JP2017509691A5 - - Google Patents
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- Publication number
- JP2017509691A5 JP2017509691A5 JP2016565103A JP2016565103A JP2017509691A5 JP 2017509691 A5 JP2017509691 A5 JP 2017509691A5 JP 2016565103 A JP2016565103 A JP 2016565103A JP 2016565103 A JP2016565103 A JP 2016565103A JP 2017509691 A5 JP2017509691 A5 JP 2017509691A5
- Authority
- JP
- Japan
- Prior art keywords
- film coating
- coating composition
- medium chain
- pva
- polymer
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 239000000203 mixture Substances 0.000 claims 21
- 239000007888 film coating Substances 0.000 claims 19
- 238000009501 film coating Methods 0.000 claims 19
- PEDCQBHIVMGVHV-UHFFFAOYSA-N Glycerol Natural products OCC(O)CO PEDCQBHIVMGVHV-UHFFFAOYSA-N 0.000 claims 10
- 239000004372 Polyvinyl alcohol Substances 0.000 claims 5
- 125000005456 glyceride group Chemical group 0.000 claims 5
- 229920002451 polyvinyl alcohol Polymers 0.000 claims 5
- 235000011187 glycerol Nutrition 0.000 claims 4
- 229920000642 polymer Polymers 0.000 claims 4
- 239000007900 aqueous suspension Substances 0.000 claims 3
- 239000000314 lubricant Substances 0.000 claims 3
- 239000000843 powder Substances 0.000 claims 3
- 239000000758 substrate Substances 0.000 claims 3
- 239000004094 surface-active agent Substances 0.000 claims 3
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical group [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 claims 2
- DBMJMQXJHONAFJ-UHFFFAOYSA-M Sodium laurylsulphate Chemical compound [Na+].CCCCCCCCCCCCOS([O-])(=O)=O DBMJMQXJHONAFJ-UHFFFAOYSA-M 0.000 claims 2
- 229910052799 carbon Inorganic materials 0.000 claims 2
- GHVNFZFCNZKVNT-UHFFFAOYSA-N decanoic acid Chemical compound CCCCCCCCCC(O)=O GHVNFZFCNZKVNT-UHFFFAOYSA-N 0.000 claims 2
- 229920003088 hydroxypropyl methyl cellulose Polymers 0.000 claims 2
- WWZKQHOCKIZLMA-UHFFFAOYSA-N octanoic acid Chemical compound CCCCCCCC(O)=O WWZKQHOCKIZLMA-UHFFFAOYSA-N 0.000 claims 2
- GHBFNMLVSPCDGN-UHFFFAOYSA-N rac-1-monooctanoylglycerol Chemical compound CCCCCCCC(=O)OCC(O)CO GHBFNMLVSPCDGN-UHFFFAOYSA-N 0.000 claims 2
- 235000019333 sodium laurylsulphate Nutrition 0.000 claims 2
- 239000000454 talc Substances 0.000 claims 2
- 229910052623 talc Inorganic materials 0.000 claims 2
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 claims 2
- 239000005995 Aluminium silicate Substances 0.000 claims 1
- 239000005632 Capric acid (CAS 334-48-5) Substances 0.000 claims 1
- 239000005635 Caprylic acid (CAS 124-07-2) Substances 0.000 claims 1
- 229920002153 Hydroxypropyl cellulose Polymers 0.000 claims 1
- DPXJVFZANSGRMM-UHFFFAOYSA-N acetic acid;2,3,4,5,6-pentahydroxyhexanal;sodium Chemical compound [Na].CC(O)=O.OCC(O)C(O)C(O)C(O)C=O DPXJVFZANSGRMM-UHFFFAOYSA-N 0.000 claims 1
- 239000000654 additive Substances 0.000 claims 1
- 235000012211 aluminium silicate Nutrition 0.000 claims 1
- 239000001768 carboxy methyl cellulose Substances 0.000 claims 1
- 229920001577 copolymer Polymers 0.000 claims 1
- 150000005690 diesters Chemical class 0.000 claims 1
- 239000006185 dispersion Substances 0.000 claims 1
- -1 glycerol triester Chemical class 0.000 claims 1
- 239000001863 hydroxypropyl cellulose Substances 0.000 claims 1
- 235000010977 hydroxypropyl cellulose Nutrition 0.000 claims 1
- 239000001866 hydroxypropyl methyl cellulose Substances 0.000 claims 1
- 235000010979 hydroxypropyl methyl cellulose Nutrition 0.000 claims 1
- 229960003943 hypromellose Drugs 0.000 claims 1
- 239000012729 immediate-release (IR) formulation Substances 0.000 claims 1
