JP2017105793A5 - - Google Patents

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Publication number
JP2017105793A5
JP2017105793A5 JP2017006285A JP2017006285A JP2017105793A5 JP 2017105793 A5 JP2017105793 A5 JP 2017105793A5 JP 2017006285 A JP2017006285 A JP 2017006285A JP 2017006285 A JP2017006285 A JP 2017006285A JP 2017105793 A5 JP2017105793 A5 JP 2017105793A5
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JP
Japan
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compound
following formula
pharmaceutical composition
salt
formula
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JP2017006285A
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English (en)
Japanese (ja)
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JP6550083B2 (ja
JP2017105793A (ja
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Publication of JP2017105793A publication Critical patent/JP2017105793A/ja
Publication of JP2017105793A5 publication Critical patent/JP2017105793A5/ja
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Publication of JP6550083B2 publication Critical patent/JP6550083B2/ja
Expired - Fee Related legal-status Critical Current
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JP2017006285A 2013-09-27 2017-01-18 Hivインテグラーゼ阻害薬として有用な置換されたキノリジン誘導体 Expired - Fee Related JP6550083B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361883463P 2013-09-27 2013-09-27
US61/883,463 2013-09-27

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2016516931A Division JP6081662B2 (ja) 2013-09-27 2014-09-26 Hivインテグラーゼ阻害薬として有用な置換されたキノリジン誘導体

Publications (3)

Publication Number Publication Date
JP2017105793A JP2017105793A (ja) 2017-06-15
JP2017105793A5 true JP2017105793A5 (enExample) 2017-09-07
JP6550083B2 JP6550083B2 (ja) 2019-07-24

Family

ID=52744477

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2016516931A Expired - Fee Related JP6081662B2 (ja) 2013-09-27 2014-09-26 Hivインテグラーゼ阻害薬として有用な置換されたキノリジン誘導体
JP2017006285A Expired - Fee Related JP6550083B2 (ja) 2013-09-27 2017-01-18 Hivインテグラーゼ阻害薬として有用な置換されたキノリジン誘導体

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2016516931A Expired - Fee Related JP6081662B2 (ja) 2013-09-27 2014-09-26 Hivインテグラーゼ阻害薬として有用な置換されたキノリジン誘導体

Country Status (31)

Country Link
US (2) US9861620B2 (enExample)
EP (1) EP3049081B1 (enExample)
JP (2) JP6081662B2 (enExample)
KR (2) KR101809392B1 (enExample)
CN (1) CN105744936B (enExample)
AP (1) AP2016009157A0 (enExample)
AU (1) AU2014324829B2 (enExample)
BR (1) BR112016006651B8 (enExample)
CA (1) CA2924829C (enExample)
CL (1) CL2016000698A1 (enExample)
CR (1) CR20160140A (enExample)
DO (1) DOP2016000069A (enExample)
EA (1) EA030695B1 (enExample)
EC (1) ECSP16016726A (enExample)
ES (1) ES2768658T3 (enExample)
GT (1) GT201600056A (enExample)
HK (1) HK1221648A1 (enExample)
IL (1) IL244438B (enExample)
MA (1) MA38922A3 (enExample)
MD (1) MD4794B1 (enExample)
MX (1) MX367057B (enExample)
NI (1) NI201600040A (enExample)
PE (1) PE20160501A1 (enExample)
PH (1) PH12016500553B1 (enExample)
SA (1) SA516370826B1 (enExample)
SG (1) SG11201602217XA (enExample)
SV (1) SV2016005171A (enExample)
TN (1) TN2016000090A1 (enExample)
UA (1) UA117499C2 (enExample)
WO (1) WO2015048363A1 (enExample)
ZA (1) ZA201601708B (enExample)

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TWI695003B (zh) 2014-12-23 2020-06-01 美商基利科學股份有限公司 多環胺甲醯基吡啶酮化合物及其醫藥用途
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RS65891B1 (sr) 2018-05-31 2024-09-30 Shionogi & Co Policiklični karbamoilpiridonski derivati za lečenje hiv-a
PE20201414A1 (es) 2018-05-31 2020-12-07 Shionogi & Co Derivado policiclico de piridona
LT3938047T (lt) 2019-03-22 2022-10-10 Gilead Sciences, Inc. Tilteliniai tricikliniai karbamoilpiridono junginiai ir jų naudojimas farmacijoje
US20200398978A1 (en) 2019-06-20 2020-12-24 Bell Helicopter Textron Inc. Low-drag rotor blade extension
MA57224B1 (fr) 2019-07-31 2022-10-31 Advanced Biodesign Aminothiolesters et leurs utilisations
CN112521386B (zh) * 2019-09-19 2023-05-26 周雨恬 具有抗病毒作用的多环吡啶酮化合物及其药物组合和用途
TWI902729B (zh) 2019-11-28 2025-11-01 日商鹽野義製藥股份有限公司 以組合整合酶阻礙劑及抗hiv藥為特徵之hiv感染症的預防及治療用醫藥
WO2021107065A1 (ja) 2019-11-28 2021-06-03 塩野義製薬株式会社 多環性ピリドピラジン誘導体
BR112022015771A2 (pt) 2020-02-24 2022-10-11 Gilead Sciences Inc Compostos tetracíclicos para tratar a infecção por hiv
TW202222798A (zh) 2020-09-30 2022-06-16 美商基利科學股份有限公司 橋接三環胺甲醯基吡啶酮化合物及其用途
PT4196479T (pt) 2021-01-19 2024-01-03 Gilead Sciences Inc Compostos de piridotriazinas substituídos e suas utilizações
FR3119314B1 (fr) 2021-01-29 2025-01-10 Advanced Biodesign Nanocapsule lipidique comprenant au moins un composé aminothiolester ou un de ses dérivés pharmaceutiquement acceptable
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