JP2016509589A5 - - Google Patents
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- Publication number
- JP2016509589A5 JP2016509589A5 JP2015550733A JP2015550733A JP2016509589A5 JP 2016509589 A5 JP2016509589 A5 JP 2016509589A5 JP 2015550733 A JP2015550733 A JP 2015550733A JP 2015550733 A JP2015550733 A JP 2015550733A JP 2016509589 A5 JP2016509589 A5 JP 2016509589A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- phenyl
- benzyl
- alkyl
- plant
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 claims 18
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 7
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 claims 6
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims 4
- 208000031888 Mycoses Diseases 0.000 claims 3
- 229910052736 halogen Inorganic materials 0.000 claims 3
- 150000002367 halogens Chemical class 0.000 claims 3
- 125000005842 heteroatom Chemical group 0.000 claims 3
- 150000003839 salts Chemical class 0.000 claims 3
- 229920006395 saturated elastomer Polymers 0.000 claims 3
- 238000006467 substitution reaction Methods 0.000 claims 3
- -1 -S (O) 2 R 5 Chemical group 0.000 claims 2
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims 2
- 125000000217 alkyl group Chemical group 0.000 claims 2
- 125000005129 aryl carbonyl group Chemical group 0.000 claims 2
- 230000002538 fungal effect Effects 0.000 claims 2
- 238000000034 method Methods 0.000 claims 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 2
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims 2
- 239000002689 soil Substances 0.000 claims 2
- 125000004890 (C1-C6) alkylamino group Chemical group 0.000 claims 1
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 claims 1
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims 1
- 125000006771 (C1-C6) haloalkylthio group Chemical group 0.000 claims 1
- VEXZGXHMUGYJMC-UHFFFAOYSA-N Hydrochloric acid Chemical group Cl VEXZGXHMUGYJMC-UHFFFAOYSA-N 0.000 claims 1
- CPELXLSAUQHCOX-UHFFFAOYSA-N Hydrogen bromide Chemical compound Br CPELXLSAUQHCOX-UHFFFAOYSA-N 0.000 claims 1
- 241001360088 Zymoseptoria tritici Species 0.000 claims 1
- 125000004457 alkyl amino carbonyl group Chemical group 0.000 claims 1
- 239000012876 carrier material Substances 0.000 claims 1
- 229910052801 chlorine Inorganic materials 0.000 claims 1
- 125000001309 chloro group Chemical group Cl* 0.000 claims 1
- 125000004093 cyano group Chemical group *C#N 0.000 claims 1
- XMBWDFGMSWQBCA-UHFFFAOYSA-N hydrogen iodide Chemical compound I XMBWDFGMSWQBCA-UHFFFAOYSA-N 0.000 claims 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 1
- 230000003287 optical effect Effects 0.000 claims 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims 1
- 241000894007 species Species 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261747128P | 2012-12-28 | 2012-12-28 | |
| US61/747,128 | 2012-12-28 | ||
| PCT/US2013/077478 WO2014105821A1 (en) | 2012-12-28 | 2013-12-23 | 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2016509589A JP2016509589A (ja) | 2016-03-31 |
| JP2016509589A5 true JP2016509589A5 (OSRAM) | 2017-02-09 |
