JP2019507791A5 - - Google Patents

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Publication number
JP2019507791A5
JP2019507791A5 JP2018547929A JP2018547929A JP2019507791A5 JP 2019507791 A5 JP2019507791 A5 JP 2019507791A5 JP 2018547929 A JP2018547929 A JP 2018547929A JP 2018547929 A JP2018547929 A JP 2018547929A JP 2019507791 A5 JP2019507791 A5 JP 2019507791A5
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JP
Japan
Prior art keywords
compound
pharmaceutically acceptable
dihydroxybutan
sulfonamide
thio
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2018547929A
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English (en)
Japanese (ja)
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JP2019507791A (ja
JP6883917B2 (ja
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Publication date
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Priority claimed from PCT/US2017/021570 external-priority patent/WO2017156270A1/en
Publication of JP2019507791A publication Critical patent/JP2019507791A/ja
Publication of JP2019507791A5 publication Critical patent/JP2019507791A5/ja
Priority to JP2021078242A priority Critical patent/JP7126014B2/ja
Application granted granted Critical
Publication of JP6883917B2 publication Critical patent/JP6883917B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2018547929A 2016-03-11 2017-03-09 結晶性関節障害を処置するためのcxcr−2阻害剤 Expired - Fee Related JP6883917B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2021078242A JP7126014B2 (ja) 2016-03-11 2021-05-05 結晶性関節障害を処置するためのcxcr-2阻害剤

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662307348P 2016-03-11 2016-03-11
US62/307,348 2016-03-11
PCT/US2017/021570 WO2017156270A1 (en) 2016-03-11 2017-03-09 Cxcr-2 inhibitors for treating crystal arthropathy disorders

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2021078242A Division JP7126014B2 (ja) 2016-03-11 2021-05-05 結晶性関節障害を処置するためのcxcr-2阻害剤

Publications (3)

Publication Number Publication Date
JP2019507791A JP2019507791A (ja) 2019-03-22
JP2019507791A5 true JP2019507791A5 (enExample) 2020-04-30
JP6883917B2 JP6883917B2 (ja) 2021-06-09

Family

ID=59789863

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2018547929A Expired - Fee Related JP6883917B2 (ja) 2016-03-11 2017-03-09 結晶性関節障害を処置するためのcxcr−2阻害剤
JP2021078242A Active JP7126014B2 (ja) 2016-03-11 2021-05-05 結晶性関節障害を処置するためのcxcr-2阻害剤

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2021078242A Active JP7126014B2 (ja) 2016-03-11 2021-05-05 結晶性関節障害を処置するためのcxcr-2阻害剤

Country Status (10)

Country Link
US (1) US10772886B2 (enExample)
EP (1) EP3426253A4 (enExample)
JP (2) JP6883917B2 (enExample)
CN (2) CN113893252A (enExample)
AU (1) AU2017231832B2 (enExample)
BR (1) BR112018068393A2 (enExample)
CA (1) CA3017345A1 (enExample)
CO (1) CO2018010880A2 (enExample)
MX (1) MX386771B (enExample)
WO (1) WO2017156270A1 (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN113893252A (zh) 2016-03-11 2022-01-07 阿迪亚生命科学公司 用于治疗结晶性关节病症的cxcr-2抑制剂
WO2019055509A1 (en) * 2017-09-12 2019-03-21 Ardea Biosciences, Inc. INHIBITORS OF CXCR-2 FOR THE TREATMENT OF DISORDERS
US11136315B2 (en) 2018-01-11 2021-10-05 Medshine Discovery Inc. CXCR2 antagonist
WO2021004531A1 (zh) * 2019-07-11 2021-01-14 南京明德新药研发有限公司 一种cxcr2拮抗剂的晶型及其应用
KR102260478B1 (ko) * 2019-08-19 2021-06-02 연세대학교 산학협력단 일나트륨 요소화물 결정 용해용 조성물
TW202210068A (zh) * 2020-06-05 2022-03-16 美商雅力思提雅治療公司 用於治療家族性地中海型發熱病的cxcr-2抑制劑
WO2022162021A1 (en) * 2021-01-27 2022-08-04 Astrazeneca Ab Verinurad compositions and methods of use

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KR100883476B1 (ko) 2004-01-30 2009-02-16 쉐링 코포레이션 Cxc-케모킨 수용체 리간드의 결정성 다형체
BRPI0514735B8 (pt) 2004-08-28 2021-05-25 Astrazeneca Ab derivados de pirimidino sulfonamida como moduladores do receptor de quimiocina.
AU2008206231A1 (en) * 2007-01-19 2008-07-24 Takeda Pharmaceuticals U.S.A., Inc. Methods for preventing or reducing the number of gout flares using xanthine oxidoreductase inhibitors and anti-inflammatory agents
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KR20110014141A (ko) 2008-03-20 2011-02-10 카롤러스 테라퓨틱스, 인코포레이티드 염증을 치료하는 방법
CN102159555A (zh) 2008-07-16 2011-08-17 阿斯利康(瑞典)有限公司 嘧啶基氨磺酰衍生物及其治疗趋化因子介导的疾病的用途
MX2011003328A (es) 2008-10-06 2011-06-20 Carolus Therapeutics Inc Metodos para tratar inflamacion.
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PH12014500107A1 (en) 2011-07-12 2014-03-03 Astrazeneca Ab N- (6- ( (2r,3s) -3,4-dihydroxybutan-2-yloxy) -2- (4 - fluorobenzylthio) pyrimidin- 4 - yl) -3- methylazetidine- 1 - sulfonamide as chemokine receptor modulator
JP2015528001A (ja) 2012-07-11 2015-09-24 ティッシュテック,インク. Hc−ha/ptx3複合体を含む組成物およびその使用方法
EP3220951A1 (en) 2014-11-17 2017-09-27 MedImmune Limited Therapeutic combinations and methods for treating neoplasia
US20180221312A1 (en) 2016-03-11 2018-08-09 Ardea Biosciences, Inc. Cxcr-2 inhibitors for treating disorders
CN113893252A (zh) 2016-03-11 2022-01-07 阿迪亚生命科学公司 用于治疗结晶性关节病症的cxcr-2抑制剂
WO2019055509A1 (en) 2017-09-12 2019-03-21 Ardea Biosciences, Inc. INHIBITORS OF CXCR-2 FOR THE TREATMENT OF DISORDERS

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