JP2015520165A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2015520165A5 JP2015520165A5 JP2015512903A JP2015512903A JP2015520165A5 JP 2015520165 A5 JP2015520165 A5 JP 2015520165A5 JP 2015512903 A JP2015512903 A JP 2015512903A JP 2015512903 A JP2015512903 A JP 2015512903A JP 2015520165 A5 JP2015520165 A5 JP 2015520165A5
- Authority
- JP
- Japan
- Prior art keywords
- salt
- compound
- formula
- process according
- hydrogen
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261648534P | 2012-05-17 | 2012-05-17 | |
| US61/648,534 | 2012-05-17 | ||
| PCT/US2013/041687 WO2013173779A1 (en) | 2012-05-17 | 2013-05-17 | Process for making amino acid compounds |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2015520165A JP2015520165A (ja) | 2015-07-16 |
| JP2015520165A5 true JP2015520165A5 (OSRAM) | 2016-06-30 |
| JP6196294B2 JP6196294B2 (ja) | 2017-09-13 |
Family
ID=48483247
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015512903A Active JP6196294B2 (ja) | 2012-05-17 | 2013-05-17 | アミノ酸化合物を製造するためのプロセス |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US9278917B2 (OSRAM) |
| EP (1) | EP2850054B1 (OSRAM) |
| JP (1) | JP6196294B2 (OSRAM) |
| KR (1) | KR102074535B1 (OSRAM) |
| CN (1) | CN104520263B (OSRAM) |
| AU (1) | AU2013262516B2 (OSRAM) |
| BR (1) | BR112014028585B1 (OSRAM) |
| CA (1) | CA2873658C (OSRAM) |
| ES (1) | ES2668477T3 (OSRAM) |
| HR (1) | HRP20180948T1 (OSRAM) |
| IL (1) | IL235630A (OSRAM) |
| MA (1) | MA37751B1 (OSRAM) |
| MX (1) | MX350443B (OSRAM) |
| MY (1) | MY171538A (OSRAM) |
| NZ (1) | NZ702939A (OSRAM) |
| PL (1) | PL2850054T3 (OSRAM) |
| RU (1) | RU2643146C2 (OSRAM) |
| SG (1) | SG11201407625WA (OSRAM) |
| SI (1) | SI2850054T1 (OSRAM) |
| TR (1) | TR201807444T4 (OSRAM) |
| WO (1) | WO2013173779A1 (OSRAM) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ702935A (en) | 2012-05-17 | 2017-02-24 | Genentech Inc | Process for making hydroxylated cyclopentylpyrimidine compounds |
| ES2588878T3 (es) | 2012-05-17 | 2016-11-07 | Array Biopharma, Inc. | Proceso para preparar compuestos de ciclopentilpirimidina hidroxilada |
| CA2873661C (en) | 2012-05-17 | 2020-07-21 | Genentech, Inc. | Process of making hydroxylated cyclopentapyrimidine compounds and salts thereof |
| EP3719014A1 (en) | 2012-05-17 | 2020-10-07 | Genentech, Inc. | Solid forms of an akt inhibiting pyrimidinyl-cyclopentane compound, compositions and methods thereof |
| CN112898210B (zh) * | 2013-11-15 | 2025-02-21 | 豪夫迈·罗氏有限公司 | 用于制备嘧啶基环戊烷化合物的方法 |
| CA3190507A1 (en) * | 2014-09-26 | 2016-03-31 | F. Hoffmann-La Roche Ag | Processes for preparing (cyclopentyl[d]pyrimidin-4-yl)piperazine compounds |
Family Cites Families (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4663327A (en) | 1984-05-23 | 1987-05-05 | Bayer Aktiengesellschaft | 1-heteroaryl-4-aryl-pyrazolin-5-ones |
| JPH09506369A (ja) | 1993-12-12 | 1997-06-24 | アグロジーン・リミテッド | 菌類感染から植物を保護するための新規方法 |
| AU724216B2 (en) | 1997-04-07 | 2000-09-14 | Merck & Co., Inc. | A method of treating cancer |
| US6201023B1 (en) | 1997-06-10 | 2001-03-13 | Agrogene Ltd. | Methods and compositions to protect crops against plant parasitic nematodes |
| EP0982300A3 (en) | 1998-07-29 | 2000-03-08 | Societe Civile Bioprojet | Non-imidazole alkylamines as histamine H3 - receptor ligands and their therapeutic applications |
| US6376496B1 (en) | 1999-03-03 | 2002-04-23 | Merck & Co., Inc. | Inhibitors of prenyl-protein transferase |
| WO2001022963A1 (en) | 1999-09-27 | 2001-04-05 | Merck & Co., Inc. | Method of preventing osteoporosis |
| WO2004108673A2 (en) | 2003-06-09 | 2004-12-16 | Boehringer Ingelheim International Gmbh | Inhibitors of papilloma virus |
| FR2892416B1 (fr) * | 2005-10-20 | 2008-06-27 | Sanofi Aventis Sa | Derives de 6-heteroarylpyridoindolone, leur preparation et leur application en therapeutique |
| US8927546B2 (en) | 2006-02-28 | 2015-01-06 | Dart Neuroscience (Cayman) Ltd. | Therapeutic piperazines |
