JP2018024683A5 - - Google Patents

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Publication number
JP2018024683A5
JP2018024683A5 JP2017170788A JP2017170788A JP2018024683A5 JP 2018024683 A5 JP2018024683 A5 JP 2018024683A5 JP 2017170788 A JP2017170788 A JP 2017170788A JP 2017170788 A JP2017170788 A JP 2017170788A JP 2018024683 A5 JP2018024683 A5 JP 2018024683A5
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JP
Japan
Prior art keywords
oxo
methyl
peak
range
angstroms
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2017170788A
Other languages
English (en)
Japanese (ja)
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JP2018024683A (ja
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Publication date
Application filed filed Critical
Publication of JP2018024683A publication Critical patent/JP2018024683A/ja
Publication of JP2018024683A5 publication Critical patent/JP2018024683A5/ja
Pending legal-status Critical Current

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JP2017170788A 2012-09-26 2017-09-06 逆転写酵素阻害剤の結晶形態 Pending JP2018024683A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261705780P 2012-09-26 2012-09-26
US61/705,780 2012-09-26

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2015534567A Division JP6387349B2 (ja) 2012-09-26 2013-09-20 逆転写酵素阻害剤の結晶形態

Publications (2)

Publication Number Publication Date
JP2018024683A JP2018024683A (ja) 2018-02-15
JP2018024683A5 true JP2018024683A5 (https=) 2018-07-05

Family

ID=50388877

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2015534567A Active JP6387349B2 (ja) 2012-09-26 2013-09-20 逆転写酵素阻害剤の結晶形態
JP2017170788A Pending JP2018024683A (ja) 2012-09-26 2017-09-06 逆転写酵素阻害剤の結晶形態

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2015534567A Active JP6387349B2 (ja) 2012-09-26 2013-09-20 逆転写酵素阻害剤の結晶形態

Country Status (9)

Country Link
US (1) US9150539B2 (https=)
EP (1) EP2900240B1 (https=)
JP (2) JP6387349B2 (https=)
CN (2) CN104684557A (https=)
BR (1) BR112015005997A8 (https=)
CA (1) CA2882947A1 (https=)
ES (1) ES2773105T3 (https=)
MX (1) MX362517B (https=)
WO (1) WO2014052171A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2930585A1 (en) 2013-12-04 2015-06-11 Merck Sharp & Dohme Corp. Process for making reverse transcriptase inhibitors
US11077050B2 (en) 2017-03-24 2021-08-03 Merck Sharp & Dohme Corp. Formulation for parenteral administration
IL294108A (en) * 2019-12-20 2022-08-01 Epizyme Inc Crystalline hydrobromide salt of a ezh2 inhibitor, its preparation and pharmaceutical composition useful for the treatment of cancer

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7309700B2 (en) * 2004-04-02 2007-12-18 Boehringer Ingelheim International Gmbh Crystalline forms of 5,11-dihydro-11-ethyl-5-methyl-8-{2-{(1-oxido-4-quinolinyl)oxy}ethyl}-6H-dipyrido[3,2-b:2′,3′-e] [1,4]diazepin-6-one
WO2006010545A1 (en) * 2004-07-27 2006-02-02 F. Hoffmann-La Roche Ag Benzyltriazolone compounds as non-nucleoside reverse transcriptase inhibitors
BRPI0811988B1 (pt) * 2007-05-30 2021-05-25 F. Hoffmann-La Roche Ag Composto intermediário e processo para preparação de triazolonas
CN101952274A (zh) * 2007-11-20 2011-01-19 默沙东公司 非核苷逆转录酶抑制剂
SI2924034T1 (sl) * 2010-03-30 2017-05-31 Merck Canada Inc. Farmacevtski sestavek, ki obsega nenukleozidni inhibitor reverzne transkriptaze
EP2558093A4 (en) * 2010-04-08 2013-10-02 Merck Sharp & Dohme PRODRUGS OF HIV INVERTER TRANSCRIPTASE INHIBITOR

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