JP2016529228A5 - - Google Patents
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- JP2016529228A5 JP2016529228A5 JP2016525422A JP2016525422A JP2016529228A5 JP 2016529228 A5 JP2016529228 A5 JP 2016529228A5 JP 2016525422 A JP2016525422 A JP 2016525422A JP 2016525422 A JP2016525422 A JP 2016525422A JP 2016529228 A5 JP2016529228 A5 JP 2016529228A5
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- Prior art keywords
- compound
- hypotension
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- disorder
- isotopically enriched
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| MY194181A (en) * | 2016-08-30 | 2022-11-17 | Theravance Biopharma R&D Ip Llc | Compound for use in the treatment of neurogenic orthostatic hypotension |
| GB2566516A (en) | 2017-09-15 | 2019-03-20 | Univ Oxford Innovation Ltd | Electrochemical recognition and quantification of cytochrome c oxidase expression in bacteria |
| GB2571696B (en) | 2017-10-09 | 2020-05-27 | Compass Pathways Ltd | Large scale method for the preparation of Psilocybin and formulations of Psilocybin so produced |
| US12459965B2 (en) | 2017-10-09 | 2025-11-04 | Compass Pathfinder Limited | Preparation of psilocybin, different polymorphic forms, intermediates, formulations and their use |
| EP3946329A4 (en) | 2019-03-27 | 2022-11-30 | Curasen Therapeutics, Inc. | BETA ADRENE AGONIST AND METHODS OF USE |
| JP2022529781A (ja) | 2019-04-17 | 2022-06-24 | コンパス パスファインダー リミテッド | サイロシビンによるうつ病及び他の様々な障害の治療 |
| JP7737367B2 (ja) * | 2019-10-25 | 2025-09-10 | キュラセン セラピューティクス インコーポレイテッド | α１Ａ－ＡＲ部分アゴニストを用いて神経障害を治療するための方法 |
| WO2021247963A1 (en) * | 2020-06-05 | 2021-12-09 | Senda Biosciences, Inc. | (s)-alpha-fluoromethyltyrosine as decarboxylase inhibitors for use in the treatment of hypotension |
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| DE3360726D1 (en) * | 1982-01-14 | 1985-10-17 | Sumitomo Chemical Co | Process for producing threo-3-(3,4-dihydroxyphenyl)serine |
| CA1223602A (en) | 1983-05-25 | 1987-06-30 | Naohito Ohashi | Process for producing 3-(3,4-dihydroxyphenyl) serine |
| JP3764179B2 (ja) | 1994-07-05 | 2006-04-05 | 克寛 西野 | 運動・意識または言語障害の機能改善剤 |
| DE19619510A1 (de) | 1995-05-18 | 1996-11-21 | Sumitomo Chemical Co | Verfahren zur Herstellung von Threo-3-(3,4-dihydroxyphenyl)serin |
| JP3489319B2 (ja) | 1996-03-12 | 2004-01-19 | 住友化学工業株式会社 | カルボン酸誘導体、その製造法および用途 |
| JPH115738A (ja) | 1997-06-15 | 1999-01-12 | Katsuhiro Nishino | 脳虚血に伴う神経脱落症状の予防剤および超急性期治療剤 |
| US6376531B1 (en) * | 1998-11-13 | 2002-04-23 | Rupert Charles Bell | Method of treatment using deuterium compounds |
| DE10261807A1 (de) * | 2002-12-19 | 2004-07-01 | Turicum Drug Development Ag | Deuterierte Catecholaminderivate sowie diese Verbindungen enthaltende Arzneimittel |
| WO2005084330A2 (en) | 2004-03-02 | 2005-09-15 | Synergia Pharma, Inc. | Compositions and methods for treating nasal congestion |
| USRE46555E1 (en) * | 2006-02-17 | 2017-09-19 | Teva Pharmaceuticals International Gmbh | Deuterated catecholamine derivatives and medicaments comprising said compounds |
| US8008285B2 (en) | 2007-03-09 | 2011-08-30 | Chelsea Therapeutics, Inc. | Droxidopa and pharmaceutical composition thereof for the treatment of fibromyalgia |
| ES2395868T3 (es) | 2007-03-12 | 2013-02-15 | Chelsea Therapeutics, Inc. | Droxidopa y composición farmacéutica de la misma para el tratamiento de la hipotensión mediada neuralmente |
| NZ581707A (en) | 2007-05-07 | 2011-05-27 | Chelsea Therapeutics Inc | Droxidopa and pharmaceutical composition thereof for the treatment of mood disorders, sleep disorders, or attention deficit disorders |
| US7745665B2 (en) | 2007-06-04 | 2010-06-29 | Auspex Pharmaceuticals, Inc. | Substituted phenethylamines |
| WO2010054286A2 (en) * | 2008-11-10 | 2010-05-14 | Auspex Pharmaceuticals, Inc. | Substituted hydroxyphenylamine compounds |
| US9072730B2 (en) | 2009-05-14 | 2015-07-07 | The Board Of Trustees Of The Leland Stanford Junior University | Method of improving cognitive functions in individuals with down syndrome and/or alzheimer's disease |
| JPWO2011001976A1 (ja) | 2009-07-01 | 2012-12-13 | 大日本住友製薬株式会社 | スレオ−３−（３，４−ジヒドロキシフェニル）−ｌ−セリンの製造法 |
| JP5880913B2 (ja) | 2011-05-17 | 2016-03-09 | 三郎 佐古田 | パーキンソン病の体幹症状（姿勢反射異常）の治療剤 |
| US20130253061A1 (en) | 2012-03-20 | 2013-09-26 | Chelsea Therapeutics, Inc. | Method of droxidopa synthesis |
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2014
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- 2014-07-08 AU AU2014287418A patent/AU2014287418A1/en not_active Abandoned
- 2014-07-08 MX MX2016000219A patent/MX384131B/es unknown
- 2014-07-08 EA EA201600093A patent/EA201600093A1/ru unknown
- 2014-07-08 CA CA2917159A patent/CA2917159C/en active Active
- 2014-07-08 PE PE2016000010A patent/PE20160556A1/es unknown
- 2014-07-08 SG SG11201510764QA patent/SG11201510764QA/en unknown
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- 2014-07-08 WO PCT/US2014/045731 patent/WO2015006315A1/en not_active Ceased
- 2014-07-08 EP EP19188210.9A patent/EP3611159B1/en active Active
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- 2014-07-08 EP EP14822407.4A patent/EP3019467A4/en not_active Withdrawn
- 2014-07-08 JP JP2016525422A patent/JP6567515B2/ja not_active Expired - Fee Related
- 2014-07-08 BR BR112016000338A patent/BR112016000338A8/pt not_active Application Discontinuation
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2016
- 2016-01-05 IL IL243488A patent/IL243488A0/en unknown
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2017
- 2017-07-21 US US15/656,035 patent/US20170319694A1/en not_active Abandoned
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2018
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2019
- 2019-05-21 IL IL266767A patent/IL266767A/en unknown
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2021
- 2021-08-11 US US17/399,708 patent/US20220072131A1/en not_active Abandoned
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