| JP6336480B2 JP6336480B2 (ja) | 2018-06-06 |
Family
ID=51022027
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015550733A Active JP6336480B2 (ja) | 2012-12-28 | 2013-12-23 | １−（置換ベンゾイル）−５−フルオロ−４−イミノ−３−メチル−３，４−ジヒドロピリミジン−２（１ｈ）−オンの誘導体 |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US9271497B2 (OSRAM) |
| EP (2) | EP3689142A1 (OSRAM) |
| JP (1) | JP6336480B2 (OSRAM) |
| KR (1) | KR20150103095A (OSRAM) |
| CN (1) | CN104994859B (OSRAM) |
| AU (1) | AU2013370470B2 (OSRAM) |
| BR (1) | BR102013033840B1 (OSRAM) |
| CA (1) | CA2893776A1 (OSRAM) |
| CL (1) | CL2015001861A1 (OSRAM) |
| EC (1) | ECSP15032926A (OSRAM) |
| GT (1) | GT201500196A (OSRAM) |
| HK (1) | HK1214518A1 (OSRAM) |
| IL (1) | IL239562B (OSRAM) |
| MX (1) | MX2015008443A (OSRAM) |
| RU (2) | RU2656101C2 (OSRAM) |
| UA (1) | UA117123C2 (OSRAM) |
| WO (1) | WO2014105821A1 (OSRAM) |
| ZA (1) | ZA201504195B (OSRAM) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK2938191T3 (en) | 2012-12-28 | 2018-05-07 | Dow Agrosciences Llc | SYNERGISTIC FUNGICIDE MIXTURES FOR FERTILIZER IN GRAIN PLANTS |
| JP6324994B2 (ja) | 2012-12-28 | 2018-05-16 | アダマ・マクテシム・リミテッド | Ｎ−（置換）−５−フルオロ−４−イミノ−３−メチル−２−オキソ−３，４−ジヒドロピリミジン−１（２ｈ）−カルボキシレート誘導体 |
| MX2015008444A (es) | 2012-12-28 | 2015-09-23 | Dow Agrosciences Llc | Derivados de n-(sustituido)-5-flouro-4-imino-3-metil-2-oxo-3,4-dih idropirimidin-1 (2h)-carboximida. |
| ES2874475T3 (es) | 2012-12-31 | 2021-11-05 | Adama Makhteshim Ltd | Derivados de la 3,4-dihidropirimidin-2(1h)-ona 3-alquil-5-fluoro-4-iminosustituida como fungicidas |
| US9532570B2 (en) | 2013-12-31 | 2017-01-03 | Adama Makhteshim Ltd. | Synergistic fungicidal mixtures comprising 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1H)-one for fungal control in cereals |
| EA036389B1 (ru) | 2013-12-31 | 2020-11-03 | Адама Мактешим Лтд. | 5-фтор-4-имино-3-(алкил/замещенный алкил)-1-(арилсульфонил)-3,4-дигидропиримидин-2(1h)-он и способы их получения |
| JP6742319B2 (ja) | 2014-12-30 | 2020-08-19 | ダウ アグロサイエンシィズ エルエルシー | 殺真菌活性を有するピコリンアミド化合物 |
| CA2972408A1 (en) | 2014-12-30 | 2016-07-07 | Dow Agrosciences Llc | Use of picolinamide compounds with fungicidal activity |
| CN113173838A (zh) | 2014-12-30 | 2021-07-27 | 美国陶氏益农公司 | 具有杀真菌活性的吡啶酰胺化合物 |
| EP3255991B1 (en) | 2014-12-30 | 2020-09-30 | Dow Agrosciences LLC | Picolinamides as fungicides |
| AU2015374375B2 (en) | 2014-12-30 | 2019-03-21 | Dow Agrosciences Llc | Picolinamides with fungicidal activity |
| TWI774761B (zh) | 2017-05-02 | 2022-08-21 | 美商科迪華農業科技有限責任公司 | 用於穀物中的真菌防治之協同性混合物 |
| TW201842851A (zh) | 2017-05-02 | 2018-12-16 | 美商陶氏農業科學公司 | 用於穀類中的真菌防治之協同性混合物 |
| CA3062074A1 (en) | 2017-05-02 | 2018-11-08 | Dow Agrosciences Llc | Use of an acyclic picolinamide compound as a fungicide for fungal diseases on turfgrasses |
| CN107192785B (zh) * | 2017-06-09 | 2019-10-15 | 西南大学 | 放线菌jy-22抗真菌成分分离方法及其在复配剂中的应用 |
| WO2019038583A1 (en) | 2017-07-17 | 2019-02-28 | Adama Makhteshim Ltd. | 5-FLUORO-4-IMINO-3-METHYL-1-TOSYL-3,4-DIHYDROPYRIMIDIN-2-ONE POLYMORPHS |
