CN105916598B - 含有中链甘油酯的即释型膜包衣及用其包被的基质 - Google Patents

含有中链甘油酯的即释型膜包衣及用其包被的基质 Download PDF

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Publication number
CN105916598B
CN105916598B CN201580005058.8A CN201580005058A CN105916598B CN 105916598 B CN105916598 B CN 105916598B CN 201580005058 A CN201580005058 A CN 201580005058A CN 105916598 B CN105916598 B CN 105916598B
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China
Prior art keywords
film coating
coating composition
medium chain
glycerides
chain glycerides
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CN201580005058.8A
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English (en)
Chinese (zh)
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CN105916598A (zh
Inventor
J·特克伊
B·J·普鲁萨克
J·R·金贝儿
D·杜
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BPSI Holdings LLC
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BPSI Holdings LLC
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2813—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/282—Organic compounds, e.g. fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2893—Tablet coating processes
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08J—WORKING-UP; GENERAL PROCESSES OF COMPOUNDING; AFTER-TREATMENT NOT COVERED BY SUBCLASSES C08B, C08C, C08F, C08G or C08H
    • C08J3/00—Processes of treating or compounding macromolecular substances
    • C08J3/02—Making solutions, dispersions, lattices or gels by other methods than by solution, emulsion or suspension polymerisation techniques
    • C08J3/03—Making solutions, dispersions, lattices or gels by other methods than by solution, emulsion or suspension polymerisation techniques in aqueous media

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Inorganic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Polymers & Plastics (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Paints Or Removers (AREA)
  • Application Of Or Painting With Fluid Materials (AREA)
CN201580005058.8A 2014-01-21 2015-01-14 含有中链甘油酯的即释型膜包衣及用其包被的基质 Active CN105916598B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201461929735P 2014-01-21 2014-01-21
US61/929,735 2014-01-21
PCT/US2015/011422 WO2015112400A1 (en) 2014-01-21 2015-01-14 Immediate release film coatings containing medium chain glycerides and substrates coated therewith

Publications (2)

Publication Number Publication Date
CN105916598A CN105916598A (zh) 2016-08-31
CN105916598B true CN105916598B (zh) 2020-07-17

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CN201580005058.8A Active CN105916598B (zh) 2014-01-21 2015-01-14 含有中链甘油酯的即释型膜包衣及用其包被的基质

Country Status (14)

Country Link
US (2) US9504654B2 (https=)
EP (1) EP3096891B1 (https=)
JP (1) JP6541687B2 (https=)
KR (1) KR102287342B1 (https=)
CN (1) CN105916598B (https=)
AU (1) AU2015209674B2 (https=)
BR (1) BR112016016623B1 (https=)
CA (1) CA2933202C (https=)
ES (1) ES2802156T3 (https=)
HU (1) HUE049598T2 (https=)
MX (1) MX378845B (https=)
PL (1) PL3096891T3 (https=)
RU (1) RU2686183C2 (https=)
WO (1) WO2015112400A1 (https=)

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KR102158339B1 (ko) * 2016-02-05 2020-09-21 삼진제약주식회사 인습성이 개선된 카르베딜롤 속방성 제제
RU2753049C2 (ru) * 2016-08-04 2021-08-11 БиПиЭсАй ХОЛДИНГЗ, ЭлЭлСи Легкие для глотания покрытия и покрытые ими субстраты
US20180338922A1 (en) * 2017-05-26 2018-11-29 Esperion Therapeutics, Inc. Fixed dose formulations
TR201721437A2 (tr) * 2017-12-25 2019-07-22 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Fesoterodi̇ni̇n modi̇fi̇ye salim sağlayan formülasyonlari
KR102103530B1 (ko) 2018-06-29 2020-04-22 주식회사 코피텍 필름 코팅용 조성물 및 이를 코팅한 정제
KR102265977B1 (ko) 2018-07-16 2021-06-16 주식회사 코피텍 방습성이 개선된 필름 코팅용 조성물 및 이를 코팅한 정제
JPWO2023063296A1 (https=) * 2021-10-11 2023-04-20

Citations (1)

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CN102421421A (zh) * 2009-05-12 2012-04-18 Bpsi控股有限责任公司 含有抗黏性剂细微颗粒的包衣和覆有该包衣的基体

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JPS59193831A (ja) * 1983-04-18 1984-11-02 Sankyo Co Ltd 腸溶性製剤の製造法
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KR100425226B1 (ko) * 2001-07-03 2004-03-30 주식회사 팜트리 아세클로페낙을 함유하는 경제적인 경구용 제제의 조성 및제법
EP1465592A2 (en) * 2001-12-19 2004-10-13 Alza Corporation Formulation and dosage form for increasing oral bioavailability of hydrophilic macromolecules
FR2838647B1 (fr) * 2002-04-23 2006-02-17 Particules enrobees a liberation prolongee, leur procede de preparation et comprimes les contenant
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CN102421421A (zh) * 2009-05-12 2012-04-18 Bpsi控股有限责任公司 含有抗黏性剂细微颗粒的包衣和覆有该包衣的基体

Also Published As

Publication number Publication date
JP6541687B2 (ja) 2019-07-10
US9504654B2 (en) 2016-11-29
AU2015209674B2 (en) 2018-11-08
MX378845B (es) 2025-03-10
KR102287342B1 (ko) 2021-08-06
AU2015209674A1 (en) 2016-06-23
CA2933202C (en) 2022-05-31
US20170035697A1 (en) 2017-02-09
RU2016133221A (ru) 2018-03-02
WO2015112400A1 (en) 2015-07-30
BR112016016623B1 (pt) 2022-02-01
RU2016133221A3 (https=) 2018-07-17
US20150202160A1 (en) 2015-07-23
EP3096891B1 (en) 2020-04-08
ES2802156T3 (es) 2021-01-15
EP3096891A1 (en) 2016-11-30
CA2933202A1 (en) 2015-07-30
PL3096891T3 (pl) 2020-08-24
BR112016016623A2 (https=) 2017-08-08
JP2017509691A (ja) 2017-04-06
MX2016008583A (es) 2017-02-02
RU2686183C2 (ru) 2019-04-24
HUE049598T2 (hu) 2020-09-28
KR20160111375A (ko) 2016-09-26
EP3096891A4 (en) 2017-10-04
CN105916598A (zh) 2016-08-31
US9789067B2 (en) 2017-10-17

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