JP2018524341A5 - - Google Patents
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- Publication number
- JP2018524341A5 JP2018524341A5 JP2017567803A JP2017567803A JP2018524341A5 JP 2018524341 A5 JP2018524341 A5 JP 2018524341A5 JP 2017567803 A JP2017567803 A JP 2017567803A JP 2017567803 A JP2017567803 A JP 2017567803A JP 2018524341 A5 JP2018524341 A5 JP 2018524341A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- represented
- reacting
- phenoxyphenylamidine
- reaction scheme
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- LIWAQLJGPBVORC-UHFFFAOYSA-N ethylmethylamine Chemical compound CCNC LIWAQLJGPBVORC-UHFFFAOYSA-N 0.000 claims 6
- HJKLEAOXCZIMPI-UHFFFAOYSA-N 2,2-diethoxyethanamine Chemical compound CCOC(CN)OCC HJKLEAOXCZIMPI-UHFFFAOYSA-N 0.000 claims 5
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 5
- 229910052739 hydrogen Inorganic materials 0.000 claims 5
- 239000001257 hydrogen Substances 0.000 claims 5
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 5
- 244000005700 microbiome Species 0.000 claims 5
- PAYRUJLWNCNPSJ-UHFFFAOYSA-N Aniline Chemical compound NC1=CC=CC=C1 PAYRUJLWNCNPSJ-UHFFFAOYSA-N 0.000 claims 4
- 125000001246 bromo group Chemical group Br* 0.000 claims 4
- 125000001309 chloro group Chemical group Cl* 0.000 claims 4
- 238000000034 method Methods 0.000 claims 4
- 239000003905 agrochemical Substances 0.000 claims 3
- 125000001153 fluoro group Chemical group F* 0.000 claims 3
- 238000009472 formulation Methods 0.000 claims 3
- 239000000203 mixture Substances 0.000 claims 3
- FJLHLDBEZKTSOK-UHFFFAOYSA-N n-ethyl-n-methylformamide Chemical compound CCN(C)C=O FJLHLDBEZKTSOK-UHFFFAOYSA-N 0.000 claims 3
- 150000002905 orthoesters Chemical class 0.000 claims 3
- 150000002989 phenols Chemical class 0.000 claims 3
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 3
- XVIRIXVOLLJIPF-UHFFFAOYSA-N 1-nitro-2-(2-nitrophenoxy)benzene Chemical compound [O-][N+](=O)C1=CC=CC=C1OC1=CC=CC=C1[N+]([O-])=O XVIRIXVOLLJIPF-UHFFFAOYSA-N 0.000 claims 2
- GOJFAKBEASOYNM-UHFFFAOYSA-N 2-(2-aminophenoxy)aniline Chemical compound NC1=CC=CC=C1OC1=CC=CC=C1N GOJFAKBEASOYNM-UHFFFAOYSA-N 0.000 claims 2
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims 2
- 150000001409 amidines Chemical class 0.000 claims 2
- 125000004429 atom Chemical group 0.000 claims 2
- 150000001875 compounds Chemical class 0.000 claims 2
- 230000009261 transgenic effect Effects 0.000 claims 2
- CDAWCLOXVUBKRW-UHFFFAOYSA-N 2-aminophenol Chemical compound NC1=CC=CC=C1O CDAWCLOXVUBKRW-UHFFFAOYSA-N 0.000 claims 1
- IQUPABOKLQSFBK-UHFFFAOYSA-N 2-nitrophenol Chemical class OC1=CC=CC=C1[N+]([O-])=O IQUPABOKLQSFBK-UHFFFAOYSA-N 0.000 claims 1
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 claims 1
- CUHQNMDILUNSTO-UHFFFAOYSA-N N'-(2-chloro-5-methyl-4-phenoxyphenyl)-N-ethyl-N-methylmethanimidamide Chemical compound ClC1=C(C=C(C(=C1)OC1=CC=CC=C1)C)N=CN(C)CC CUHQNMDILUNSTO-UHFFFAOYSA-N 0.000 claims 1
- GSORKECERZGSJX-UHFFFAOYSA-N N-ethyl-N'-(2-fluoro-5-methyl-4-phenoxyphenyl)-N-methylmethanimidamide Chemical compound C(C)N(C=NC1=C(C=C(C(=C1)C)OC1=CC=CC=C1)F)C GSORKECERZGSJX-UHFFFAOYSA-N 0.000 claims 1
- 150000001204 N-oxides Chemical class 0.000 claims 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims 1
- 229910052799 carbon Inorganic materials 0.000 claims 1
- 150000004696 coordination complex Chemical class 0.000 claims 1
- 229910052736 halogen Inorganic materials 0.000 claims 1
- 150000002367 halogens Chemical class 0.000 claims 1
- NVFPHKSEIQNWCE-UHFFFAOYSA-N n'-methylmethanimidamide Chemical compound CNC=N NVFPHKSEIQNWCE-UHFFFAOYSA-N 0.000 claims 1
