JP2019516708A5 - - Google Patents
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- Publication number
- JP2019516708A5 JP2019516708A5 JP2018560490A JP2018560490A JP2019516708A5 JP 2019516708 A5 JP2019516708 A5 JP 2019516708A5 JP 2018560490 A JP2018560490 A JP 2018560490A JP 2018560490 A JP2018560490 A JP 2018560490A JP 2019516708 A5 JP2019516708 A5 JP 2019516708A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- catalyst
- halogen
- alkoxy
- aryl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2022118930A JP2022141912A (ja) | 2016-05-19 | 2022-07-26 | 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成 |
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662338562P | 2016-05-19 | 2016-05-19 | |
| US62/338,562 | 2016-05-19 | ||
| US201662416811P | 2016-11-03 | 2016-11-03 | |
| US62/416,811 | 2016-11-03 | ||
| PCT/US2017/033489 WO2017201377A1 (en) | 2016-05-19 | 2017-05-19 | Synthesis of 6-aryl-4-aminopicolinates and 2-aryl-6-aminopyrimidine-4-carboxylates by direct suzuki coupling |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022118930A Division JP2022141912A (ja) | 2016-05-19 | 2022-07-26 | 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2019516708A JP2019516708A (ja) | 2019-06-20 |
| JP2019516708A5 true JP2019516708A5 (enExample) | 2020-07-02 |
| JP7113762B2 JP7113762B2 (ja) | 2022-08-05 |
Family
ID=60326419
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018560490A Active JP7113762B2 (ja) | 2016-05-19 | 2017-05-19 | 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成 |
| JP2022118930A Ceased JP2022141912A (ja) | 2016-05-19 | 2022-07-26 | 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022118930A Ceased JP2022141912A (ja) | 2016-05-19 | 2022-07-26 | 直接的な鈴木カップリングによる６－アリール－４－アミノピコリネートおよび２－アリール－６－アミノピリミジン－４－カルボキシレートの合成 |
Country Status (12)
| Country | Link |
|---|---|
| US (3) | US10087164B2 (enExample) |
| EP (1) | EP3458442B1 (enExample) |
| JP (2) | JP7113762B2 (enExample) |
| KR (1) | KR20190007048A (enExample) |
| CN (1) | CN109415319A (enExample) |
| AU (2) | AU2017268424B2 (enExample) |
| BR (1) | BR112018073348B8 (enExample) |
| CA (1) | CA3023935A1 (enExample) |
| IL (1) | IL263075A (enExample) |
| MX (1) | MX2018014174A (enExample) |
| RU (1) | RU2018144344A (enExample) |
| WO (1) | WO2017201377A1 (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10087164B2 (en) * | 2016-05-19 | 2018-10-02 | Dow Agrosciences Llc | Synthesis of 6-aryl-4-aminopicolinates and 2-aryl-6-aminopyrimidine-4-carboxylates by direct Suzuki coupling |
| CN113015721B (zh) | 2018-09-19 | 2025-07-25 | 科迪华农业科技有限责任公司 | 毒莠定卤素类似物的制备 |
| WO2020133403A1 (zh) * | 2018-12-29 | 2020-07-02 | 青岛清原化合物有限公司 | 取代的嘧啶芳酯衍生物及其制备方法、除草组合物和应用 |
| CN115279737A (zh) | 2020-03-18 | 2022-11-01 | 科迪华农业科技有限责任公司 | 4-氨基-6-(杂环)吡啶甲酸酯的改进合成 |
