JP2019526552A - インダノン調製方法 - Google Patents
インダノン調製方法 Download PDFInfo
- Publication number
- JP2019526552A JP2019526552A JP2019508193A JP2019508193A JP2019526552A JP 2019526552 A JP2019526552 A JP 2019526552A JP 2019508193 A JP2019508193 A JP 2019508193A JP 2019508193 A JP2019508193 A JP 2019508193A JP 2019526552 A JP2019526552 A JP 2019526552A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- methyl
- compound
- mmol
- inden
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/51—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by pyrolysis, rearrangement or decomposition
- C07C45/516—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by pyrolysis, rearrangement or decomposition involving transformation of nitrogen-containing compounds to >C = O groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C269/06—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B37/00—Reactions without formation or introduction of functional groups containing hetero atoms, involving either the formation of a carbon-to-carbon bond between two carbon atoms not directly linked already or the disconnection of two directly linked carbon atoms
- C07B37/10—Cyclisation
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
- C07C303/40—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids by reactions not involving the formation of sulfonamide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
- C07C49/687—Unsaturated compounds containing a keto groups being part of a ring containing halogen
- C07C49/697—Unsaturated compounds containing a keto groups being part of a ring containing halogen containing six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
- C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/04—One of the condensed rings being a six-membered aromatic ring
- C07C2602/08—One of the condensed rings being a six-membered aromatic ring the other ring being five-membered, e.g. indane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
- C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C311/07—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN2016095275 | 2016-08-15 | ||
| CNPCT/CN2016/095275 | 2016-08-15 | ||
| PCT/EP2017/070595 WO2017191332A2 (en) | 2016-08-15 | 2017-08-14 | Process of making organic compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2019526552A true JP2019526552A (ja) | 2019-09-19 |
| JP2019526552A5 JP2019526552A5 (cg-RX-API-DMAC10.html) | 2020-09-24 |
Family
ID=59699677
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019508193A Ceased JP2019526552A (ja) | 2016-08-15 | 2017-08-14 | インダノン調製方法 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US10494323B2 (cg-RX-API-DMAC10.html) |
| EP (1) | EP3497078B1 (cg-RX-API-DMAC10.html) |
| JP (1) | JP2019526552A (cg-RX-API-DMAC10.html) |
| CN (1) | CN109563029B (cg-RX-API-DMAC10.html) |
| ES (1) | ES2853704T3 (cg-RX-API-DMAC10.html) |
| MX (1) | MX2019000984A (cg-RX-API-DMAC10.html) |
| WO (1) | WO2017191332A2 (cg-RX-API-DMAC10.html) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2019536038A (ja) * | 2016-11-23 | 2019-12-12 | ウーテーアー・エス・アー・マニファクチュール・オロロジェール・スイス | 分離レバー脱進機によって維持される、撓み支承体を有する回転共振器 |
| JP2023533571A (ja) * | 2020-07-10 | 2023-08-03 | アダマ・アガン・リミテッド | ピロキサスルホン、フェノキサスルホン、及び５，５－ジメチル－４ｈ－１，２－オキサゾールの各種のスルホン類似体を調製するためのプロセス及び中間体 |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005519081A (ja) * | 2002-02-28 | 2005-06-30 | ジボダン エス エー | インダンおよびインダノンならびにそれらの香料における使用 |
| JP2019532123A (ja) * | 2016-08-15 | 2019-11-07 | ジボダン エス エー | 有機化合物 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3944679A (en) | 1973-04-13 | 1976-03-16 | The Japan Tobacco & Salt Public Corporation | Process for imparting a coumarin-like aroma and flavor to tobacco, foods and drinks |
