JP2019526552A - インダノン調製方法 - Google Patents

インダノン調製方法 Download PDF

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Publication number
JP2019526552A
JP2019526552A JP2019508193A JP2019508193A JP2019526552A JP 2019526552 A JP2019526552 A JP 2019526552A JP 2019508193 A JP2019508193 A JP 2019508193A JP 2019508193 A JP2019508193 A JP 2019508193A JP 2019526552 A JP2019526552 A JP 2019526552A
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Prior art keywords
formula
methyl
compound
mmol
inden
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JP2019508193A
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Japanese (ja)
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JP2019526552A5 (enExample
Inventor
グラニエ,ティエリー
ツォウ,ユエ
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ジボダン エス エー
ジボダン エス エー
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Publication of JP2019526552A publication Critical patent/JP2019526552A/ja
Publication of JP2019526552A5 publication Critical patent/JP2019526552A5/ja
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/51Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by pyrolysis, rearrangement or decomposition
    • C07C45/516Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by pyrolysis, rearrangement or decomposition involving transformation of nitrogen-containing compounds to >C = O groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/06Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B37/00Reactions without formation or introduction of functional groups containing hetero atoms, involving either the formation of a carbon-to-carbon bond between two carbon atoms not directly linked already or the disconnection of two directly linked carbon atoms
    • C07B37/10Cyclisation
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00Preparation of carboxylic acid amides
    • C07C231/12Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/36Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
    • C07C303/40Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids by reactions not involving the formation of sulfonamide groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/587Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/687Unsaturated compounds containing a keto groups being part of a ring containing halogen
    • C07C49/697Unsaturated compounds containing a keto groups being part of a ring containing halogen containing six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/06Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08Systems containing only non-condensed rings with a five-membered ring the ring being saturated
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00Systems containing two condensed rings
    • C07C2602/02Systems containing two condensed rings the rings having only two atoms in common
    • C07C2602/04One of the condensed rings being a six-membered aromatic ring
    • C07C2602/08One of the condensed rings being a six-membered aromatic ring the other ring being five-membered, e.g. indane
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/01Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/02Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C311/07Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
JP2019508193A 2016-08-15 2017-08-14 インダノン調製方法 Ceased JP2019526552A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN2016095275 2016-08-15
CNPCT/CN2016/095275 2016-08-15
PCT/EP2017/070595 WO2017191332A2 (en) 2016-08-15 2017-08-14 Process of making organic compounds

Publications (2)

Publication Number Publication Date
JP2019526552A true JP2019526552A (ja) 2019-09-19
JP2019526552A5 JP2019526552A5 (enExample) 2020-09-24

Family

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Family Applications (1)

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JP2019508193A Ceased JP2019526552A (ja) 2016-08-15 2017-08-14 インダノン調製方法

Country Status (7)

Country Link
US (1) US10494323B2 (enExample)
EP (1) EP3497078B1 (enExample)
JP (1) JP2019526552A (enExample)
CN (1) CN109563029B (enExample)
ES (1) ES2853704T3 (enExample)
MX (1) MX2019000984A (enExample)
WO (1) WO2017191332A2 (enExample)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2019536038A (ja) * 2016-11-23 2019-12-12 ウーテーアー・エス・アー・マニファクチュール・オロロジェール・スイス 分離レバー脱進機によって維持される、撓み支承体を有する回転共振器
JP2023533571A (ja) * 2020-07-10 2023-08-03 アダマ・アガン・リミテッド ピロキサスルホン、フェノキサスルホン、及び5,5-ジメチル-4h-1,2-オキサゾールの各種のスルホン類似体を調製するためのプロセス及び中間体

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005519081A (ja) * 2002-02-28 2005-06-30 ジボダン エス エー インダンおよびインダノンならびにそれらの香料における使用
JP2019532123A (ja) * 2016-08-15 2019-11-07 ジボダン エス エー 有機化合物

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3944679A (en) 1973-04-13 1976-03-16 The Japan Tobacco & Salt Public Corporation Process for imparting a coumarin-like aroma and flavor to tobacco, foods and drinks
KR100595963B1 (ko) 2004-04-13 2006-07-05 한국화학연구원 인덴 유도체 및 이의 제조방법
US20050261513A1 (en) 2004-05-18 2005-11-24 Womack Gary B Process for producing indenol esters or ethers