| BR102019004480B1 (pt) | 2018-03-08 | 2023-03-28 | Dow Agrosciences Llc | Picolinamidas como fungicidas |
| US11639334B2 (en) | 2018-10-15 | 2023-05-02 | Corteva Agriscience Llc | Methods for synthesis of oxypicolinamides |
| CR20210270A (es) | 2018-11-05 | 2021-07-20 | Adama Makhteshim Ltd | Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de los mismos |
| CN114599639A (zh) | 2019-09-23 | 2022-06-07 | 阿达玛马克西姆有限公司 | 用于制备5-(氟-4-亚氨基-3-甲基)-1-甲苯磺酰基-3,4-二氢嘧啶-(1h)-酮的方法 |
| EP4044811A4 (en) | 2019-10-18 | 2023-09-27 | Corteva Agriscience LLC | METHOD FOR SYNTHESIS OF PICOLINAMIDS |
Family Cites Families (33)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH421973A (de) | 1962-05-01 | 1966-10-15 | Hoffmann La Roche | Verfahren zur Herstellung eines Cytosin-Derivates |
| US3309359A (en) | 1965-10-22 | 1967-03-14 | Hoffmann La Roche | N-mono-acyl-5-fluorocytosine derivatives and process |
| US3368938A (en) | 1966-01-13 | 1968-02-13 | Hoffmann La Roche | Controlling fungi with 5-fluorocytosine |
| US3868373A (en) | 1970-01-27 | 1975-02-25 | Hoffmann La Roche | 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines |
| CH579057A5 (OSRAM) | 1973-09-07 | 1976-08-31 | Hoffmann La Roche | |
| FR2530636A1 (fr) | 1982-07-23 | 1984-01-27 | Rhone Poulenc Agrochimie | Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides |
| EP0139613A1 (de) | 1983-08-29 | 1985-05-02 | Ciba-Geigy Ag | N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung |
| US4845081A (en) | 1984-10-18 | 1989-07-04 | University Of Florida | Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes |
| EP0332579B1 (de) | 1988-03-09 | 1994-08-10 | Ciba-Geigy Ag | Mittel zum Schutz von Pflanzen gegen Krankheiten |
| DE3821711A1 (de) | 1988-06-28 | 1990-02-08 | Bayer Ag | Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel |
| JP3109012B2 (ja) | 1992-06-18 | 2000-11-13 | クミアイ化学工業株式会社 | チアゾロ［５，４−ｄ］ピリミジン誘導体及び農園芸用殺菌剤 |
| JP3217191B2 (ja) | 1992-07-16 | 2001-10-09 | ビーエーエスエフ アクチェンゲゼルシャフト | ヘテロ芳香族化合物およびこれを含有する植物保護剤 |
| CN1105113C (zh) | 1995-07-05 | 2003-04-09 | 纳幕尔杜邦公司 | 杀真菌嘧啶酮 |
| TR199801813T2 (xx) | 1996-03-11 | 1998-12-21 | Novartis Ag | B�cek �ld�r�c� olarak pirimidin-4- on t�revleri. |
| HRP970239B1 (en) | 1997-05-09 | 2004-04-30 | Inst Ru Er Bouekovic | Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity |
| GT199900185A (es) | 1998-11-06 | 2001-04-18 | Novedosa pirimidin-4-enamina como fungicida. | |
| WO2003018051A1 (en) | 2001-08-27 | 2003-03-06 | Vic Jira | Anti-fungal composition |
| EP1731523A4 (en) | 2004-04-01 | 2009-08-12 | Takeda Pharmaceutical | THIAZOLOPYRIMIDINDERIVAT |
| US20080004253A1 (en) | 2006-06-30 | 2008-01-03 | Bryan James Branstetter | Thiazolopyrimidine modulators of TRPV1 |
| AU2008219166B2 (en) | 2007-02-16 | 2013-05-16 | Amgen Inc. | Nitrogen-containing heterocyclyl ketones and their use as c-Met inhibitors |
| DK2252594T3 (en) | 2008-01-22 | 2015-11-23 | Dow Agrosciences Llc | 4-amino-5-fluoro-pyrimidine derivatives as fungicides |
| US20100284959A1 (en) * | 2008-01-23 | 2010-11-11 | Gene Arrest Ltd. | Sequence specific double-stranded dna/rna binding compounds and uses thereof |