| CN115298167A (zh) * | 2020-03-18 | 2022-11-04 | 科迪华农业科技有限责任公司 | 6-芳基-4-氨基吡啶甲酸酯的改进合成 |
| EP4149926A1 (en) * | 2020-05-11 | 2023-03-22 | Corteva Agriscience LLC | Preparation of compounds having pesticidal activity |
| WO2023248174A1 (en) * | 2022-06-22 | 2023-12-28 | Hetero Labs Limited | An improved process for preparation of voxelotor |
| CN115819334B (zh) * | 2022-06-28 | 2025-03-18 | 安徽众邦生物工程有限公司 | 一种氯氟吡啶酯的制备方法 |
Family Cites Families (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR037228A1 (es) | 2001-07-30 | 2004-11-03 | Dow Agrosciences Llc | Compuestos del acido 6-(aril o heteroaril)-4-aminopicolinico, composicion herbicida que los comprende y metodo para controlar vegetacion no deseada |
| WO2007082076A1 (en) * | 2006-01-13 | 2007-07-19 | Dow Agrosciences Llc | 2-(poly-substituted aryl)-6-amino-5-halo-4-pyrimidinecarboxylic acids and their use as herbicides |
| EP2311815B1 (en) * | 2007-08-13 | 2012-12-19 | Dow AgroSciences LLC | 2-(2-Fluoro-substituted phenyl)-6-amino-5-chloro-4-pyrimidinecarboxylates and their use as herbicides |
| AU2008293462B2 (en) * | 2007-08-30 | 2013-08-15 | Corteva Agriscience Llc | 2-(substituted phenyl)-6-amino-5-alkoxy, thioalkoxy and aminoalkyl-4-pyrimidinecarboxylates and their use as herbicides |
| PL2327694T3 (pl) * | 2007-10-02 | 2013-12-31 | Dow Agrosciences Llc | Podstawione kwasy 4-aminopikolinowe i ich zastosowanie jako herbicydów |
| MX2010011468A (es) * | 2008-04-18 | 2010-12-14 | Dow Agrosciences Llc | 2-(fenil substituido)-6-hidroxi o alcoxi-5-substituido-4-pirimidin carboxilatos y sus usos como herbicidas. |
| GB0808664D0 (en) * | 2008-05-13 | 2008-06-18 | Syngenta Ltd | Chemical compounds |
| GB0902474D0 (en) * | 2009-02-13 | 2009-04-01 | Syngenta Ltd | Chemical compounds |
| GB0907625D0 (en) * | 2009-05-01 | 2009-06-10 | Syngenta Ltd | Method of controlling undesired vegetation |
| CA2825392C (en) * | 2011-01-25 | 2016-10-25 | Dow Agrosciences Llc | 6-amino-2-substituted-5-vinylsilylpyrimidine-4-carboxylic acids and esters and 4-amino-6-substituted-3-vinylsilylpyridine-2-carboxylic acids and esters as herbicides |
| TWI520943B (zh) | 2011-01-25 | 2016-02-11 | 陶氏農業科學公司 | 用於製備４－胺基－３－氯－５－氟－６－（經取代的）吡啶甲酸酯的方法（二） |
| TWI529163B (zh) * | 2011-01-25 | 2016-04-11 | 陶氏農業科學公司 | 用於製備４－胺基－５－氟－３－鹵素－６－（經取代之）吡啶甲酸酯的方法 |
| TWI592401B (zh) * | 2011-01-25 | 2017-07-21 | 陶氏農業科學公司 | 用於製備４－胺基－３－氯－５－氟－６－（經取代的）吡啶甲酸酯的方法（一） |
| HUE028580T2 (en) * | 2011-07-27 | 2016-12-28 | Bayer Ip Gmbh | Substituted Picolinic Acids and Pyrimidine Carboxylic Acids, Process for their Preparation and Use as Herbicides and Plant Growth Regulators |
| BR112014015962B8 (pt) * | 2011-12-30 | 2022-10-11 | Dow Agrosciences Llc | Métodos para produzir 4-amino-3-cloro-6-(4-cloro-2-flúor-3-metóxi-fenil)piridina-2-carboxilato de metila |