| UA95641C2 (xx) * | 2006-07-06 | 2011-08-25 | Эррей Биофарма Инк. | Гідроксильовані піримідильні циклопентани як інгібітори акт протеїнкінази$гидроксилированные пиримидильные циклопентаны как ингибиторы акт протеинкиназы |
| US8063050B2 (en) | 2006-07-06 | 2011-11-22 | Array Biopharma Inc. | Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors |
| EP2209775A1 (en) | 2007-10-09 | 2010-07-28 | UCB Pharma, S.A. | Heterobicyclic compounds as histamine h4-receptor antagonists |
| JP5734956B2 (ja) | 2009-04-15 | 2015-06-17 | アッヴィ・インコーポレイテッド | 抗ウィルス化合物 |
| EA020151B1 (ru) | 2009-10-23 | 2014-09-30 | Эли Лилли Энд Компани | Ингибиторы akt и фармацевтические составы, их содержащие |
| US9050334B2 (en) | 2010-07-16 | 2015-06-09 | Innov88 Llc | MIF inhibitors and their uses |
| WO2012177925A1 (en) | 2011-06-21 | 2012-12-27 | The Board Institute, Inc. | Akt inhibitors for treating cancer expressing a magi3 - akt3 fusion gene |
| ES2588878T3 (es) | 2012-05-17 | 2016-11-07 | Array Biopharma, Inc. | Proceso para preparar compuestos de ciclopentilpirimidina hidroxilada |
| CA2873661C (en) | 2012-05-17 | 2020-07-21 | Genentech, Inc. | Process of making hydroxylated cyclopentapyrimidine compounds and salts thereof |
| CA2889855A1 (en) | 2012-11-01 | 2014-05-08 | Robert S. Katz | Methods for treating fibromyalgia |
| CN105263910A (zh) | 2013-02-18 | 2016-01-20 | 斯克利普斯研究所 | 具有治疗潜力的血管加压素受体调节剂 |
| AU2014237198A1 (en) | 2013-03-15 | 2015-11-05 | Shifa Biomedical Corporation | Anti-PCSK9 compounds and methods for the treatment and/or prevention of cardiovascular diseases |
-
2013
- 2013-05-17 HR HRP20180948TT patent/HRP20180948T1/hr unknown
- 2013-05-17 SI SI201331043T patent/SI2850054T1/en unknown
- 2013-05-17 RU RU2014150991A patent/RU2643146C2/ru active
- 2013-05-17 CN CN201380037572.0A patent/CN104520263B/zh active Active
- 2013-05-17 WO PCT/US2013/041687 patent/WO2013173779A1/en not_active Ceased
- 2013-05-17 MA MA37751A patent/MA37751B1/fr unknown
- 2013-05-17 SG SG11201407625WA patent/SG11201407625WA/en unknown
- 2013-05-17 EP EP13724711.0A patent/EP2850054B1/en active Active
- 2013-05-17 US US14/401,095 patent/US9278917B2/en active Active
- 2013-05-17 CA CA2873658A patent/CA2873658C/en active Active
- 2013-05-17 JP JP2015512903A patent/JP6196294B2/ja active Active
- 2013-05-17 BR BR112014028585-3A patent/BR112014028585B1/pt active IP Right Grant
- 2013-05-17 KR KR1020147035263A patent/KR102074535B1/ko active Active
- 2013-05-17 AU AU2013262516A patent/AU2013262516B2/en active Active
- 2013-05-17 MX MX2014013863A patent/MX350443B/es active IP Right Grant
- 2013-05-17 ES ES13724711.0T patent/ES2668477T3/es active Active
- 2013-05-17 TR TR2018/07444T patent/TR201807444T4/tr unknown
- 2013-05-17 MY MYPI2014703417A patent/MY171538A/en unknown
- 2013-05-17 NZ NZ702939A patent/NZ702939A/en not_active IP Right Cessation
- 2013-05-17 PL PL13724711T patent/PL2850054T3/pl unknown
-
2014
- 2014-11-11 IL IL235630A patent/IL235630A/en active IP Right Grant
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2015520165A5 (OSRAM) | ||
| RU2012103850A (ru) | Би-арил-мета-пиримидиновые ингибиторы киназ | |
| JP2011057686A5 (OSRAM) | ||
| JP2013521295A5 (OSRAM) | ||
| JP2009507932A5 (OSRAM) | ||
| JP2007269812A5 (OSRAM) | ||
| JP2011105738A5 (OSRAM) | ||
| JP2012507568A5 (OSRAM) | ||
| ME02558B (me) | Inhibitori replikacije virusa gripa | |
| JP2015518892A5 (OSRAM) | ||
| JP2007522220A5 (OSRAM) | ||
| JP2011513410A5 (OSRAM) | ||
| JP2011510079A5 (OSRAM) | ||
| EP4219465A3 (en) | Prmt5 inhibitors and uses thereof | |
| JP2011227454A5 (OSRAM) | ||
| JP2013500304A5 (OSRAM) | ||
| JP2015518837A5 (OSRAM) | ||
| AR083105A1 (es) | Metodo para preparar 2-amino-n-(2,2,2-trifluoroetil)acetamida | |
| MX2007007098A (es) | Derivados de pirrol que tienen actividad antagonista del receptor crth2. | |
| RU2014150991A (ru) | Способ получения аминокислотных соединений | |
| JP2007526383A5 (OSRAM) | ||
| EP2759540A3 (en) | Beta-3 receptor ligands and their use in therapy | |
| JP2006518752A5 (OSRAM) | ||
| JP2012511558A5 (OSRAM) | ||
| JP2009532434A5 (OSRAM) |