemical class 0.000 claims description 2
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims description 2
- 239000004480 active ingredient Substances 0.000 claims description 2
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims description 2
- 239000003795 chemical substances by application Substances 0.000 claims description 2
- 125000001309 chloro group Chemical group Cl* 0.000 claims description 2
- 125000001153 fluoro group Chemical group F* 0.000 claims description 2
- 230000002140 halogenating effect Effects 0.000 claims description 2
- 125000005842 heteroatom Chemical group 0.000 claims description 2
- 229910052757 nitrogen Inorganic materials 0.000 claims description 2
- 239000001301 oxygen Substances 0.000 claims description 2
- 230000000361 pesticidal effect Effects 0.000 claims description 2
- 239000011541 reaction mixture Substances 0.000 claims description 2
- -1 stereoisomers Chemical class 0.000 claims description 2
- 239000011593 sulfur Substances 0.000 claims description 2
- 239000012752 auxiliary agent Substances 0.000 claims 1
- 239000000126 substance Substances 0.000 description 26
- 125000000217 alkyl group Chemical group 0.000 description 15
- 125000004438 haloalkoxy group Chemical group 0.000 description 2
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 description 2
- 125000004429 atom Chemical group 0.000 description 1
- 125000004966 cyanoalkyl group Chemical group 0.000 description 1
- 238000002405 diagnostic procedure Methods 0.000 description 1
- 125000004663 dialkyl amino group Chemical group 0.000 description 1
- 125000004439 haloalkylsulfanyl group Chemical group 0.000 description 1
- 125000004440 haloalkylsulfinyl group Chemical group 0.000 description 1
- 125000005843 halogen group Chemical group 0.000 description 1
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN201611041146 | 2016-12-01 | ||
| IN201611041146 | 2016-12-01 | ||
| IN201711010969 | 2017-03-28 | ||
| IN201711010969 | 2017-03-28 | ||
| PCT/EP2017/080295 WO2018099812A1 (en) | 2016-12-01 | 2017-11-24 | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2020503277A JP2020503277A (ja) | 2020-01-30 |
| JP2020503277A5 true JP2020503277A5 (OSRAM) | 2021-01-07 |
| JP7282031B2 JP7282031B2 (ja) | 2023-05-26 |
Family
ID=60812015
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019529623A Active JP7282031B2 (ja) | 2016-12-01 | 2017-11-24 | 硫黄含有置換基を有する殺有害生物的に活性な複素環式誘導体 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US10961248B2 (OSRAM) |
| EP (1) | EP3548466B1 (OSRAM) |
| JP (1) | JP7282031B2 (OSRAM) |
| CN (2) | CN110023287B (OSRAM) |
| DK (1) | DK3548466T3 (OSRAM) |
| ES (1) | ES2910790T3 (OSRAM) |
| HU (1) | HUE058180T2 (OSRAM) |
| WO (1) | WO2018099812A1 (OSRAM) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2019229088A1 (en) | 2018-05-30 | 2019-12-05 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| WO2019229089A1 (en) | 2018-05-31 | 2019-12-05 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| US20220061324A1 (en) | 2018-12-31 | 2022-03-03 | Syngenta Crop Protection Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| ES2979156T3 (es) | 2019-09-20 | 2024-09-24 | Syngenta Crop Protection Ag | Derivados heterocíclicos plaguicidamente activos con sustituyentes que contienen azufre y sulfoximina |
| CN111223532B (zh) * | 2019-11-14 | 2023-06-20 | 腾讯科技（深圳）有限公司 | 确定目标化合物的反应物的方法、设备、装置、介质 |
| CA3201212A1 (en) * | 2020-12-14 | 2022-06-23 | Rizwan Shabbir SHAIKH | Sulfoximine pesticides |
| WO2022208370A1 (en) | 2021-03-31 | 2022-10-06 | Pi Industries Ltd. | Fused heterocyclic compounds and their use as pest control agents |
| AU2024235487A1 (en) | 2023-03-14 | 2025-09-25 | Syngenta Crop Protection Ag | Control of pests resistant to insecticides |
| TW202517614A (zh) | 2023-07-12 | 2025-05-01 | 瑞士商先正達農作物保護股份公司 | ２－（三氟甲基）吡啶－４－胺的合成 |
| WO2025177310A1 (en) | 2024-02-23 | 2025-08-28 | Pi Industries Ltd. | Fused heterocyclic compounds and its uses thereof |
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| BR8600161A (pt) | 1985-01-18 | 1986-09-23 | Plant Genetic Systems Nv | Gene quimerico,vetores de plasmidio hibrido,intermediario,processo para controlar insetos em agricultura ou horticultura,composicao inseticida,processo para transformar celulas de plantas para expressar uma toxina de polipeptideo produzida por bacillus thuringiensis,planta,semente de planta,cultura de celulas e plasmidio |
| CA1340685C (en) | 1988-07-29 | 1999-07-27 | Frederick Meins | Dna sequences encoding polypeptides having beta-1,3-glucanase activity |
| US5169629A (en) | 1988-11-01 | 1992-12-08 | Mycogen Corporation | Process of controlling lepidopteran pests, using bacillus thuringiensis isolate denoted b.t ps81gg |
| CA2005658A1 (en) | 1988-12-19 | 1990-06-19 | Eliahu Zlotkin | Insecticidal toxins, genes encoding these toxins, antibodies binding to them and transgenic plant cells and plants expressing these toxins |
