CA2893776A1 - 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives - Google Patents

1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives Download PDF

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Publication number
CA2893776A1
CA2893776A1 CA2893776A CA2893776A CA2893776A1 CA 2893776 A1 CA2893776 A1 CA 2893776A1 CA 2893776 A CA2893776 A CA 2893776A CA 2893776 A CA2893776 A CA 2893776A CA 2893776 A1 CA2893776 A1 CA 2893776A1
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CA
Canada
Prior art keywords
compounds
plant
formula
methyl
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA2893776A
Other languages
English (en)
French (fr)
Inventor
Beth Lorsbach
W. John Owen
Chenglin Yao
Lindsay Stelzer
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Adama Makhteshim Ltd
Original Assignee
Dow AgroSciences LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow AgroSciences LLC filed Critical Dow AgroSciences LLC
Publication of CA2893776A1 publication Critical patent/CA2893776A1/en
Abandoned legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine

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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA2893776A 2012-12-28 2013-12-23 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives Abandoned CA2893776A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261747128P 2012-12-28 2012-12-28
US61/747,128 2012-12-28
PCT/US2013/077478 WO2014105821A1 (en) 2012-12-28 2013-12-23 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives

Publications (1)

Publication Number Publication Date
CA2893776A1 true CA2893776A1 (en) 2014-07-03

Family

ID=51022027

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2893776A Abandoned CA2893776A1 (en) 2012-12-28 2013-12-23 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives

Country Status (18)

Country Link
US (1) US9271497B2 (OSRAM)
EP (2) EP3689142A1 (OSRAM)
JP (1) JP6336480B2 (OSRAM)
KR (1) KR20150103095A (OSRAM)
CN (1) CN104994859B (OSRAM)
AU (1) AU2013370470B2 (OSRAM)
BR (1) BR102013033840B1 (OSRAM)
CA (1) CA2893776A1 (OSRAM)
CL (1) CL2015001861A1 (OSRAM)
EC (1) ECSP15032926A (OSRAM)
GT (1) GT201500196A (OSRAM)
HK (1) HK1214518A1 (OSRAM)
IL (1) IL239562B (OSRAM)
MX (1) MX2015008443A (OSRAM)
RU (2) RU2656101C2 (OSRAM)
UA (1) UA117123C2 (OSRAM)
WO (1) WO2014105821A1 (OSRAM)
ZA (1) ZA201504195B (OSRAM)

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JP6324994B2 (ja) 2012-12-28 2018-05-16 アダマ・マクテシム・リミテッド Ｎ−（置換）−５−フルオロ−４−イミノ−３−メチル−２−オキソ−３，４−ジヒドロピリミジン−１（２ｈ）−カルボキシレート誘導体
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ES2874475T3 (es) 2012-12-31 2021-11-05 Adama Makhteshim Ltd Derivados de la 3,4-dihidropirimidin-2(1h)-ona 3-alquil-5-fluoro-4-iminosustituida como fungicidas
US9532570B2 (en) 2013-12-31 2017-01-03 Adama Makhteshim Ltd. Synergistic fungicidal mixtures comprising 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1H)-one for fungal control in cereals
EA036389B1 (ru) 2013-12-31 2020-11-03 Адама Мактешим Лтд. 5-фтор-4-имино-3-(алкил/замещенный алкил)-1-(арилсульфонил)-3,4-дигидропиримидин-2(1h)-он и способы их получения
JP6742319B2 (ja) 2014-12-30 2020-08-19 ダウ アグロサイエンシィズ エルエルシー 殺真菌活性を有するピコリンアミド化合物
CA2972408A1 (en) 2014-12-30 2016-07-07 Dow Agrosciences Llc Use of picolinamide compounds with fungicidal activity
CN113173838A (zh) 2014-12-30 2021-07-27 美国陶氏益农公司 具有杀真菌活性的吡啶酰胺化合物
EP3255991B1 (en) 2014-12-30 2020-09-30 Dow Agrosciences LLC Picolinamides as fungicides
AU2015374375B2 (en) 2014-12-30 2019-03-21 Dow Agrosciences Llc Picolinamides with fungicidal activity
TWI774761B (zh) 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
TW201842851A (zh) 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
CA3062074A1 (en) 2017-05-02 2018-11-08 Dow Agrosciences Llc Use of an acyclic picolinamide compound as a fungicide for fungal diseases on turfgrasses
CN107192785B (zh) * 2017-06-09 2019-10-15 西南大学 放线菌jy-22抗真菌成分分离方法及其在复配剂中的应用
WO2019038583A1 (en) 2017-07-17 2019-02-28 Adama Makhteshim Ltd. 5-FLUORO-4-IMINO-3-METHYL-1-TOSYL-3,4-DIHYDROPYRIMIDIN-2-ONE POLYMORPHS
BR102019004480B1 (pt) 2018-03-08 2023-03-28 Dow Agrosciences Llc Picolinamidas como fungicidas
US11639334B2 (en) 2018-10-15 2023-05-02 Corteva Agriscience Llc Methods for synthesis of oxypicolinamides
CR20210270A (es) 2018-11-05 2021-07-20 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de los mismos
CN114599639A (zh) 2019-09-23 2022-06-07 阿达玛马克西姆有限公司 用于制备5-(氟-4-亚氨基-3-甲基)-1-甲苯磺酰基-3,4-二氢嘧啶-(1h)-酮的方法
EP4044811A4 (en) 2019-10-18 2023-09-27 Corteva Agriscience LLC METHOD FOR SYNTHESIS OF PICOLINAMIDS

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Also Published As

Publication number Publication date
RU2015131110A (ru) 2017-02-03
ECSP15032926A (es) 2015-11-30
HK1216147A1 (zh) 2016-10-21
HK1214518A1 (zh) 2016-07-29
RU2656101C2 (ru) 2018-05-31
US20150342188A1 (en) 2015-12-03
CL2015001861A1 (es) 2015-10-02
KR20150103095A (ko) 2015-09-09
EP2945635A1 (en) 2015-11-25
CN104994859A (zh) 2015-10-21
IL239562A0 (en) 2015-08-31
ZA201504195B (en) 2017-08-30
CN104994859B (zh) 2018-10-26
EP3689142A1 (en) 2020-08-05
MX2015008443A (es) 2015-09-23
IL239562B (en) 2018-02-28
EP2945635A4 (en) 2016-05-25
US9271497B2 (en) 2016-03-01
JP2016509589A (ja) 2016-03-31
BR102013033840B1 (pt) 2019-09-10
UA117123C2 (uk) 2018-06-25
GT201500196A (es) 2016-03-02
RU2018118951A3 (OSRAM) 2019-02-26
WO2014105821A1 (en) 2014-07-03
JP6336480B2 (ja) 2018-06-06
BR102013033840A2 (pt) 2015-10-06
AU2013370470B2 (en) 2018-05-10
RU2018118951A (ru) 2018-11-02
AU2013370470A1 (en) 2015-07-02

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Legal Events

Date Code Title Description
FZDE Discontinued

Effective date: 20191224