| KR100595963B1 (ko) | 2004-04-13 | 2006-07-05 | 한국화학연구원 | 인덴 유도체 및 이의 제조방법 |
| US20050261513A1 (en) | 2004-05-18 | 2005-11-24 | Womack Gary B | Process for producing indenol esters or ethers |
-
2017
- 2017-08-14 US US16/320,376 patent/US10494323B2/en active Active
- 2017-08-14 ES ES17757502T patent/ES2853704T3/es active Active
- 2017-08-14 JP JP2019508193A patent/JP2019526552A/ja not_active Ceased
- 2017-08-14 MX MX2019000984A patent/MX2019000984A/es unknown
- 2017-08-14 WO PCT/EP2017/070595 patent/WO2017191332A2/en not_active Ceased
- 2017-08-14 CN CN201780049982.5A patent/CN109563029B/zh active Active
- 2017-08-14 EP EP17757502.4A patent/EP3497078B1/en active Active
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005519081A (ja) * | 2002-02-28 | 2005-06-30 | ジボダン エス エー | インダンおよびインダノンならびにそれらの香料における使用 |
| JP2019532123A (ja) * | 2016-08-15 | 2019-11-07 | ジボダン エス エー | 有機化合物 |
Non-Patent Citations (7)
| Title |
|---|
| DING, RAN; HUANG, ZHI-DAO; LIU, ZHENG-LI; WANG, TIAN-XIANG; XU, YUN-HE; LOH, TECK-PENG: "Palladium-catalyzed cross-coupling of enamides with sterically hindered α-bromocarbonyls", CHEMICAL COMMUNICATIONS (CAMBRIDGE, UNITED KINGDOM), vol. 52(32),, JPN6021023984, 2016, pages 5617 - 5620, ISSN: 0004531840 * |
| WANG, SHAOYIN; ZHU, YUANXUN; WANG, YANGUANG; LU, PING: "Synthesis of functionalized indenes via cascade reaction of aziridines and propargyl alcohols", ORGANIC LETTERS, vol. 11(12),, JPN6021023985, 2009, pages 2615 - 2618, ISSN: 0004531841 * |
| WILLIAM M KRAFT: "THE PREPARATION OF INDANONE DERIVATIVES BY A CARBAMATE-ALDEHYDE 1 REACTION", JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, vol. VOL:70, NR:11, JPN5019007648, November 1948 (1948-11-01), US, pages 3569 - 3571, ISSN: 0004735695 * |
| WOMACK, GARY B.; ANGELES, JOHN G.; FANELLI, VINCENT E.; HEYER, CHRISTIE A.: "Conversion of 2-Alkylcinnamaldehydes to 2-Alkylindanones via a Catalytic Intramolecular Friedel-C", JOURNAL OF ORGANIC CHEMISTRY, vol. 72(18),, JPN6021023983, 2007, pages 7046 - 7049, ISSN: 0004531839 * |
| WOMACK, GARY B.; ANGELES, JOHN G.; FANELLI, VINCENT E.; INDRADAS, BRINDA; SNOWDEN, ROGER L.; SONN: "Indanones and Indenols from 2-Alkylcinnamaldehydes via the Intramolecular Friedel-Crafts Reaction", JOURNAL OF ORGANIC CHEMISTRY, vol. 74(15),, JPN6021023982, 2009, pages 5738 - 5741, ISSN: 0004531838 * |
| XIAOHUI FAN; ET AL: "ASSEMBLY OF INDENAMINE DERIVATIVES THROUGH IN SITU FORMED N-SULFONYLIMINIUM ION 以下備考", CHEMICAL COMMUNICATIONS, vol. VOL:50, NR:31, JPN5019007650, January 2014 (2014-01-01), pages 4119 - 4122, ISSN: 0004531837 * |
| 標準化学用語辞典 第２版, JPN6021023981, 2005, ISSN: 0004735696 * |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2019536038A (ja) * | 2016-11-23 | 2019-12-12 | ウーテーアー・エス・アー・マニファクチュール・オロロジェール・スイス | 分離レバー脱進機によって維持される、撓み支承体を有する回転共振器 |
| JP2019537015A (ja) * | 2016-11-23 | 2019-12-19 | ウーテーアー・エス・アー・マニファクチュール・オロロジェール・スイス | 分離レバー脱進機によって維持される、撓み支承体を有する回転共振器 |
| JP2023533571A (ja) * | 2020-07-10 | 2023-08-03 | アダマ・アガン・リミテッド | ピロキサスルホン、フェノキサスルホン、及び５，５－ジメチル－４ｈ－１，２－オキサゾールの各種のスルホン類似体を調製するためのプロセス及び中間体 |
Also Published As
| Publication number | Publication date |
|---|---|
| MX2019000984A (es) | 2019-07-04 |
| WO2017191332A3 (en) | 2018-01-04 |
| US20190263743A1 (en) | 2019-08-29 |
| EP3497078A2 (en) | 2019-06-19 |
| WO2017191332A2 (en) | 2017-11-09 |
| US10494323B2 (en) | 2019-12-03 |
| CN109563029A (zh) | 2019-04-02 |
| CN109563029B (zh) | 2021-10-26 |
| EP3497078B1 (en) | 2020-12-23 |
| ES2853704T3 (es) | 2021-09-17 |
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