| ES2199931T3 (es) | 1989-03-24 | 2004-03-01 | Syngenta Participations Ag | Plantas transgenicas resistentes a enfermedades. |
| GB8910624D0 (en) | 1989-05-09 | 1989-06-21 | Ici Plc | Bacterial strains |
| CA2015951A1 (en) | 1989-05-18 | 1990-11-18 | Mycogen Corporation | Novel bacillus thuringiensis isolates active against lepidopteran pests, and genes encoding novel lepidopteran-active toxins |
| ES2074547T3 (es) | 1989-11-07 | 1995-09-16 | Pioneer Hi Bred Int | Lectinas larvicidas, y resistencia inducida de las plantas a los insectos. |
| US5639949A (en) | 1990-08-20 | 1997-06-17 | Ciba-Geigy Corporation | Genes for the synthesis of antipathogenic substances |
| UA48104C2 (uk) | 1991-10-04 | 2002-08-15 | Новартіс Аг | Фрагмент днк, який містить послідовність,що кодує інсектицидний протеїн, оптимізовану для кукурудзи,фрагмент днк, який забезпечує направлену бажану для серцевини стебла експресію зв'язаного з нею структурного гена в рослині, фрагмент днк, який забезпечує специфічну для пилку експресію зв`язаного з нею структурного гена в рослині, рекомбінантна молекула днк, спосіб одержання оптимізованої для кукурудзи кодуючої послідовності інсектицидного протеїну, спосіб захисту рослин кукурудзи щонайменше від однієї комахи-шкідника |
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| US5631072A (en) | 1995-03-10 | 1997-05-20 | Avondale Incorporated | Method and means for increasing efficacy and wash durability of insecticide treated fabric |
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| JP6168055B2 (ja) | 2012-06-18 | 2017-07-26 | 住友化学株式会社 | 縮合複素環化合物 |
| UY35421A (es) * | 2013-03-15 | 2014-10-31 | Nihon Nohyaku Co Ltd | Compuesto heterocíclico condensado o su sal, insecticida agrícola u hortícola que comprende el comp uesto y método de uso del insecticida |
| WO2015002211A1 (ja) | 2013-07-01 | 2015-01-08 | 住友化学株式会社 | 縮合複素環化合物及びその有害生物防除用途 |
| EP3016949B1 (en) | 2013-07-02 | 2020-05-13 | Syngenta Participations AG | Pesticidally active bi- or tricyclic heterocycles with sulfur containing substituents |
| CN106414441B9 (zh) | 2014-02-17 | 2019-09-20 | 拜耳作物科学股份公司 | 作为害虫防治剂的2-(杂)芳基-取代的稠合双环杂环衍生物 |
| WO2016005263A1 (en) | 2014-07-08 | 2016-01-14 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
| CN106661023B (zh) | 2014-08-07 | 2019-05-28 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性杂环衍生物 |
| WO2016023954A2 (en) | 2014-08-12 | 2016-02-18 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
| ES2701859T3 (es) | 2014-08-21 | 2019-02-26 | Syngenta Participations Ag | Derivados heterocíclicos activos como plaguicida con sustituyentes que contienen azufre |
| WO2016046071A1 (en) | 2014-09-25 | 2016-03-31 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
| BR112017007510A2 (pt) | 2014-10-16 | 2018-06-19 | Syngenta Participations Ag | derivados heterocíclicos tetracíclicos com substituintes contendo enxofre ativos em termos pesticidas |
| BR112017009454B1 (pt) * | 2014-11-07 | 2022-05-03 | Syngenta Participations Ag | Composto, composição pesticida, método para controle de pragas e método para a proteção de material de propagação de plantas do ataque por pragas |
| WO2016091731A1 (en) | 2014-12-11 | 2016-06-16 | Syngenta Participations Ag | Pesticidally active tetracyclic derivatives with sulfur containing substituents |
| JP2018052816A (ja) | 2014-12-26 | 2018-04-05 | 日本農薬株式会社 | シクロアルキル基を有する縮合複素環化合物又はその塩類及び該化合物を含有する農園芸用殺虫剤並びにその使用方法 |
| BR112017015514B1 (pt) | 2015-01-19 | 2022-08-30 | Syngenta Participations Ag | Derivados policíclicos ativos com substituintes contendo enxofre ativo em termos pesticidas, composição pesticida e métodos para controle de pragas e proteção de sementes do ataque por pragas |
| UY36547A (es) | 2015-02-05 | 2016-06-01 | Bayer Cropscience Ag | Derivados heterocíclicos condensados bicíclicos sustituidos por 2-(het)arilo como pesticidas |
| WO2017084879A1 (en) | 2015-11-16 | 2017-05-26 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
| WO2017134066A1 (en) | 2016-02-05 | 2017-08-10 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
-
2017
- 2017-11-24 US US16/465,014 patent/US10961248B2/en active Active
- 2017-11-24 JP JP2019529623A patent/JP7282031B2/ja active Active
- 2017-11-24 EP EP17821477.1A patent/EP3548466B1/en active Active
- 2017-11-24 CN CN201780074390.9A patent/CN110023287B/zh not_active Expired - Fee Related
- 2017-11-24 ES ES17821477T patent/ES2910790T3/es active Active
- 2017-11-24 CN CN202311578234.XA patent/CN117624038A/zh active Pending
- 2017-11-24 WO PCT/EP2017/080295 patent/WO2018099812A1/en not_active Ceased
- 2017-11-24 DK DK17821477.1T patent/DK3548466T3/da active
- 2017-11-24 HU HUE17821477A patent/HUE058180T2/hu unknown
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