- NLYAJNPCOHFWQQ-UHFFFAOYSA-N kaolin Chemical compound O.O.O=[Al]O[Si](=O)O[Si](=O)O[Al]=O NLYAJNPCOHFWQQ-UHFFFAOYSA-N 0.000 claims 1
- 238000004519 manufacturing process Methods 0.000 claims 1
- 229960002446 octanoic acid Drugs 0.000 claims 1
- 239000000049 pigment Substances 0.000 claims 1
- 235000019422 polyvinyl alcohol Nutrition 0.000 claims 1
- 235000019812 sodium carboxymethyl cellulose Nutrition 0.000 claims 1
- 229920001027 sodium carboxymethylcellulose Polymers 0.000 claims 1
- 230000004584 weight gain Effects 0.000 claims 1
- 235000019786 weight gain Nutrition 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201461929735P | 2014-01-21 | 2014-01-21 | |
| US61/929,735 | 2014-01-21 | ||
| PCT/US2015/011422 WO2015112400A1 (en) | 2014-01-21 | 2015-01-14 | Immediate release film coatings containing medium chain glycerides and substrates coated therewith |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017509691A JP2017509691A (ja) | 2017-04-06 |
| JP2017509691A5 true JP2017509691A5 (https=) | 2018-02-01 |
| JP6541687B2 JP6541687B2 (ja) | 2019-07-10 |
Family
ID=53543848
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016565103A Active JP6541687B2 (ja) | 2014-01-21 | 2015-01-14 | 中鎖グリセリドを含有する即時放出フィルムコーティング、及びそれによってコーティングされている基材 |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US9504654B2 (https=) |
| EP (1) | EP3096891B1 (https=) |
| JP (1) | JP6541687B2 (https=) |
| KR (1) | KR102287342B1 (https=) |
| CN (1) | CN105916598B (https=) |
| AU (1) | AU2015209674B2 (https=) |
| BR (1) | BR112016016623B1 (https=) |
| CA (1) | CA2933202C (https=) |
| ES (1) | ES2802156T3 (https=) |
| HU (1) | HUE049598T2 (https=) |
| MX (1) | MX378845B (https=) |
| PL (1) | PL3096891T3 (https=) |
| RU (1) | RU2686183C2 (https=) |
| WO (1) | WO2015112400A1 (https=) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR102158339B1 (ko) * | 2016-02-05 | 2020-09-21 | 삼진제약주식회사 | 인습성이 개선된 카르베딜롤 속방성 제제 |
| RU2753049C2 (ru) * | 2016-08-04 | 2021-08-11 | БиПиЭсАй ХОЛДИНГЗ, ЭлЭлСи | Легкие для глотания покрытия и покрытые ими субстраты |
| US20180338922A1 (en) * | 2017-05-26 | 2018-11-29 | Esperion Therapeutics, Inc. | Fixed dose formulations |
| TR201721437A2 (tr) * | 2017-12-25 | 2019-07-22 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Fesoterodi̇ni̇n modi̇fi̇ye salim sağlayan formülasyonlari |
| KR102103530B1 (ko) | 2018-06-29 | 2020-04-22 | 주식회사 코피텍 | 필름 코팅용 조성물 및 이를 코팅한 정제 |
| KR102265977B1 (ko) | 2018-07-16 | 2021-06-16 | 주식회사 코피텍 | 방습성이 개선된 필름 코팅용 조성물 및 이를 코팅한 정제 |
| JPWO2023063296A1 (https=) * | 2021-10-11 | 2023-04-20 |
Family Cites Families (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS57171428A (en) * | 1981-04-13 | 1982-10-22 | Sankyo Co Ltd | Preparation of coated solid preparation |
| DE3220434A1 (de) | 1982-05-29 | 1983-12-01 | Robert Bosch Gmbh, 7000 Stuttgart | Verfahren zur ueberwachung einer messgroesse |
| JPS5973529A (ja) | 1982-10-12 | 1984-04-25 | Sankyo Co Ltd | 被覆固形製剤の製造法 |
| JPS59193831A (ja) * | 1983-04-18 | 1984-11-02 | Sankyo Co Ltd | 腸溶性製剤の製造法 |
| US6248363B1 (en) * | 1999-11-23 | 2001-06-19 | Lipocine, Inc. | Solid carriers for improved delivery of active ingredients in pharmaceutical compositions |
| US6448323B1 (en) * | 1999-07-09 | 2002-09-10 | Bpsi Holdings, Inc. | Film coatings and film coating compositions based on polyvinyl alcohol |
| KR100425226B1 (ko) * | 2001-07-03 | 2004-03-30 | 주식회사 팜트리 | 아세클로페낙을 함유하는 경제적인 경구용 제제의 조성 및제법 |
| EP1465592A2 (en) * | 2001-12-19 | 2004-10-13 | Alza Corporation | Formulation and dosage form for increasing oral bioavailability of hydrophilic macromolecules |
