JP2019535799A5 - - Google Patents

Download PDF

Info

Publication number
JP2019535799A5
JP2019535799A5 JP2019528746A JP2019528746A JP2019535799A5 JP 2019535799 A5 JP2019535799 A5 JP 2019535799A5 JP 2019528746 A JP2019528746 A JP 2019528746A JP 2019528746 A JP2019528746 A JP 2019528746A JP 2019535799 A5 JP2019535799 A5 JP 2019535799A5
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
treatment
composition according
disorders
neurological
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2019528746A
Other languages
English (en)
Japanese (ja)
Other versions
JP7051853B2 (ja
JP2019535799A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2017/057418 external-priority patent/WO2018096510A1/en
Publication of JP2019535799A publication Critical patent/JP2019535799A/ja
Publication of JP2019535799A5 publication Critical patent/JP2019535799A5/ja
Application granted granted Critical
Publication of JP7051853B2 publication Critical patent/JP7051853B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2019528746A 2016-11-28 2017-11-27 ヘテロアリールフェノキシベンズアミドカッパオピオイドリガンド Active JP7051853B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201662426980P 2016-11-28 2016-11-28
US62/426,980 2016-11-28
US201762576435P 2017-10-24 2017-10-24
US62/576,435 2017-10-24
US201762585016P 2017-11-13 2017-11-13
US62/585,016 2017-11-13
PCT/IB2017/057418 WO2018096510A1 (en) 2016-11-28 2017-11-27 Heteroarylphenoxy benzamide kappa opioid ligands

Publications (3)

Publication Number Publication Date
JP2019535799A JP2019535799A (ja) 2019-12-12
JP2019535799A5 true JP2019535799A5 (enExample) 2021-01-14
JP7051853B2 JP7051853B2 (ja) 2022-04-11

Family

ID=60782279

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2019528746A Active JP7051853B2 (ja) 2016-11-28 2017-11-27 ヘテロアリールフェノキシベンズアミドカッパオピオイドリガンド

Country Status (18)

Country Link
US (1) US10316021B2 (enExample)
EP (1) EP3544972B8 (enExample)
JP (1) JP7051853B2 (enExample)
CN (1) CN110234638B (enExample)
AU (1) AU2017365123B2 (enExample)
DK (1) DK3544972T3 (enExample)
ES (1) ES2947293T3 (enExample)
FI (1) FI3544972T3 (enExample)
HR (1) HRP20230518T1 (enExample)
HU (1) HUE061945T2 (enExample)
IL (1) IL266962B (enExample)
MX (1) MX389806B (enExample)
PH (1) PH12019501172A1 (enExample)
PL (1) PL3544972T3 (enExample)
PT (1) PT3544972T (enExample)
RS (1) RS64258B1 (enExample)
TW (1) TWI720272B (enExample)
WO (1) WO2018096510A1 (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2018223177B2 (en) * 2017-02-24 2024-05-02 Xeniopro GmbH Aromatic compounds which enhance notch signaling, for use in therapy
WO2018154118A2 (en) * 2017-02-24 2018-08-30 Reinmueller Viktoria Novel aromatic compounds
US11266627B1 (en) 2021-05-04 2022-03-08 Janssen Pharmaceuticals, Inc. Compositions and methods for the treatment of depression
CN111233768B (zh) * 2020-03-18 2021-08-03 徐州圣元化工有限公司 一种3-(二氟甲基)-1-甲基-1h-吡唑-4-羧酸乙酯的制备方法
CA3140164A1 (en) * 2020-04-05 2021-10-14 Pfizer Inc. Compounds and methods for the treatment of covid-19
US12161622B2 (en) 2021-05-04 2024-12-10 Janssen Pharmaceuticals, Inc. Compositions and methods for the treatment of depression
IL315415A (en) 2022-03-07 2024-11-01 Janssen Pharmaceuticals Inc The compositions containing eticarpant
CA3254365A1 (en) * 2022-03-07 2023-09-14 Janssen Pharmaceuticals, Inc. POLYMORPHIC FORMS OF ATICAPRANT INTENDED FOR USE IN THE TREATMENT OF MAJOR DEPRESSION
CA3254503A1 (en) * 2022-03-07 2023-09-14 Janssen Pharmaceuticals, Inc. PURE FORMS OF CRYSTALLINE ATICAPRANT
EP4602033A1 (en) * 2022-10-12 2025-08-20 Adama Makhteshim Ltd. Process for the preparation of aminopyridazine derivatives

