JP2016536370A5 - - Google Patents

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JP2016536370A5
JP2016536370A5 JP2016552486A JP2016552486A JP2016536370A5 JP 2016536370 A5 JP2016536370 A5 JP 2016536370A5 JP 2016552486 A JP2016552486 A JP 2016552486A JP 2016552486 A JP2016552486 A JP 2016552486A JP 2016536370 A5 JP2016536370 A5 JP 2016536370A5
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JP
Japan
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equivalents
tris
salt
hydroxymethyl
bases
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JP2016552486A
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English (en)
Japanese (ja)
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JP6535338B2 (ja
JP2016536370A (ja
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Priority claimed from PCT/US2014/064441 external-priority patent/WO2015069956A2/en
Publication of JP2016536370A publication Critical patent/JP2016536370A/ja
Publication of JP2016536370A5 publication Critical patent/JP2016536370A5/ja
Priority to JP2019102367A priority Critical patent/JP6957557B2/ja
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Publication of JP6535338B2 publication Critical patent/JP6535338B2/ja
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JP2016552486A 2013-11-06 2014-11-06 新規製剤 Active JP6535338B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2019102367A JP6957557B2 (ja) 2013-11-06 2019-05-31 新規製剤

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201361900919P 2013-11-06 2013-11-06
US201361900946P 2013-11-06 2013-11-06
US201361900878P 2013-11-06 2013-11-06
US61/900,946 2013-11-06
US61/900,878 2013-11-06
US61/900,919 2013-11-06
PCT/US2014/064441 WO2015069956A2 (en) 2013-11-06 2014-11-06 Novel formulations

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2019102367A Division JP6957557B2 (ja) 2013-11-06 2019-05-31 新規製剤

Publications (3)

Publication Number Publication Date
JP2016536370A JP2016536370A (ja) 2016-11-24
JP2016536370A5 true JP2016536370A5 (enExample) 2018-01-18
JP6535338B2 JP6535338B2 (ja) 2019-06-26

Family

ID=53042097

Family Applications (4)

Application Number Title Priority Date Filing Date
JP2016552485A Ceased JP2016535787A (ja) 2013-11-06 2014-11-06 新規方法
JP2016552486A Active JP6535338B2 (ja) 2013-11-06 2014-11-06 新規製剤
JP2019102367A Active JP6957557B2 (ja) 2013-11-06 2019-05-31 新規製剤
JP2021164647A Pending JP2022003084A (ja) 2013-11-06 2021-10-06 新規製剤

Family Applications Before (1)

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JP2016552485A Ceased JP2016535787A (ja) 2013-11-06 2014-11-06 新規方法

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2019102367A Active JP6957557B2 (ja) 2013-11-06 2019-05-31 新規製剤
JP2021164647A Pending JP2022003084A (ja) 2013-11-06 2021-10-06 新規製剤

Country Status (14)

Country Link
US (9) US20160279155A1 (enExample)
EP (3) EP3065729A4 (enExample)
JP (4) JP2016535787A (enExample)
KR (1) KR20160079109A (enExample)
CN (3) CN112402434A (enExample)
AU (2) AU2014346682B2 (enExample)
CA (1) CA2929821A1 (enExample)
ES (1) ES2834131T3 (enExample)
HK (1) HK1224228A1 (enExample)
IL (1) IL245420B (enExample)
MX (2) MX386250B (enExample)
RU (1) RU2691951C2 (enExample)
SG (1) SG11201604153UA (enExample)
WO (3) WO2015069948A1 (enExample)

Families Citing this family (8)

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JP2021023226A (ja) * 2019-08-06 2021-02-22 学校法人慶應義塾 アクアポリン活性調節剤候補のハイスループットスクリーニング方法
CN110790787B (zh) * 2019-11-12 2022-06-14 广东药科大学 一类水溶性前药、其制备方法及其作为药物的用途
IL300341A (en) * 2020-08-05 2023-04-01 Jiangsu Simcere Pharm Co Ltd A pharmaceutical composition of an aquaporin inhibitor and a method for its preparation
CN117105810B (zh) * 2023-10-23 2024-02-09 中国农业大学 一种具有广谱抗菌活性的化合物及其抗菌组合物
CN118178653A (zh) * 2024-03-22 2024-06-14 山东第一医科大学附属省立医院(山东省立医院) 跨膜水交换蛋白aqp4抑制剂在制备抗肿瘤药物上的应用

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