| FR2838647B1 (fr) * | 2002-04-23 | 2006-02-17 | Particules enrobees a liberation prolongee, leur procede de preparation et comprimes les contenant | |
| DE10311585A1 (de) * | 2003-03-14 | 2004-09-23 | Basf Ag | Wirkstoffhaltige Adsorbate |
| MXPA06010488A (es) | 2004-03-31 | 2006-12-19 | Bpsi Holdings Inc | Revestimientos entericos para sustratos oralmente ingeribles. |
| TWI354569B (en) * | 2004-05-28 | 2011-12-21 | Bristol Myers Squibb Co | Coated tablet formulation and method |
| US20080096979A1 (en) * | 2004-11-08 | 2008-04-24 | Rubicon Research Pvt. Ltd. | Aqueous Pharmaceutical Coating |
| WO2006111980A2 (en) | 2005-04-20 | 2006-10-26 | Ideal Cures Pvt. Ltd. | Pva based film coating and film coating compositions |
| JP2007217390A (ja) * | 2006-02-20 | 2007-08-30 | Hitoshi Ichihashi | カプリロカプロイルマクロゴール−８グリセリドを含む医薬組成物 |
| US20080181928A1 (en) | 2006-12-22 | 2008-07-31 | Miv Therapeutics, Inc. | Coatings for implantable medical devices for liposome delivery |
| BRPI0919249B1 (pt) | 2008-09-25 | 2017-12-19 | Isp Investments Inc. | Coating composition, method for coating solids and coated product |
| TWI438012B (zh) | 2008-12-25 | 2014-05-21 | Toray Industries | 固態製劑用之塗覆劑及使用其之固態製劑 |
| WO2010112965A1 (en) * | 2009-03-30 | 2010-10-07 | Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi | Isolation coating of diclofenac tablets |
| WO2010122583A2 (en) | 2009-04-24 | 2010-10-28 | Rubicon Research Private Limited | Oral pharmaceutical compositions of acid labile substances |
| KR101783945B1 (ko) * | 2009-05-12 | 2017-10-10 | 비피에스아이 홀딩스, 엘엘씨. | 향상된 수분차단 속방출형 필름의 코팅 시스템 및 이에 의하여 코팅된 기재 |
| KR20120033305A (ko) * | 2009-05-12 | 2012-04-06 | 비피에스아이 홀딩스, 엘엘씨. | 미립자인 비점착제를 포함하는 필름 코팅 및 상기 필름코팅이 코팅된 기재 |
| SG10201500152UA (en) * | 2009-12-22 | 2015-03-30 | Abbvie Inc | Abt-263 capsule |
| US20130095141A1 (en) * | 2010-03-08 | 2013-04-18 | Beverly A. Schad | Food grade dry film coating composition and methods of making and using the same |
| WO2012120364A2 (en) * | 2011-03-09 | 2012-09-13 | Ideal Cures Pvt. Ltd. | Novel immediate release film coating compositions |
| US20150320679A1 (en) * | 2012-12-12 | 2015-11-12 | Leo Laboratories Limited | Gel compositions |
| WO2014096983A1 (en) * | 2012-12-21 | 2014-06-26 | Wockhardt Limited | Stable pharmaceutical compositions of saxagliptin or salts thereof |
| GB201319792D0 (en) * | 2013-11-08 | 2013-12-25 | Sigmoid Pharma Ltd | Formulations |
-
2015
- 2015-01-14 RU RU2016133221A patent/RU2686183C2/ru active
- 2015-01-14 CA CA2933202A patent/CA2933202C/en active Active
- 2015-01-14 WO PCT/US2015/011422 patent/WO2015112400A1/en not_active Ceased
- 2015-01-14 AU AU2015209674A patent/AU2015209674B2/en active Active
- 2015-01-14 KR KR1020167017556A patent/KR102287342B1/ko active Active
- 2015-01-14 JP JP2016565103A patent/JP6541687B2/ja active Active
- 2015-01-14 HU HUE15740927A patent/HUE049598T2/hu unknown
- 2015-01-14 BR BR112016016623-0A patent/BR112016016623B1/pt active IP Right Grant
- 2015-01-14 US US14/597,025 patent/US9504654B2/en active Active
- 2015-01-14 PL PL15740927T patent/PL3096891T3/pl unknown
- 2015-01-14 CN CN201580005058.8A patent/CN105916598B/zh active Active
- 2015-01-14 ES ES15740927T patent/ES2802156T3/es active Active
- 2015-01-14 EP EP15740927.7A patent/EP3096891B1/en active Active
- 2015-01-14 MX MX2016008583A patent/MX378845B/es unknown
-
2016
- 2016-10-24 US US15/332,319 patent/US9789067B2/en active Active
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