| MX2011001091A (es) | 2008-08-01 | 2011-03-15 | Dow Agrosciences Llc | Uso de 5-fluorocitosina como un fungicida. |
| SI2389375T1 (sl) | 2009-01-23 | 2015-11-30 | Euro-Celtique S.A. | Derivati hidroksamske kisline |
| UA106889C2 (uk) * | 2009-08-07 | 2014-10-27 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні n1-ацил-5-фторпіримідинону |
| AU2010279411B2 (en) | 2009-08-07 | 2014-10-23 | Adama Makhteshim Ltd. | N1-sulfonyl-5-fluoropyrimidinone derivatives |
| UA112284C2 (uk) * | 2009-08-07 | 2016-08-25 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні 5-фторпіримідинону |
| UA107671C2 (en) * | 2009-08-07 | 2015-02-10 | Dow Agrosciences Llc | N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives |
| BR112012002807B1 (pt) * | 2009-08-07 | 2018-07-10 | Adama Makhteshim Ltd. | Derivados de 5-flúor-2-oxopirimidina-1(2h)- caboxilato, composição e processo para controle e prevenção de ataque fúngico em uma planta de ataque fúngico em uma planta |
| HRP20161107T1 (hr) * | 2010-04-26 | 2016-12-30 | Adama Makhteshim Ltd | Derivati n3-supstituiranog-n1-sulfonil-5-fluoropirimidinona |
| WO2012108873A1 (en) | 2011-02-11 | 2012-08-16 | Dow Agrosciences Llc | Stable agrochemical oil dispersions |
| MX2015008444A (es) * | 2012-12-28 | 2015-09-23 | Dow Agrosciences Llc | Derivados de n-(sustituido)-5-flouro-4-imino-3-metil-2-oxo-3,4-dih idropirimidin-1 (2h)-carboximida. |
| JP6324994B2 (ja) * | 2012-12-28 | 2018-05-16 | アダマ・マクテシム・リミテッド | Ｎ−（置換）−５−フルオロ−４−イミノ−３−メチル−２−オキソ−３，４−ジヒドロピリミジン−１（２ｈ）−カルボキシレート誘導体 |
-
2013
- 2013-12-23 EP EP19217878.8A patent/EP3689142A1/en active Pending
- 2013-12-23 JP JP2015550733A patent/JP6336480B2/ja active Active
- 2013-12-23 AU AU2013370470A patent/AU2013370470B2/en not_active Ceased
- 2013-12-23 US US14/655,568 patent/US9271497B2/en active Active
- 2013-12-23 RU RU2015131110A patent/RU2656101C2/ru not_active IP Right Cessation
- 2013-12-23 HK HK16102498.5A patent/HK1214518A1/zh unknown
- 2013-12-23 CN CN201380068093.5A patent/CN104994859B/zh active Active
- 2013-12-23 KR KR1020157020064A patent/KR20150103095A/ko not_active Withdrawn
- 2013-12-23 CA CA2893776A patent/CA2893776A1/en not_active Abandoned
- 2013-12-23 UA UAA201507549A patent/UA117123C2/uk unknown
- 2013-12-23 MX MX2015008443A patent/MX2015008443A/es unknown
- 2013-12-23 EP EP13869394.0A patent/EP2945635A4/en not_active Withdrawn
- 2013-12-23 RU RU2018118951A patent/RU2018118951A/ru not_active Application Discontinuation
- 2013-12-23 WO PCT/US2013/077478 patent/WO2014105821A1/en not_active Ceased
- 2013-12-27 BR BR102013033840A patent/BR102013033840B1/pt active IP Right Grant
-
2015
- 2015-06-10 ZA ZA2015/04195A patent/ZA201504195B/en unknown
- 2015-06-21 IL IL239562A patent/IL239562B/en active IP Right Grant
- 2015-06-26 CL CL2015001861A patent/CL2015001861A1/es unknown
- 2015-06-26 GT GT201500196A patent/GT201500196A/es unknown
- 2015-07-28 EC ECIEPI201532926A patent/ECSP15032926A/es unknown
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