JP2019516708A5 - - Google Patents

Download PDF

Info

Publication number
JP2019516708A5
JP2019516708A5 JP2018560490A JP2018560490A JP2019516708A5 JP 2019516708 A5 JP2019516708 A5 JP 2019516708A5 JP 2018560490 A JP2018560490 A JP 2018560490A JP 2018560490 A JP2018560490 A JP 2018560490A JP 2019516708 A5 JP2019516708 A5 JP 2019516708A5
Authority
JP
Japan
Prior art keywords
alkyl
catalyst
halogen
alkoxy
aryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2018560490A
Other languages
English (en)
Japanese (ja)
Other versions
JP7113762B2 (ja
JP2019516708A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2017/033489 external-priority patent/WO2017201377A1/en
Publication of JP2019516708A publication Critical patent/JP2019516708A/ja
Publication of JP2019516708A5 publication Critical patent/JP2019516708A5/ja
Priority to JP2022118930A priority Critical patent/JP2022141912A/ja
Application granted granted Critical
Publication of JP7113762B2 publication Critical patent/JP7113762B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2018560490A 2016-05-19 2017-05-19 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成 Active JP7113762B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2022118930A JP2022141912A (ja) 2016-05-19 2022-07-26 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201662338562P 2016-05-19 2016-05-19
US62/338,562 2016-05-19
US201662416811P 2016-11-03 2016-11-03
US62/416,811 2016-11-03
PCT/US2017/033489 WO2017201377A1 (en) 2016-05-19 2017-05-19 Synthesis of 6-aryl-4-aminopicolinates and 2-aryl-6-aminopyrimidine-4-carboxylates by direct suzuki coupling

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2022118930A Division JP2022141912A (ja) 2016-05-19 2022-07-26 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成

Publications (3)

Publication Number Publication Date
JP2019516708A JP2019516708A (ja) 2019-06-20
JP2019516708A5 true JP2019516708A5 (enExample) 2020-07-02
JP7113762B2 JP7113762B2 (ja) 2022-08-05

Family

ID=60326419

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2018560490A Active JP7113762B2 (ja) 2016-05-19 2017-05-19 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成
JP2022118930A Ceased JP2022141912A (ja) 2016-05-19 2022-07-26 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2022118930A Ceased JP2022141912A (ja) 2016-05-19 2022-07-26 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成

Country Status (12)

Country Link
US (3) US10087164B2 (enExample)
EP (1) EP3458442B1 (enExample)
JP (2) JP7113762B2 (enExample)
KR (1) KR20190007048A (enExample)
CN (1) CN109415319A (enExample)
AU (2) AU2017268424B2 (enExample)
BR (1) BR112018073348B8 (enExample)
CA (1) CA3023935A1 (enExample)
IL (1) IL263075A (enExample)
MX (1) MX2018014174A (enExample)
RU (1) RU2018144344A (enExample)
WO (1) WO2017201377A1 (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN109415319A (zh) * 2016-05-19 2019-03-01 美国陶氏益农公司 通过直接苏楚基偶联合成芳基羧酸酯
US11401242B2 (en) * 2018-09-19 2022-08-02 Corteva Agriscience Llc Preparation of halogen analogs of picloram
WO2020133403A1 (zh) * 2018-12-29 2020-07-02 青岛清原化合物有限公司 取代的嘧啶芳酯衍生物及其制备方法、除草组合物和应用
CN115279737A (zh) * 2020-03-18 2022-11-01 科迪华农业科技有限责任公司 4-氨基-6-(杂环)吡啶甲酸酯的改进合成
BR112022018513A2 (pt) 2020-03-18 2022-11-01 Corteva Agriscience Llc Síntese melhorada de 6-aril-4-aminopicolinatos
WO2021231196A1 (en) * 2020-05-11 2021-11-18 Corteva Agriscience Llc Preparation of compounds having pesticidal activity
WO2023248174A1 (en) * 2022-06-22 2023-12-28 Hetero Labs Limited An improved process for preparation of voxelotor
CN115819334B (zh) * 2022-06-28 2025-03-18 安徽众邦生物工程有限公司 一种氯氟吡啶酯的制备方法