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005519081A (ja) * 2002-02-28 2005-06-30 ジボダン エス エー インダンおよびインダノンならびにそれらの香料における使用
JP2019532123A (ja) * 2016-08-15 2019-11-07 ジボダン エス エー 有機化合物

Non-Patent Citations (7)

* Cited by examiner, † Cited by third party
Title
DING, RAN; HUANG, ZHI-DAO; LIU, ZHENG-LI; WANG, TIAN-XIANG; XU, YUN-HE; LOH, TECK-PENG: "Palladium-catalyzed cross-coupling of enamides with sterically hindered α-bromocarbonyls", CHEMICAL COMMUNICATIONS (CAMBRIDGE, UNITED KINGDOM), vol. 52(32),, JPN6021023984, 2016, pages 5617 - 5620, ISSN: 0004531840 *
WANG, SHAOYIN; ZHU, YUANXUN; WANG, YANGUANG; LU, PING: "Synthesis of functionalized indenes via cascade reaction of aziridines and propargyl alcohols", ORGANIC LETTERS, vol. 11(12),, JPN6021023985, 2009, pages 2615 - 2618, ISSN: 0004531841 *
WILLIAM M KRAFT: "THE PREPARATION OF INDANONE DERIVATIVES BY A CARBAMATE-ALDEHYDE 1 REACTION", JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, vol. VOL:70, NR:11, JPN5019007648, November 1948 (1948-11-01), US, pages 3569 - 3571, ISSN: 0004735695 *
WOMACK, GARY B.; ANGELES, JOHN G.; FANELLI, VINCENT E.; HEYER, CHRISTIE A.: "Conversion of 2-Alkylcinnamaldehydes to 2-Alkylindanones via a Catalytic Intramolecular Friedel-C", JOURNAL OF ORGANIC CHEMISTRY, vol. 72(18),, JPN6021023983, 2007, pages 7046 - 7049, ISSN: 0004531839 *
WOMACK, GARY B.; ANGELES, JOHN G.; FANELLI, VINCENT E.; INDRADAS, BRINDA; SNOWDEN, ROGER L.; SONN: "Indanones and Indenols from 2-Alkylcinnamaldehydes via the Intramolecular Friedel-Crafts Reaction", JOURNAL OF ORGANIC CHEMISTRY, vol. 74(15),, JPN6021023982, 2009, pages 5738 - 5741, ISSN: 0004531838 *
XIAOHUI FAN; ET AL: "ASSEMBLY OF INDENAMINE DERIVATIVES THROUGH IN SITU FORMED N-SULFONYLIMINIUM ION 以下備考", CHEMICAL COMMUNICATIONS, vol. VOL:50, NR:31, JPN5019007650, January 2014 (2014-01-01), pages 4119 - 4122, ISSN: 0004531837 *
標準化学用語辞典 第2版, JPN6021023981, 2005, ISSN: 0004735696 *

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2019536038A (ja) * 2016-11-23 2019-12-12 ウーテーアー・エス・アー・マニファクチュール・オロロジェール・スイス 分離レバー脱進機によって維持される、撓み支承体を有する回転共振器
JP2019537015A (ja) * 2016-11-23 2019-12-19 ウーテーアー・エス・アー・マニファクチュール・オロロジェール・スイス 分離レバー脱進機によって維持される、撓み支承体を有する回転共振器
JP2023533571A (ja) * 2020-07-10 2023-08-03 アダマ・アガン・リミテッド ピロキサスルホン、フェノキサスルホン、及び5,5-ジメチル-4h-1,2-オキサゾールの各種のスルホン類似体を調製するためのプロセス及び中間体

Also Published As

Publication number Publication date
EP3497078B1 (en) 2020-12-23
MX2019000984A (es) 2019-07-04
CN109563029A (zh) 2019-04-02
CN109563029B (zh) 2021-10-26
US20190263743A1 (en) 2019-08-29
WO2017191332A2 (en) 2017-11-09
WO2017191332A3 (en) 2018-01-04
ES2853704T3 (es) 2021-09-17
US10494323B2 (en) 2019-12-03
EP3497078A2 (en) 2019-06-19

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