JP2016000739A5 - - Google Patents

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Publication number
JP2016000739A5
JP2016000739A5 JP2015139845A JP2015139845A JP2016000739A5 JP 2016000739 A5 JP2016000739 A5 JP 2016000739A5 JP 2015139845 A JP2015139845 A JP 2015139845A JP 2015139845 A JP2015139845 A JP 2015139845A JP 2016000739 A5 JP2016000739 A5 JP 2016000739A5
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JP
Japan
Prior art keywords
xrpd
pattern
diffractometer
angstroms
angles
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2015139845A
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English (en)
Japanese (ja)
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JP6404186B2 (ja
JP2016000739A (ja
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Publication date
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Publication of JP2016000739A publication Critical patent/JP2016000739A/ja
Publication of JP2016000739A5 publication Critical patent/JP2016000739A5/ja
Application granted granted Critical
Publication of JP6404186B2 publication Critical patent/JP6404186B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2015139845A 2009-08-27 2015-07-13 無水形態のピリジン誘導体 Active JP6404186B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23743509P 2009-08-27 2009-08-27
US61/237,435 2009-08-27

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2012526048A Division JP2013503134A (ja) 2009-08-27 2010-08-25 無水形態のピリジン誘導体

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2017114602A Division JP2017193564A (ja) 2009-08-27 2017-06-09 無水形態のピリジン誘導体

Publications (3)

Publication Number Publication Date
JP2016000739A JP2016000739A (ja) 2016-01-07
JP2016000739A5 true JP2016000739A5 (enExample) 2017-08-10
JP6404186B2 JP6404186B2 (ja) 2018-10-10

Family

ID=42790943

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2012526048A Pending JP2013503134A (ja) 2009-08-27 2010-08-25 無水形態のピリジン誘導体
JP2015139845A Active JP6404186B2 (ja) 2009-08-27 2015-07-13 無水形態のピリジン誘導体
JP2017114602A Pending JP2017193564A (ja) 2009-08-27 2017-06-09 無水形態のピリジン誘導体

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2012526048A Pending JP2013503134A (ja) 2009-08-27 2010-08-25 無水形態のピリジン誘導体

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2017114602A Pending JP2017193564A (ja) 2009-08-27 2017-06-09 無水形態のピリジン誘導体

Country Status (17)

Country Link
US (1) US8796269B2 (enExample)
EP (1) EP2470545B1 (enExample)
JP (3) JP2013503134A (enExample)
KR (1) KR20120056258A (enExample)
CN (1) CN102639536B (enExample)
AU (1) AU2010288502B2 (enExample)
CA (1) CA2772168C (enExample)
DK (1) DK2470545T3 (enExample)
EA (1) EA021411B1 (enExample)
ES (1) ES2440938T3 (enExample)
IL (1) IL217922A (enExample)
IN (1) IN2012DN01292A (enExample)
MX (1) MX2012002369A (enExample)
PL (1) PL2470545T3 (enExample)
SG (1) SG178231A1 (enExample)
WO (1) WO2011023733A1 (enExample)
ZA (1) ZA201200812B (enExample)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2010288502B2 (en) * 2009-08-27 2013-12-12 KaNDy Therapeutics Ltd. Anhydrate forms of a pyridine derivative
EP3915560A1 (en) * 2014-06-25 2021-12-01 Emory University Methods of managing conditioned fear with neurokinin receptor antagonists
HUE047732T2 (hu) 2015-05-18 2020-05-28 Nerre Therapeutics Ltd NK-1/NK-3 receptor antagonista vértolulások kezeléséhez
US11028099B2 (en) * 2016-12-15 2021-06-08 Glaxosmithkline Intellectual Property Development Limited NRF2 activators
PL3765024T3 (pl) 2018-03-14 2024-08-05 KaNDy Therapeutics Limited <div>Nowa formulacja farmaceutyczna zawierająca podwójnych antagonistów receptora nk-1/nk-3</div>
WO2021030335A1 (en) * 2019-08-12 2021-02-18 Millendo Therapeutics, Inc. A stereoisomerically pure nk-3 receptor antagonist and crystalline forms thereof
JP7673064B2 (ja) 2019-11-15 2025-05-08 カンディー セラピューティクス リミテッド Nt-814の重要な中間体である6-クロロ-4-(4-フルオロ-2-メチルフェニル)ピリジン-3-アミンを作製するための新規な化学的方法
EP4431512A1 (en) 2023-03-16 2024-09-18 Bayer Consumer Care AG Novel dual nk-1/nk-3 receptor antagonists
WO2025242585A1 (en) 2024-05-24 2025-11-27 Bayer Consumer Care Ag Crystalline forms of salts of elinzanetant and compositions containing salts of elinzanetant
WO2025242583A1 (en) 2024-05-24 2025-11-27 Bayer Consumer Care Ag Novel formulation comprising elinzanetant in a solid dispersion
WO2025242584A1 (en) 2024-05-24 2025-11-27 Bayer Consumer Care Ag A stable soft gelatin capsule formulation for elinzanetant
TW202604529A (zh) * 2024-06-18 2026-02-01 瑞士商拜耳保健消費品股份有限公司 用於製造依林奈坦(elinzanetant)前驅物之改良方法
US12533358B1 (en) 2025-05-14 2026-01-27 Bayer Consumer Care Ag Methods of treatment with elinzanetant

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK1394150T3 (da) * 1999-02-24 2011-03-21 Hoffmann La Roche 4-phenylpyridinderivater og deres anvendelse som NK-1-receptorantagonister
GB0203022D0 (en) * 2002-02-08 2002-03-27 Glaxo Group Ltd Chemical compounds
PL378404A1 (pl) * 2003-01-31 2006-04-03 F. Hoffmann-La Roche Ag Nowa odmiana krystaliczna 2-(3,5-bis-trifluorometylofenylo)-N-[6-(1,1-diokso-1<$Elambda>6 -tiomorfolin-4-ylo)-4-(4-fluoro-2-metylofenylo)pirydyn-3-ylo]-N-metyloizobutyroamidu
HRP20070471T3 (hr) * 2003-07-03 2007-11-30 F. Hoffmann - La Roche Ag Dvojni nk1/nk3 antagonisti za liječenje shizofrenije
US7683056B2 (en) * 2005-09-09 2010-03-23 Glaxosmithkline Llc Pyridine derivatives and their use in the treatment of psychotic disorders
KR20100101051A (ko) * 2007-12-11 2010-09-16 씨아이피엘에이 엘티디. 조피클론 결정성 다형체, 이들의 제조 공정 및 이들의 약제 조성물
GB0814340D0 (en) * 2008-08-05 2008-09-10 Smithkline Beecham Corp Anhydrous crystol form fo a pyridine derivative
AU2010288502B2 (en) * 2009-08-27 2013-12-12 KaNDy Therapeutics Ltd. Anhydrate forms of a pyridine derivative
JP6342662B2 (ja) * 2014-01-29 2018-06-13 京セラ株式会社 ドリルおよびそれを用いた切削加工物の製造方法

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