Family Cites Families (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR037228A1 (es) * 2001-07-30 2004-11-03 Dow Agrosciences Llc Compuestos del acido 6-(aril o heteroaril)-4-aminopicolinico, composicion herbicida que los comprende y metodo para controlar vegetacion no deseada
JP4332589B2 (ja) * 2006-01-13 2009-09-16 ダウ アグロサイエンシィズ エルエルシー ２−（多置換アリール）−６−アミノ−５−ハロ−４−ピリミジンカルボン酸および除草剤としてのそれらの使用
ES2401348T3 (es) * 2007-08-13 2013-04-18 Dow Agrosciences, Llc 2-(Fenil 2-fluoro-substituido)-6-amino-5-cloro-4-pirimidinacarboxilatos y su uso como herbicidas
DE602008005319D1 (de) * 2007-08-30 2011-04-14 Dow Agrosciences Llc 2-(substituierte phenyl)-6-amino-5-alkoxy-, thioalkoxy- und aminoalkyl-4-pyrimidincarboxylate und ihre verwendung als herbizide
BR122016003312B8 (pt) * 2007-10-02 2022-06-28 Dow Agrosciences Llc Ácidos 2-substituído-6-amino-5-alquil, alquenil ou alquinil-4-pirimidinacarboxílicos e ácidos 6-substituído-4-amino-3-alquil, alquenil ou alquinil picolínicos, composição herbicida que os compreende e método de controlar vegetação indesejável
PL2279178T3 (pl) * 2008-04-18 2015-10-30 Dow Agrosciences Llc 2-(podstawione-fenylo)-6-hydroksy- lub alkoksy-5-podstawione-4 pirymidynokarboksylany i ich zastosowanie jako herbicydów
GB0808664D0 (en) * 2008-05-13 2008-06-18 Syngenta Ltd Chemical compounds
GB0902474D0 (en) * 2009-02-13 2009-04-01 Syngenta Ltd Chemical compounds
GB0907625D0 (en) * 2009-05-01 2009-06-10 Syngenta Ltd Method of controlling undesired vegetation
TWI592401B (zh) * 2011-01-25 2017-07-21 陶氏農業科學公司 用於製備４－胺基－３－氯－５－氟－６－（經取代的）吡啶甲酸酯的方法（一）
TWI547482B (zh) 2011-01-25 2016-09-01 陶氏農業科學公司 增加可回收之3-氯-4,5,6-三氟-2-氰吡啶之量的改良方法
TWI529163B (zh) * 2011-01-25 2016-04-11 陶氏農業科學公司 用於製備４－胺基－５－氟－３－鹵素－６－（經取代之）吡啶甲酸酯的方法
MX336729B (es) * 2011-01-25 2016-01-28 Dow Agrosciences Llc Acidos 6-amino-2-sustituido-5-vinilsililpirimidin-4-carboxilicos y esteres y acidos 4-amino-6-sustituido-3-vinilsililpiridin-picoli nicos y esteres como herbicidas.
PL2736897T3 (pl) * 2011-07-27 2016-04-29 Bayer Ip Gmbh Podstawione kwasy pikolinowe i kwasy pirymidyno-4-karboksylowe, sposób ich otrzymywania i ich zastosowanie jako herbicydy i regulatory wzrostu roślin
MX356476B (es) * 2011-12-30 2018-05-30 Dow Agrosciences Llc Métodos para aislar 4-cloro-2-fluor-3-fenil boronatos sustituidos y métodos para su uso.
NZ627192A (en) 2011-12-30 2015-09-25 Dow Agrosciences Llc Methods of producing methyl 4-amino-3-chloro-6-(4-chloro-2-fluoro-3-methoxyphenyl)pyridine-2-carboxylate
AR091856A1 (es) * 2012-07-24 2015-03-04 Dow Agrosciences Llc Proceso para la preparacion de 4-amino-5-fluor-3-halo-6-(substituido) picolinatos
CN102875456B (zh) * 2012-10-23 2013-12-11 西华大学 3,6-二氯-2-氨基吡啶的化学合成方法
US20140170058A1 (en) * 2012-12-13 2014-06-19 Dow Agrosciences Llc Process for the removal of palladium from 4-amino-3-halo-5-fluoro-6-(aryl) pyridine-2-carboxylates and 4-amino-3-halo-6-(aryl)pyridine-2-carboxylates
PL2967057T3 (pl) * 2013-03-15 2019-05-31 Dow Agrosciences Llc Nowe karboksylany 4-aminopirydyny i 6-aminopirymidyny jako herbicydy
RU2672584C2 (ru) 2013-03-15 2018-11-16 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи 4-амино-6-(гетероциклил)пиколинаты и 6-амино-2-(гетероциклил)пиримидин-4-карбоксилаты и их применение в качестве гербицидов
US9637505B2 (en) * 2013-03-15 2017-05-02 Dow Agrosciences Llc 4-amino-6-(heterocyclic)picolinates and 6-amino-2-(heterocyclic)pyrimidine-4-carboxylates and their use as herbicides
WO2014151009A1 (en) 2013-03-15 2014-09-25 Dow Agrosciences Llc 4-amino-6-(heterocyclic)picolinates and 6-amino-2-(heterocyclic) pyrimidine-4-carboxylates and their use as herbicides
US9113629B2 (en) * 2013-03-15 2015-08-25 Dow Agrosciences Llc 4-amino-6-(4-substituted-phenyl)-picolinates and 6-amino-2-(4-substituted-phenyl)-pyrimidine-4-carboxylates and their use as herbicides
CN109415319A (zh) * 2016-05-19 2019-03-01 美国陶氏益农公司 通过直接苏楚基偶联合成芳基羧酸酯

