JP2018528928A5 - - Google Patents

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Publication number
JP2018528928A5
JP2018528928A5 JP2017567608A JP2017567608A JP2018528928A5 JP 2018528928 A5 JP2018528928 A5 JP 2018528928A5 JP 2017567608 A JP2017567608 A JP 2017567608A JP 2017567608 A JP2017567608 A JP 2017567608A JP 2018528928 A5 JP2018528928 A5 JP 2018528928A5
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JP
Japan
Prior art keywords
formula
compound
crystalline form
side chain
hydrogen
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Application number
JP2017567608A
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English (en)
Japanese (ja)
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JP6801835B2 (ja
JP2018528928A (ja
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Priority claimed from PCT/EP2016/066281 external-priority patent/WO2017005902A1/en
Publication of JP2018528928A publication Critical patent/JP2018528928A/ja
Publication of JP2018528928A5 publication Critical patent/JP2018528928A5/ja
Application granted granted Critical
Publication of JP6801835B2 publication Critical patent/JP6801835B2/ja
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JP2017567608A 2015-07-09 2016-07-08 β−ターンペプチド模倣環状塩の液相合成及び結晶化 Active JP6801835B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562190596P 2015-07-09 2015-07-09
US62/190,596 2015-07-09
PCT/EP2016/066281 WO2017005902A1 (en) 2015-07-09 2016-07-08 Solution phase synthesis and crystallization of beta-turn peptidomimetic cyclic salts

Publications (3)

Publication Number Publication Date
JP2018528928A JP2018528928A (ja) 2018-10-04
JP2018528928A5 true JP2018528928A5 (enExample) 2019-04-18
JP6801835B2 JP6801835B2 (ja) 2020-12-16

Family

ID=56413639

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2017567608A Active JP6801835B2 (ja) 2015-07-09 2016-07-08 β−ターンペプチド模倣環状塩の液相合成及び結晶化

Country Status (8)

Country Link
US (4) US10125165B2 (enExample)
EP (2) EP3319978B1 (enExample)
JP (1) JP6801835B2 (enExample)
KR (1) KR102056257B1 (enExample)
CN (2) CN107849089B (enExample)
AU (1) AU2016290654C1 (enExample)
TW (1) TWI708779B (enExample)
WO (1) WO2017005902A1 (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102056257B1 (ko) * 2015-07-09 2019-12-16 미메토젠 파르마슈티칼스 인크. 베타-턴 펩티도미메틱 사이클릭 염의 용액상 합성 및 결정화
SI3464336T1 (sl) 2016-06-01 2022-06-30 Athira Pharma, Inc. Spojine
KR102826649B1 (ko) * 2018-05-31 2025-06-30 쎄데르마 용액-상 펩티드의 합성 방법 및 그에 따른 보호 전략
US11427612B2 (en) * 2018-08-21 2022-08-30 Wayne State University Epimerization-free N to C solid-phase peptide synthesis
CN117279928A (zh) * 2021-05-07 2023-12-22 中外制药株式会社 包含n-取代氨基酸残基的环状化合物的制备方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AUPP254898A0 (en) * 1998-03-24 1998-04-23 University Of Queensland, The Peptide turn mimetics
WO2001052843A1 (en) 2000-01-18 2001-07-26 Mcgill University β-TURN PEPTIDOMIMETIC CYCLIC COMPOUNDS
HRP20041179B1 (hr) * 2002-06-11 2012-11-30 Eli Lilly And Company Prekursorski oblici lijekova za aminokiseline s pobuđivačkom aktivnosti
AU2009232352B2 (en) * 2008-04-04 2013-09-05 Mimetogen Pharmaceuticals Inc. Beta-turn peptidomimetic cyclic compounds for treating dry eye
AU2010217889B2 (en) * 2009-02-27 2014-12-18 Mimetogen Pharmaceuticals Inc. Peptidomimetic cyclic compounds for treating retinitis pigmentosa
EP2598604B1 (de) * 2010-07-29 2015-11-25 Merck Patent GmbH Flüssigkristallines medium enthaltend thiophenderivate
JP5710436B2 (ja) * 2011-09-26 2015-04-30 株式会社東芝 パターン形成方法
EP2864347B1 (en) * 2012-06-22 2020-10-28 Mimetogen Pharmaceuticals, Inc. Synthesis of beta-turn peptidomimetic cyclic compounds
JP6516974B2 (ja) * 2013-06-14 2019-05-22 豊田合成株式会社 ゴム組成物及びゴム製品
CN105142777B (zh) * 2013-06-20 2017-12-26 埃克森美孚化学专利公司 长桥Salen催化剂
KR102056257B1 (ko) * 2015-07-09 2019-12-16 미메토젠 파르마슈티칼스 인크. 베타-턴 펩티도미메틱 사이클릭 염의 용액상 합성 및 결정화

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