JP2018518506A - 大環状ベンゾジアゼピン二量体、その結合体の製造および使用 - Google Patents

大環状ベンゾジアゼピン二量体、その結合体の製造および使用 Download PDF

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JP2018518506A
JP2018518506A JP2017566642A JP2017566642A JP2018518506A JP 2018518506 A JP2018518506 A JP 2018518506A JP 2017566642 A JP2017566642 A JP 2017566642A JP 2017566642 A JP2017566642 A JP 2017566642A JP 2018518506 A JP2018518506 A JP 2018518506A
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JP2018518506A5 (enExample
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ジャン・ヨン
ロバート・エム・ボルジレリ
アンドリュー・ジェイ・テベン
エリック・エム・スタング
アンドリュー・エフ・ドネル
グレッチェン・エム・シュローダー
ハイディ・エル・ペレス
ドナ・ディ・ウェイ
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Bristol Myers Squibb Co
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Bristol Myers Squibb Co
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
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    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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    • C07K16/3069—Reproductive system, e.g. ovaria, uterus, testes, prostate

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  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
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