- 150000005181 nitrobenzenes Chemical class 0.000 claims 1
- 229910052757 nitrogen Inorganic materials 0.000 claims 1
- 229910052760 oxygen Inorganic materials 0.000 claims 1
- 239000001301 oxygen Substances 0.000 claims 1
- 238000002360 preparation method Methods 0.000 claims 1
- 150000003839 salts Chemical class 0.000 claims 1
- 125000004434 sulfur atom Chemical group 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP15175854 | 2015-07-08 | ||
| EP15175854.7 | 2015-07-08 | ||
| PCT/EP2016/065753 WO2017005710A1 (en) | 2015-07-08 | 2016-07-05 | Phenoxyhalogenphenylamidines and the use thereof as fungicides |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2018524341A JP2018524341A (ja) | 2018-08-30 |
| JP2018524341A5 true JP2018524341A5 (https=) | 2019-08-15 |
| JP6811000B2 JP6811000B2 (ja) | 2021-01-13 |
Family
ID=53524681
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017567803A Expired - Fee Related JP6811000B2 (ja) | 2015-07-08 | 2016-07-05 | フェノキシハロゲンフェニルアミジン類及び殺菌剤としてのそれらの使用 |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US10912297B2 (https=) |
| EP (1) | EP3319937A1 (https=) |
| JP (1) | JP6811000B2 (https=) |
| CN (1) | CN107922317A (https=) |
| AR (1) | AR105292A1 (https=) |
| AU (1) | AU2016289731B2 (https=) |
| BR (1) | BR112018000390A2 (https=) |
| CA (1) | CA2991436A1 (https=) |
| IL (1) | IL256455B (https=) |
| MX (1) | MX2018000050A (https=) |
| RU (1) | RU2735177C2 (https=) |
| TW (1) | TWI720993B (https=) |
| UY (1) | UY36781A (https=) |
| WO (1) | WO2017005710A1 (https=) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2020502105A (ja) * | 2016-12-14 | 2020-01-23 | バイエル・クロップサイエンス・アクチェンゲゼルシャフト | フェノキシフェニルアミジンおよびその殺菌剤としての使用 |
| CA3059301A1 (en) | 2017-04-20 | 2018-10-25 | Pi Industries Ltd. | Novel phenylamine compounds |
| WO2018211442A1 (en) | 2017-05-18 | 2018-11-22 | Pi Industries Ltd. | Formimidamidine compounds useful against phytopathogenic microorganisms |
| EP3972414A4 (en) * | 2019-05-23 | 2023-07-26 | Corteva Agriscience LLC | ARYLAMIDINES FUNGICIDES |
| GB202000994D0 (en) | 2020-01-23 | 2020-03-11 | Syngenta Crop Protection Ag | Fungicidal compositions |
| CN115209737B (zh) | 2020-02-27 | 2025-08-15 | 先正达农作物保护股份公司 | 杀真菌组合物 |
| EP3708565A1 (en) | 2020-03-04 | 2020-09-16 | Bayer AG | Pyrimidinyloxyphenylamidines and the use thereof as fungicides |
| WO2021180976A1 (en) | 2020-03-13 | 2021-09-16 | Syngenta Crop Protection Ag | Methods of controlling or preventing infestation of plants by the phytopathogenic microorganism corynespora cassiicola, cercospora sojina and/or cercospora kikuchii |
| US20230112306A1 (en) | 2020-03-13 | 2023-04-13 | Syngenta Crop Protection Ag | Methods of controlling or preventing infestation of soybean plants by the phytopathogenic microorganism corynespora cassiicola |
| BR112022018267A2 (pt) | 2020-03-13 | 2022-10-25 | Syngenta Crop Protection Ag | Métodos de controle ou prevenção de infestação de plantas pelo microrganismo fitopatogênico corynespora cassiicola |
| US20230371512A1 (en) | 2020-10-05 | 2023-11-23 | Syngenta Crop Protection Ag | Fungicidal compositions |
| UY39505A (es) | 2020-11-09 | 2022-06-30 | Syngenta Crop Protection Ag | Composiciones de mezcla fungicida que comprenden un compuesto derivado de la picolinamida como ingrediente activo |
| PY21103556A (es) | 2020-12-02 | 2023-05-03 | Syngenta Crop Protection Ag | Composiciones fungicidas |
| WO2022117650A1 (en) | 2020-12-02 | 2022-06-09 | Syngenta Crop Protection Ag | Fungicidal compositions |
