JP2019529543A5 - - Google Patents

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Publication number
JP2019529543A5
JP2019529543A5 JP2019535434A JP2019535434A JP2019529543A5 JP 2019529543 A5 JP2019529543 A5 JP 2019529543A5 JP 2019535434 A JP2019535434 A JP 2019535434A JP 2019535434 A JP2019535434 A JP 2019535434A JP 2019529543 A5 JP2019529543 A5 JP 2019529543A5
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JP
Japan
Prior art keywords
pharmaceutical composition
injectable pharmaceutical
once
group
acyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2019535434A
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English (en)
Japanese (ja)
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JP6929367B2 (ja
JP2019529543A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/CN2017/101327 external-priority patent/WO2018050043A1/en
Publication of JP2019529543A publication Critical patent/JP2019529543A/ja
Publication of JP2019529543A5 publication Critical patent/JP2019529543A5/ja
Application granted granted Critical
Publication of JP6929367B2 publication Critical patent/JP6929367B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2019535434A 2016-09-13 2017-09-12 ブプレノルフィン徐放性製剤 Active JP6929367B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662394168P 2016-09-13 2016-09-13
US62/394,168 2016-09-13
PCT/CN2017/101327 WO2018050043A1 (en) 2016-09-13 2017-09-12 Sustained-release buprenorphine formulations background of invention

Publications (3)

Publication Number Publication Date
JP2019529543A JP2019529543A (ja) 2019-10-17
JP2019529543A5 true JP2019529543A5 (enExample) 2020-08-06
JP6929367B2 JP6929367B2 (ja) 2021-09-01

Family

ID=61619029

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2019535434A Active JP6929367B2 (ja) 2016-09-13 2017-09-12 ブプレノルフィン徐放性製剤

Country Status (31)

Country Link
US (1) US10744132B2 (enExample)
EP (1) EP3512518B1 (enExample)
JP (1) JP6929367B2 (enExample)
KR (1) KR102244500B1 (enExample)
CN (1) CN109789137B (enExample)
AR (1) AR110468A1 (enExample)
AU (1) AU2017325910B2 (enExample)
BR (1) BR112019004923A2 (enExample)
CA (1) CA3033046C (enExample)
CL (1) CL2019000624A1 (enExample)
CO (1) CO2019003632A2 (enExample)
DK (1) DK3512518T3 (enExample)
ES (1) ES2934721T3 (enExample)
FI (1) FI3512518T3 (enExample)
HR (1) HRP20230062T8 (enExample)
HU (1) HUE060906T2 (enExample)
LT (1) LT3512518T (enExample)
MX (1) MX374304B (enExample)
MY (1) MY196269A (enExample)
PE (1) PE20190707A1 (enExample)
PH (1) PH12019500466A1 (enExample)
PL (1) PL3512518T3 (enExample)
PT (1) PT3512518T (enExample)
RS (1) RS63894B1 (enExample)
RU (1) RU2747306C2 (enExample)
SG (1) SG11201901294QA (enExample)
SI (1) SI3512518T1 (enExample)
SM (1) SMT202300006T1 (enExample)
TW (1) TWI743193B (enExample)
WO (1) WO2018050043A1 (enExample)
ZA (1) ZA201900890B (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1057075C (zh) * 1997-09-10 2000-10-04 中国石油化工总公司 低碳烯烃直接水合连续生产低碳醇的方法
TWI838372B (zh) 2018-05-11 2024-04-11 昱展新藥生技股份有限公司 丁基原啡因衍生物之長效注射劑型及結晶型
TWI827777B (zh) * 2018-12-27 2024-01-01 昱展新藥生技股份有限公司 納曲酮注射型緩釋製劑
EP3936112A1 (en) * 2020-07-07 2022-01-12 Occlugel Hydrophilic degradable microspheres for delivering buprenorphine
AU2022270208A1 (en) * 2021-05-05 2023-12-07 Lyndra Therapeutics, Inc. Gastric residence systems comprising methadone

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2382577C (en) 1999-08-27 2008-01-22 Southern Research Institute Injectable buprenorphine microparticle compositions and their use
EP1554290B1 (en) 2002-10-25 2009-09-30 Euro-Celtique S.A. Analogs and prodrugs of buprenorphine
CN1263760C (zh) * 2002-11-12 2006-07-12 财团法人奇美医院 新颖的丁丙诺啡酯衍生物及其制备方法,以及长效作用镇痛药学组合物
TWI226830B (en) * 2002-11-12 2005-01-21 Chi Mei Foundation Medical Ct Novel ester derivatives of buprenorphine and their preparation processes, and long acting analgesic pharmaceutical compositions
ATE382050T1 (de) * 2002-11-25 2008-01-15 Chi Mei Foundation Medical Ct Buprenorphinesterderivate, verfahren zu ihrer herstellung, und langwirksame analgetische arzneimittel
PL1768650T3 (pl) 2004-06-04 2009-01-30 Camurus Ab Ciekłe formulacje depot
WO2007061739A2 (en) * 2005-11-21 2007-05-31 Schering-Plough Ltd. Pharmaceutical compositions comprising buprenorphine
GB0606124D0 (en) 2006-03-28 2006-05-03 Reckitt Benckiser Healthcare Buprenorphine derivatives and uses thereof
ES2549115T3 (es) * 2006-09-22 2015-10-23 Zynerba Pharmaceuticals, Inc. Profármacos de buprenorfina administrables por vía transdérmica y composiciones resistentes al consumo excesivo de los mismos
US20090181068A1 (en) * 2008-01-14 2009-07-16 Dunn Richard L Low Viscosity Liquid Polymeric Delivery System
GB2481018B (en) * 2010-06-08 2015-03-18 Rb Pharmaceuticals Ltd Injectable flowable composition comprising buprenorphine
GB2513060B (en) 2010-06-08 2015-01-07 Rb Pharmaceuticals Ltd Microparticle buprenorphine suspension
FR2975912B1 (fr) 2011-05-30 2013-06-14 Flamel Tech Sa Composition a liberation controlee de buprenorphine
US9393211B2 (en) 2013-03-15 2016-07-19 Oakwood Laboratories LLC High drug load buprenorphine microspheres and method of producing same
GB201404139D0 (en) * 2014-03-10 2014-04-23 Rb Pharmaceuticals Ltd Sustained release buprenorphine solution formulations
GB201419091D0 (en) * 2014-10-27 2014-12-10 Camurus Ab Formulations

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