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5376645A (en) 1990-01-23 1994-12-27 University Of Kansas Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof
KR0166088B1 (ko) 1990-01-23 1999-01-15 . 수용해도가 증가된 시클로덱스트린 유도체 및 이의 용도
GB9518953D0 (en) 1995-09-15 1995-11-15 Pfizer Ltd Pharmaceutical formulations
WO2000035298A1 (en) 1996-11-27 2000-06-22 Wm. Wrigley Jr. Company Chewing gum containing medicament active agents
GB9711643D0 (en) 1997-06-05 1997-07-30 Janssen Pharmaceutica Nv Glass thermoplastic systems
JP2000159747A (ja) * 1998-09-21 2000-06-13 Takeda Chem Ind Ltd 新規チオ―ル誘導体、その製造法および用途
US6420415B1 (en) * 1998-09-21 2002-07-16 Takeda Chemical Industries, Ltd. Thiol compounds, their production and use
IT1303737B1 (it) 1998-11-11 2001-02-23 Smithkline Beecham Spa Derivati fenilpiperidinici procedimento per la loro preparazione eloro uso come ligandi del recettore orl-1.
UA80437C2 (en) 2002-09-19 2007-09-25 Lilly Co Eli Diaryl ethers as opioid receptor antagonist
US7365209B2 (en) 2003-02-11 2008-04-29 Pharmacopeia, Inc. Nitrogen heterocycle biaryls for osteoporosis and other diseases
ATE406360T1 (de) 2003-03-07 2008-09-15 Lilly Co Eli Antagonisten der opioidrezeptoren
CA2517888C (en) 2003-03-14 2012-05-01 Ono Pharmaceutical Co., Ltd. Nitrogen-containing heterocyclic derivatives and drugs containing the same as the active ingredient
US8188277B2 (en) 2004-08-06 2012-05-29 Otsuka Pharmaceutical Co., Ltd. Aromatic compounds for suppressing the generation of collagen
CN101120055B (zh) 2005-02-18 2014-07-23 日本曹达株式会社 有机无机复合体
WO2007105637A1 (ja) 2006-03-10 2007-09-20 Ono Pharmaceutical Co., Ltd. 含窒素複素環誘導体およびそれらを有効成分とする薬剤
RS51211B (sr) 2006-04-04 2010-12-31 Emodis Gmbh. Primena formulacija koje sadrže kapa-opioid receptor-agoniste za tretman disocijativnih poremećaja
NZ586225A (en) * 2008-01-22 2012-05-25 Lilly Co Eli Kappa selective opioid receptor antagonist
EP2257536A4 (en) 2008-02-14 2011-03-23 Amira Pharmaceuticals Inc CYCLIC DIARYL ETHERS AS ANTAGONISTS OF PROSTAGLANDIN D2 RECEPTORS
CR11559A (es) 2008-03-25 2010-10-20 Lilly Co Eli Antagonista del receptor opioide selectivo kappa
US8048895B2 (en) 2008-04-18 2011-11-01 Research Triangle Institute Kappa opioid receptor ligands
US8450335B2 (en) 2008-06-27 2013-05-28 Celgene Avilomics Research, Inc. 2,4-disubstituted pyrimidines useful as kinase inhibitors
CA2746943A1 (en) 2008-12-18 2010-07-15 Boehringer Ingelheim International Gmbh Serotonin 5-ht2b receptor inhibitors
HN2010001319A (es) 2009-01-26 2013-01-15 Lilly Co Eli Antagonista del receptor opioide selectivo kappa
WO2013059648A1 (en) 2011-10-21 2013-04-25 Neurotherapeutics Pharma, Inc. 2,3,5 trisubstituted aryl and heteroaryl amino derivatives, compositions, and methods of use
WO2014053210A1 (en) 2012-10-02 2014-04-10 Merck Patent Gmbh Pyrrolidines
WO2015109080A1 (en) 2014-01-15 2015-07-23 Research Triangle Institute Kappa-opioid receptor selective opioid receptor antagonists
WO2016086149A1 (en) 2014-11-26 2016-06-02 University Of Kansas Antagonists of the kappa opioid receptor

Similar Documents

Publication Publication Date Title
JP2019535799A5 (enExample)
IL269599B1 (en) 11, 13- modified schistosoxins for pain treatment
MA49402A (fr) Polynucléotides aadc pour le traitement de la maladie de parkinson
JP2016515522A5 (enExample)
HRP20210518T1 (hr) Derivati 2,4-tiazolidindiona, namijenjeni liječenju poremećaja središnjeg živčanog sustava
WO2016100162A3 (en) 5,5-bicyclic oxazole orexin receptor antagonists
WO2016100157A3 (en) 6,5-bicyclic octahydropyrrolopyridine orexin receptor antagonists
IL269310A (en) Use of designer receptors exclusively activated by designer drugs in the treatment of seizure disorders
PL3463351T3 (pl) Leczenie choroby parkinsona
WO2017070689A3 (en) Solabegron zwitterion and uses thereof
LT3413870T (lt) Igmesinas, skirtas panaudoti alzheimerio ligos gydymui
EP3589305C0 (en) SPECIFIC INCREASE IN DOPAMINE SYNTHESIS BY TARGETING THE GUANYLATE CYCLASE 2C RECEPTOR IN THE TREATMENT OF PARKINSON'S DISEASE
EA201791398A1 (ru) Производные фумагиллола
MA40065A (fr) N, n-bis-2-mercaptoéthyle isophtalamide pour le traitement de la maladie de parkinson
ZA201807944B (en) Treatment for parkinson's disease
IT201700006355A1 (it) Composizione per il trattamento dei disturbi gastrointestinali
SG10201912846PA (en) Therapeutic agent for non-motor symptoms associated with parkinson's disease
ZA201704287B (en) 3.alpha.-ethynyl, 3.beta.-hydroxy-5.alpha.-pregnan-20-oxime for use in the treatment of cns disorders
HK1245077A1 (en) Compositions and methods of treating a neurodegenerative disease
ITUB20153076A1 (it) Composti farmaceuticamente attivi per l?impiego nel trattamento terapeutico di disturbi del movimento.