CN104994859B - 1-(取代的苯甲酰基)-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2(1h)-酮衍生物 - Google Patents

1-(取代的苯甲酰基)-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2(1h)-酮衍生物 Download PDF

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Publication number
CN104994859B
CN104994859B CN201380068093.5A CN201380068093A CN104994859B CN 104994859 B CN104994859 B CN 104994859B CN 201380068093 A CN201380068093 A CN 201380068093A CN 104994859 B CN104994859 B CN 104994859B
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China
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compound
alkyl
methyl
compounds
phenyl
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Chinese (zh)
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CN104994859A (zh
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B·洛尔斯巴赫
W·J·欧文
C·姚
L·施特尔策
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Adama Makhteshim Ltd
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Adama Makhteshim Ltd
Dow AgroSciences LLC
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine

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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CN201380068093.5A 2012-12-28 2013-12-23 1-(取代的苯甲酰基)-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2(1h)-酮衍生物 Active CN104994859B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261747128P 2012-12-28 2012-12-28
US61/747,128 2012-12-28
PCT/US2013/077478 WO2014105821A1 (en) 2012-12-28 2013-12-23 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives

Publications (2)

Publication Number Publication Date
CN104994859A CN104994859A (zh) 2015-10-21
CN104994859B true CN104994859B (zh) 2018-10-26

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CN201380068093.5A Active CN104994859B (zh) 2012-12-28 2013-12-23 1-(取代的苯甲酰基)-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2(1h)-酮衍生物

Country Status (18)

Country Link
US (1) US9271497B2 (OSRAM)
EP (2) EP2945635A4 (OSRAM)
JP (1) JP6336480B2 (OSRAM)
KR (1) KR20150103095A (OSRAM)
CN (1) CN104994859B (OSRAM)
AU (1) AU2013370470B2 (OSRAM)
BR (1) BR102013033840B1 (OSRAM)
CA (1) CA2893776A1 (OSRAM)
CL (1) CL2015001861A1 (OSRAM)
EC (1) ECSP15032926A (OSRAM)
GT (1) GT201500196A (OSRAM)
HK (1) HK1214518A1 (OSRAM)
IL (1) IL239562B (OSRAM)
MX (1) MX2015008443A (OSRAM)
RU (2) RU2018118951A (OSRAM)
UA (1) UA117123C2 (OSRAM)
WO (1) WO2014105821A1 (OSRAM)
ZA (1) ZA201504195B (OSRAM)

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EA030056B1 (ru) 2013-12-31 2018-06-29 Адама Мактешим Лтд. Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами
RU2017123619A (ru) 2014-12-30 2019-01-31 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Соединения пиколинамида с фунгицидной активностью
BR112017013758B1 (pt) 2014-12-30 2021-11-23 Dow Agrosciences Llc Compostos de picolinamida com atividade fungicida
BR112017013767A2 (pt) 2014-12-30 2018-03-13 Dow Agrosciences Llc uso de picolinamidas como fungicidas
JP6629862B2 (ja) 2014-12-30 2020-01-15 ダウ アグロサイエンシィズ エルエルシー 殺真菌活性を有するピコリンアミド
CA2972401C (en) 2014-12-30 2023-09-05 Dow Agrosciences Llc Picolinamide compounds with fungicidal activity
US20200085047A1 (en) 2017-05-02 2020-03-19 Dow Agrosciences Llc Use of an Acyclic Picolinamide Compound as a Fungicide for Control of Phytopathogenic Fungi in Vegetables
TWI774761B (zh) 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
TW201842851A (zh) 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
CN107192785B (zh) * 2017-06-09 2019-10-15 西南大学 放线菌jy-22抗真菌成分分离方法及其在复配剂中的应用
MA49639A (fr) 2017-07-17 2020-05-27 Adama Makhteshim Ltd Polymorphes de 5-fluoro-4-imino-3-méthyl-1-tosyl-3,4-dihydropyrimidin-2-one
BR102019004480B1 (pt) 2018-03-08 2023-03-28 Dow Agrosciences Llc Picolinamidas como fungicidas
KR20210076072A (ko) 2018-10-15 2021-06-23 코르테바 애그리사이언스 엘엘씨 옥시피콜린아미드의 합성 방법
CR20210270A (es) 2018-11-05 2021-07-20 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de los mismos
US12466796B2 (en) 2019-09-23 2025-11-11 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1H)-one and derivatives of the compound
EP4044811A4 (en) 2019-10-18 2023-09-27 Corteva Agriscience LLC METHOD FOR SYNTHESIS OF PICOLINAMIDS

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Publication number Publication date
US9271497B2 (en) 2016-03-01
GT201500196A (es) 2016-03-02
MX2015008443A (es) 2015-09-23
CL2015001861A1 (es) 2015-10-02
ZA201504195B (en) 2017-08-30
WO2014105821A1 (en) 2014-07-03
RU2018118951A (ru) 2018-11-02
EP2945635A1 (en) 2015-11-25
RU2018118951A3 (OSRAM) 2019-02-26
ECSP15032926A (es) 2015-11-30
JP2016509589A (ja) 2016-03-31
HK1216147A1 (zh) 2016-10-21
IL239562A0 (en) 2015-08-31
KR20150103095A (ko) 2015-09-09
CN104994859A (zh) 2015-10-21
AU2013370470A1 (en) 2015-07-02
BR102013033840B1 (pt) 2019-09-10
IL239562B (en) 2018-02-28
UA117123C2 (uk) 2018-06-25
EP3689142A1 (en) 2020-08-05
RU2656101C2 (ru) 2018-05-31
RU2015131110A (ru) 2017-02-03
CA2893776A1 (en) 2014-07-03
BR102013033840A2 (pt) 2015-10-06
EP2945635A4 (en) 2016-05-25
US20150342188A1 (en) 2015-12-03
HK1214518A1 (zh) 2016-07-29
JP6336480B2 (ja) 2018-06-06
AU2013370470B2 (en) 2018-05-10

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