| EP3915971A1 (en) | 2020-12-16 | 2021-12-01 | Bayer Aktiengesellschaft | Phenyl-s(o)n-phenylamidines and the use thereof as fungicides |
| WO2024018016A1 (en) | 2022-07-21 | 2024-01-25 | Syngenta Crop Protection Ag | Crystalline forms of 1,2,4-oxadiazole fungicides |
| WO2025031990A1 (en) | 2023-08-04 | 2025-02-13 | Syngenta Crop Protection Ag | Methods of controlling or preventing infestation of soybean plants by the phytopathogenic microorganism corynespora cassiicola |
| CN121568607A (zh) | 2023-08-04 | 2026-02-24 | 先正达农作物保护股份公司 | 控制或预防植物被植物病原性微生物多主棒孢菌侵染的方法 |
| WO2025031989A1 (en) | 2023-08-04 | 2025-02-13 | Syngenta Crop Protection Ag | Methods of controlling or preventing infestation of plants by the phytopathogenic microorganism corynespora cassiicola |
| WO2025125639A1 (en) | 2023-12-13 | 2025-06-19 | Syngenta Crop Protection Ag | Method of pathogen control in soybean |
Family Cites Families (36)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9902592D0 (en) * | 1999-02-06 | 1999-03-24 | Hoechst Schering Agrevo Gmbh | Fungicides |
| US6800651B2 (en) * | 2000-02-03 | 2004-10-05 | Eli Lilly And Company | Potentiators of glutamate receptors |
| FR2829362B1 (fr) | 2001-09-10 | 2003-11-07 | Aventis Cropscience Sa | Composition fongicide a base de derives d'arylamidine et de composes fongicides connus |
| EP1501789A1 (en) * | 2002-05-03 | 2005-02-02 | E.I. Du Pont De Nemours And Company | Amidinylphenyl compounds and their use as fungicides |
| EP1413301A1 (fr) | 2002-10-24 | 2004-04-28 | Bayer CropScience SA | Médicaments antifongiques à base de dérivés d'arylamidine |
| EP1570736A1 (en) | 2004-03-05 | 2005-09-07 | Bayer CropScience S.A. | Fungicide composition comprising an arylamidine derivative and known fungicide compounds |
| CA2564813A1 (en) | 2004-06-03 | 2005-12-22 | E.I. Du Pont De Nemours And Company | Fungicidal mixtures of amidinylphenyl compounds |
| EP1762669A1 (fr) | 2005-09-13 | 2007-03-14 | Marc Deweerdt | Ensemble de profilés |
| MX2008003432A (es) | 2005-09-13 | 2008-03-27 | Bayer Cropscience Ag | Derivados plaguicidas de bifenilamidina. |
| JP2009507895A (ja) | 2005-09-13 | 2009-02-26 | バイエル・クロツプサイエンス・アクチエンゲゼルシヤフト | 殺虫剤ベンジルオキシ−及びフェネチル−置換フェニル−アミジン誘導体 |
| BRPI0616000B1 (pt) * | 2005-09-13 | 2016-04-19 | Bayer Cropscience Ag | composto derivado de fenil-amidina, processo de preparação de composto, composto derivado de nitrofeniléter, composto derivado de aminofeniléter, método de controle de fungos fitopatogênicos de safras e método de controle de insetos daninhos. |
| EA200800818A1 (ru) | 2005-09-13 | 2008-08-29 | Байер Кропсайенс Аг | Пестицидные производные пиримидинилоксизамещенного фениламидина |
| EP1931200A1 (en) | 2005-09-13 | 2008-06-18 | Bayer CropScience AG | Fungicide composition comprising an arylamidine derivative and two known fungicide compounds |
| EP1931623B1 (en) | 2005-09-13 | 2016-04-13 | Bayer Intellectual Property GmbH | Pesticide naphthyloxy substituted phenylamidine derivatives |
| CN102766110A (zh) | 2005-09-13 | 2012-11-07 | 拜尔农科股份公司 | 农药噻唑氧基取代的苯脒衍生物 |
| ATE510823T1 (de) | 2005-09-13 | 2011-06-15 | Bayer Cropscience Ag | Fungizide pyridinyloxysubstituierte phenylamidinderivate |
| TW200804245A (en) | 2005-11-23 | 2008-01-16 | Du Pont | Amidinylphenyl compounds and their use as fungicides |
| JP2010519267A (ja) | 2007-02-22 | 2010-06-03 | シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト | 新規殺微生物剤 |
| EP1969931A1 (de) | 2007-03-12 | 2008-09-17 | Bayer CropScience Aktiengesellschaft | Fluoalkylphenylamidine und deren Verwendung als Fungizide |
| EP1969934A1 (de) | 2007-03-12 | 2008-09-17 | Bayer CropScience AG | 4-Cycloalkyl-oder 4-arylsubstituierte Phenoxyphenylamidine und deren Verwendung als Fungizide |
