CN109563029B - 用于制备二氢茚酮类的方法 - Google Patents
用于制备二氢茚酮类的方法 Download PDFInfo
- Publication number
- CN109563029B CN109563029B CN201780049982.5A CN201780049982A CN109563029B CN 109563029 B CN109563029 B CN 109563029B CN 201780049982 A CN201780049982 A CN 201780049982A CN 109563029 B CN109563029 B CN 109563029B
- Authority
- CN
- China
- Prior art keywords
- formula
- compound
- methyl
- inden
- isobutyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/51—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by pyrolysis, rearrangement or decomposition
- C07C45/516—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by pyrolysis, rearrangement or decomposition involving transformation of nitrogen-containing compounds to >C = O groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C269/06—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B37/00—Reactions without formation or introduction of functional groups containing hetero atoms, involving either the formation of a carbon-to-carbon bond between two carbon atoms not directly linked already or the disconnection of two directly linked carbon atoms
- C07B37/10—Cyclisation
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
- C07C303/40—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids by reactions not involving the formation of sulfonamide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
- C07C49/687—Unsaturated compounds containing a keto groups being part of a ring containing halogen
- C07C49/697—Unsaturated compounds containing a keto groups being part of a ring containing halogen containing six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
- C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/04—One of the condensed rings being a six-membered aromatic ring
- C07C2602/08—One of the condensed rings being a six-membered aromatic ring the other ring being five-membered, e.g. indane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
- C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C311/07—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN2016095275 | 2016-08-15 | ||
| CNPCT/CN2016/095275 | 2016-08-15 | ||
| PCT/EP2017/070595 WO2017191332A2 (en) | 2016-08-15 | 2017-08-14 | Process of making organic compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN109563029A CN109563029A (zh) | 2019-04-02 |
| CN109563029B true CN109563029B (zh) | 2021-10-26 |
Family
ID=59699677
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN201780049982.5A Active CN109563029B (zh) | 2016-08-15 | 2017-08-14 | 用于制备二氢茚酮类的方法 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US10494323B2 (enExample) |
| EP (1) | EP3497078B1 (enExample) |
| JP (1) | JP2019526552A (enExample) |
| CN (1) | CN109563029B (enExample) |
| ES (1) | ES2853704T3 (enExample) |
| MX (1) | MX2019000984A (enExample) |
| WO (1) | WO2017191332A2 (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH713150A2 (fr) * | 2016-11-23 | 2018-05-31 | Eta Sa Mft Horlogere Suisse | Mécanisme régulateur à résonateur rotatif à guidage flexible entretenu par un échappement libre à ancre. |
| EP4177245A1 (en) * | 2020-07-10 | 2023-05-10 | Adama Agan Ltd. | Process and intermediates for the preparation of fenoxasulfone |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3944679A (en) | 1973-04-13 | 1976-03-16 | The Japan Tobacco & Salt Public Corporation | Process for imparting a coumarin-like aroma and flavor to tobacco, foods and drinks |
| EP1340741A1 (en) | 2002-02-28 | 2003-09-03 | Givaudan SA | Indane derivatives and their use in perfumery |
| KR100595963B1 (ko) | 2004-04-13 | 2006-07-05 | 한국화학연구원 | 인덴 유도체 및 이의 제조방법 |
| US20050261513A1 (en) | 2004-05-18 | 2005-11-24 | Womack Gary B | Process for producing indenol esters or ethers |
| MX384407B (es) * | 2016-08-15 | 2025-03-14 | Givaudan Sa | Derivados de indanona que poseen propiedades olfativas frutales y florales. |
-
2017
- 2017-08-14 EP EP17757502.4A patent/EP3497078B1/en active Active
- 2017-08-14 JP JP2019508193A patent/JP2019526552A/ja not_active Ceased
- 2017-08-14 CN CN201780049982.5A patent/CN109563029B/zh active Active
- 2017-08-14 MX MX2019000984A patent/MX2019000984A/es unknown
- 2017-08-14 WO PCT/EP2017/070595 patent/WO2017191332A2/en not_active Ceased
- 2017-08-14 US US16/320,376 patent/US10494323B2/en active Active
- 2017-08-14 ES ES17757502T patent/ES2853704T3/es active Active
Non-Patent Citations (3)
| Title |
|---|
| ssembly of indenamine derivatives through in situ formed N-sulfonyliminium ion initiated cyclization;Xiaohui Fan等;《Chem. Commun.》;20140225;第50卷;第4119- 4122页 * |
| The Preparation of Indanone Derivatives by a Carbamate-Aldehyde Reaction;William M.Kraft;《Journal of the American chemical society》;19481101;第70卷(第11期);第3569-3571页 * |
| William M.Kraft.The Preparation of Indanone Derivatives by a Carbamate-Aldehyde Reaction.《Journal of the American chemical society》.1948,第70卷(第11期),第3569-3571页. * |
Also Published As
| Publication number | Publication date |
|---|---|
| CN109563029A (zh) | 2019-04-02 |
| WO2017191332A2 (en) | 2017-11-09 |
| MX2019000984A (es) | 2019-07-04 |
| US20190263743A1 (en) | 2019-08-29 |
| EP3497078B1 (en) | 2020-12-23 |
| US10494323B2 (en) | 2019-12-03 |
| WO2017191332A3 (en) | 2018-01-04 |
| EP3497078A2 (en) | 2019-06-19 |
| JP2019526552A (ja) | 2019-09-19 |
| ES2853704T3 (es) | 2021-09-17 |
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| GR01 | Patent grant | ||
| GR01 | Patent grant |