Similar Documents

Publication Publication Date Title
JP2019516708A5 (enExample)
JP2012521411A5 (enExample)
JP2010531876A5 (enExample)
CN110563535B (zh) 一种炔烃烷基化合成1,2-二取代烯烃类化合物的方法
JP2005525427A5 (enExample)
RU2102384C1 (ru) Способ получения 4-метил-2'-цианобифенила
TW200808725A (en) Process for the preparation of 2-substituted-5-(1-alkylthio)alkylpyridines
RU2018144344A (ru) Синтез 6-арил-4-аминопиколинатов и 2-арил-6-аминопиримидин-4-карбоксилатов прямым сочетанием сузуки
Abbiati et al. Palladium-assisted multicomponent synthesis of 2-aryl-4-aminoquinolines and 2-aryl-4-amino [1, 8] naphthyridines
Hosseini-Sarvari et al. Nano copper (I) oxide/zinc oxide catalyzed N-arylation of nitrogen-containing heterocycles with aryl halides and arylboronic acids in air
Feng et al. Palladium catalyzed direct C-2 arylation of indoles
CN103980086A (zh) 一种1,3-丁二炔催化体系的制备方法
Gour et al. A Microwave-Assisted SmI2-Catalyzed Direct N-Alkylation of Anilines with Alcohols
CN104098607B (zh) 含三环己基膦的单膦单氮杂环卡宾镍(ii)配合物及其应用
LaBerge et al. Activation and formation of aromatic C–F bonds
JP2005534711A (ja) 新規ニッケル−、パラジウム−及び白金−カルベン錯体、それらの製造及び触媒反応における使用
JP5679855B2 (ja) ジフルオロメチル化ヘテロアリール化合物の製造方法
JP2013527149A5 (enExample)
Kim et al. Sublimable bis (β-iminoenolate) palladium (II) complexes and their application as catalysts in Suzuki-Miyaura reactions
JP2017516808A5 (enExample)
JP2012031190A (ja) 炭素−炭素結合の生成方法
CN103193568B (zh) 含氟芳烃衍生物的选择性氢化还原方法
JP2014196365A5 (enExample)
JP2005523934A5 (enExample)
CN108137503A (zh) 制备1-(4-甲磺酰基-2-三氟甲基-苄基)-2-甲基-1h-吡咯并[2,3-b]吡啶-3-基-乙酸的工艺