JP2019529386A5 - - Google Patents

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Publication number
JP2019529386A5
JP2019529386A5 JP2019512638A JP2019512638A JP2019529386A5 JP 2019529386 A5 JP2019529386 A5 JP 2019529386A5 JP 2019512638 A JP2019512638 A JP 2019512638A JP 2019512638 A JP2019512638 A JP 2019512638A JP 2019529386 A5 JP2019529386 A5 JP 2019529386A5
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JP
Japan
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group
compound
pharmaceutically acceptable
acceptable salt
compound according
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JP2019512638A
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English (en)
Japanese (ja)
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JP2019529386A (ja
JP6838773B2 (ja
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Priority claimed from PCT/CN2017/100461 external-priority patent/WO2018041263A1/zh
Publication of JP2019529386A publication Critical patent/JP2019529386A/ja
Publication of JP2019529386A5 publication Critical patent/JP2019529386A5/ja
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JP2019512638A 2016-09-05 2017-09-05 抗インフルエンザウイルスのピリミジニル誘導体 Active JP6838773B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
CN201610804101.3 2016-09-05
CN201610804101 2016-09-05
CN201611238759 2016-12-28
CN201611238759.9 2016-12-28
PCT/CN2017/100461 WO2018041263A1 (zh) 2016-09-05 2017-09-05 抗流感病毒嘧啶衍生物

Publications (3)

Publication Number Publication Date
JP2019529386A JP2019529386A (ja) 2019-10-17
JP2019529386A5 true JP2019529386A5 (enExample) 2020-11-19
JP6838773B2 JP6838773B2 (ja) 2021-03-03

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ID=61300177

Family Applications (1)

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JP2019512638A Active JP6838773B2 (ja) 2016-09-05 2017-09-05 抗インフルエンザウイルスのピリミジニル誘導体

Country Status (14)

Country Link
US (4) US11136319B2 (enExample)
EP (1) EP3502112B1 (enExample)
JP (1) JP6838773B2 (enExample)
KR (1) KR102312088B1 (enExample)
CN (3) CN110627784B (enExample)
AU (1) AU2017320088B2 (enExample)
CA (1) CA3035680C (enExample)
DK (1) DK3502112T3 (enExample)
IL (1) IL265166B (enExample)
MX (1) MX394277B (enExample)
RU (1) RU2727772C1 (enExample)
SG (1) SG11201901894TA (enExample)
WO (1) WO2018041263A1 (enExample)
ZA (1) ZA201901886B (enExample)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2018033082A1 (en) 2016-08-16 2018-02-22 Sunshine Lake Pharma Co., Ltd. Inhibitors of influenza virus replication, application methods and uses thereof
CN109641868B (zh) 2016-08-30 2021-12-03 广东东阳光药业有限公司 流感病毒复制抑制剂及其使用方法和用途
RU2727772C1 (ru) * 2016-09-05 2020-07-23 Гуандун Рэйновент Байотек Ко., Лтд. Производные пиримидина против вируса гриппа
EP3555095B1 (en) 2016-12-15 2023-04-12 Sunshine Lake Pharma Co., Ltd. Inhibitors of influenza virus replication and uses thereof
US11098042B2 (en) 2017-01-05 2021-08-24 Sunshine Lake Pharma Co., Ltd. Inhibitors of influenza virus replication and uses thereof
CN110446711B (zh) 2017-03-02 2022-02-15 广东东阳光药业有限公司 流感病毒复制抑制剂及其用途
AU2019230497B2 (en) 2018-03-05 2021-08-05 Guangdong Raynovent Biotech Co., Ltd. Crystal form and salt form of pyridoimidazole compound and preparation method therefor
CN110590768B (zh) * 2018-06-13 2021-02-26 银杏树药业(苏州)有限公司 杂环化合物、其组合物及其作为抗流感病毒药物的应用
EP3992192A4 (en) * 2019-07-22 2022-08-17 Guangdong Raynovent Biotech Co., Ltd. DOMINANT SALT FORMS OF PYRIMIDINE DERIVATIVES AND CRYSTAL FORMS THEREOF
WO2021047437A1 (zh) * 2019-09-10 2021-03-18 广东众生睿创生物科技有限公司 一种用于治疗病毒性感冒的药物组合物及其制剂
CN111454166B (zh) * 2019-12-30 2021-02-26 广东莱佛士制药技术有限公司 制备(2s,3s)-3-氨基-二环[2.2.2]辛烷-2-甲酸酯的方法
CN113116899B (zh) * 2020-03-06 2022-12-20 广东众生睿创生物科技有限公司 一种用于治疗流感的药物组合物及含有该药物组合物的制剂
CN116323593B (zh) * 2020-10-29 2025-06-03 广东众生睿创生物科技有限公司 一种嘧啶衍生物的晶型及其制备方法
CN114569562B (zh) * 2020-12-01 2025-07-29 南通诺泰生物医药技术有限公司 一种抗流感病毒的药物组合物

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH12015501678B1 (en) * 2009-06-17 2022-07-06 Vertex Pharma Inhibitors of influenza viruses replication
AU2011343642A1 (en) * 2010-12-16 2013-05-02 Vertex Pharmaceuticals Incorporated Inhibitors of influenza viruses replication
US20130102600A1 (en) * 2011-10-21 2013-04-25 F. Hoffmann-La Roche Ltd Heteroaryl hydroxamic acid derivatives and their use in the treatment, amelioration or prevention of a viral disease
WO2016020526A1 (en) * 2014-08-08 2016-02-11 Janssen Sciences Ireland Uc Indoles for use in influenza virus infection
CN106854205B (zh) * 2015-12-09 2019-07-09 广东东阳光药业有限公司 流感病毒复制抑制剂及其使用方法和用途
WO2017133657A1 (en) * 2016-02-05 2017-08-10 Savira Pharmaceuticals Gmbh Pyridine and pyrimidine derivatives and their use in treatment, amelioration or prevention of influenza
WO2017133670A1 (en) * 2016-02-05 2017-08-10 Savira Pharmaceuticals Gmbh Pyridine and pyrimidine derivatives and their use in treatment, amelioration or prevention of influenza
WO2018033082A1 (en) 2016-08-16 2018-02-22 Sunshine Lake Pharma Co., Ltd. Inhibitors of influenza virus replication, application methods and uses thereof
RU2727772C1 (ru) * 2016-09-05 2020-07-23 Гуандун Рэйновент Байотек Ко., Лтд. Производные пиримидина против вируса гриппа
AU2019230497B2 (en) * 2018-03-05 2021-08-05 Guangdong Raynovent Biotech Co., Ltd. Crystal form and salt form of pyridoimidazole compound and preparation method therefor
EP3992192A4 (en) * 2019-07-22 2022-08-17 Guangdong Raynovent Biotech Co., Ltd. DOMINANT SALT FORMS OF PYRIMIDINE DERIVATIVES AND CRYSTAL FORMS THEREOF

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