| CN104080791B (zh) * | 2011-12-30 | 2016-12-07 | 陶氏益农公司 | 分离和使用(4-氯-2-氟-3-取代的-苯基)硼酸酯的方法 |
| AR091856A1 (es) | 2012-07-24 | 2015-03-04 | Dow Agrosciences Llc | Proceso para la preparacion de 4-amino-5-fluor-3-halo-6-(substituido) picolinatos |
| CN102875456B (zh) * | 2012-10-23 | 2013-12-11 | 西华大学 | 3,6-二氯-2-氨基吡啶的化学合成方法 |
| US20140170058A1 (en) * | 2012-12-13 | 2014-06-19 | Dow Agrosciences Llc | Process for the removal of palladium from 4-amino-3-halo-5-fluoro-6-(aryl) pyridine-2-carboxylates and 4-amino-3-halo-6-(aryl)pyridine-2-carboxylates |
| EP2970186B1 (en) | 2013-03-15 | 2020-06-10 | Dow AgroSciences LLC | 4-amino-6-(heterocyclic)picolinates and 6-amino-2-(heterocyclic) pyrimidine-4-carboxylates and their use as herbicides |
| US9113629B2 (en) * | 2013-03-15 | 2015-08-25 | Dow Agrosciences Llc | 4-amino-6-(4-substituted-phenyl)-picolinates and 6-amino-2-(4-substituted-phenyl)-pyrimidine-4-carboxylates and their use as herbicides |
| US9637505B2 (en) * | 2013-03-15 | 2017-05-02 | Dow Agrosciences Llc | 4-amino-6-(heterocyclic)picolinates and 6-amino-2-(heterocyclic)pyrimidine-4-carboxylates and their use as herbicides |
| WO2014151008A1 (en) * | 2013-03-15 | 2014-09-25 | Dow Agrosciences Llc | 4-amino-6-(heterocyclic)picolinates and 6-amino-2-(heterocyclic)pyrimidine-4-carboxylates and their use as herbicides |
| EP2967057B1 (en) * | 2013-03-15 | 2018-11-21 | Dow AgroSciences LLC | Novel 4-aminopyridine and 6-aminopyrimidine carboxylates as herbicides |
| US10087164B2 (en) * | 2016-05-19 | 2018-10-02 | Dow Agrosciences Llc | Synthesis of 6-aryl-4-aminopicolinates and 2-aryl-6-aminopyrimidine-4-carboxylates by direct Suzuki coupling |
-
2017
- 2017-05-19 US US15/599,716 patent/US10087164B2/en active Active
- 2017-05-19 KR KR1020187036364A patent/KR20190007048A/ko not_active Abandoned
- 2017-05-19 CN CN201780042463.6A patent/CN109415319A/zh active Pending
- 2017-05-19 CA CA3023935A patent/CA3023935A1/en active Pending
- 2017-05-19 MX MX2018014174A patent/MX2018014174A/es unknown
- 2017-05-19 JP JP2018560490A patent/JP7113762B2/ja active Active
- 2017-05-19 BR BR112018073348A patent/BR112018073348B8/pt active IP Right Grant
- 2017-05-19 RU RU2018144344A patent/RU2018144344A/ru unknown
- 2017-05-19 WO PCT/US2017/033489 patent/WO2017201377A1/en not_active Ceased
- 2017-05-19 AU AU2017268424A patent/AU2017268424B2/en not_active Ceased
- 2017-05-19 EP EP17800225.9A patent/EP3458442B1/en active Active
-
2018
- 2018-07-26 US US16/045,896 patent/US10544121B2/en active Active
- 2018-07-26 US US16/045,901 patent/US10570114B2/en active Active
- 2018-11-18 IL IL263075A patent/IL263075A/en unknown
-
2021
- 2021-05-20 AU AU2021203233A patent/AU2021203233A1/en not_active Abandoned
-
2022
- 2022-07-26 JP JP2022118930A patent/JP2022141912A/ja not_active Ceased
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