| BRPI0808846A2 (pt) | 2007-03-12 | 2019-09-24 | Bayer Cropscience Ag | fenoxifenilamidinas 3-substituídas e seu uso como fungicidas |
| WO2008110281A2 (de) | 2007-03-12 | 2008-09-18 | Bayer Cropscience Ag | 3,4-disubstituierte phenoxyphenylamidine und deren verwendung als fungizide |
| EP1969930A1 (de) | 2007-03-12 | 2008-09-17 | Bayer CropScience AG | Phenoxyphenylamidine und deren Verwendung als Fungizide |
| WO2008110279A1 (de) | 2007-03-12 | 2008-09-18 | Bayer Cropscience Ag | Dihalogenphenoxyphenylamidine und deren verwendung als fungizide |
| BRPI0808734A2 (pt) * | 2007-03-12 | 2014-08-12 | Bayer Cropscience Ag | Uso de n2-fenilamidinas como herbicidas |
| EP1969929A1 (de) | 2007-03-12 | 2008-09-17 | Bayer CropScience AG | Substituierte Phenylamidine und deren Verwendung als Fungizide |
| BRPI0810654B1 (pt) | 2007-04-19 | 2016-10-04 | Bayer Cropscience Ag | tiadiazoliloxifenilamidinas, seu uso e seu método de preparação, composição e método para combate de micro-organismos indesejados, semente resistente a micro-organismo indesejado, bem como método para proteger a dita semente contra micro-organismos |
| BRPI0913885A8 (pt) | 2008-06-27 | 2016-08-02 | Bayer Cropscience Ag | tiadiazoliloxifenilamidinas e seu uso como fungicidas |
| WO2009156098A2 (de) | 2008-06-27 | 2009-12-30 | Bayer Cropscience Ag | Thiadiazolyloxyphenylamidine und deren verwendung als fungizide |
| EP2223917A1 (de) | 2009-02-02 | 2010-09-01 | Bayer CropScience AG | Isothiazolyloxyphenylamidine und deren Verwendung als Fungizide |
| ITMI20101564A1 (it) | 2010-08-23 | 2012-02-24 | Isagro Ricerca Srl | Fenilammidine ad elevata attivita' fungicida e relativo uso |
| US20130296436A1 (en) | 2010-12-27 | 2013-11-07 | Sumitomo Chemical Company, Limited | Amidine compounds and use thereof for plant disease control |
| BR112014014030A2 (pt) | 2011-12-14 | 2017-06-13 | Syngenta Participations Ag | composições fungicidas |
| ITMI20120405A1 (it) | 2012-03-15 | 2013-09-16 | Chemtura Corp | "composizioni sinergiche ad attivita' fungicida e relativo uso" |
| BR112015004968B1 (pt) * | 2012-09-07 | 2020-09-15 | Bayer Cropscience Ag | Combinações fungicidas sinérgicas compreendendo um composto amidina e um inibidor da biossíntese do ergosterol, suas utilizações e métodos para o controle de fungos fitopatogênicos |
| JP6202090B2 (ja) | 2013-03-25 | 2017-09-27 | 住友化学株式会社 | アミジン化合物及びその用途 |
-
2016
- 2016-07-05 WO PCT/EP2016/065753 patent/WO2017005710A1/en not_active Ceased
- 2016-07-05 BR BR112018000390A patent/BR112018000390A2/pt not_active Application Discontinuation
- 2016-07-05 JP JP2017567803A patent/JP6811000B2/ja not_active Expired - Fee Related
- 2016-07-05 AU AU2016289731A patent/AU2016289731B2/en not_active Ceased
- 2016-07-05 RU RU2018104725A patent/RU2735177C2/ru active
- 2016-07-05 CA CA2991436A patent/CA2991436A1/en not_active Abandoned
- 2016-07-05 US US15/742,333 patent/US10912297B2/en not_active Expired - Fee Related
- 2016-07-05 EP EP16736062.7A patent/EP3319937A1/en not_active Withdrawn
- 2016-07-05 MX MX2018000050A patent/MX2018000050A/es unknown
- 2016-07-05 CN CN201680052071.3A patent/CN107922317A/zh active Pending
- 2016-07-06 TW TW105121310A patent/TWI720993B/zh not_active IP Right Cessation
- 2016-07-07 AR ARP160102075A patent/AR105292A1/es active IP Right Grant
- 2016-07-08 UY UY0001036781A patent/UY36781A/es not_active Application Discontinuation
-
2017
- 2017-12-20 IL IL256455A patent/IL256455B/en active IP Right Grant
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