JP2015505555A5 - - Google Patents

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Publication number
JP2015505555A5
JP2015505555A5 JP2014555310A JP2014555310A JP2015505555A5 JP 2015505555 A5 JP2015505555 A5 JP 2015505555A5 JP 2014555310 A JP2014555310 A JP 2014555310A JP 2014555310 A JP2014555310 A JP 2014555310A JP 2015505555 A5 JP2015505555 A5 JP 2015505555A5
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JP
Japan
Prior art keywords
inhibition
cancer
compound
protein kinase
autoimmune disorders
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2014555310A
Other languages
English (en)
Japanese (ja)
Other versions
JP2015505555A (ja
JP6199316B2 (ja
Filing date
Publication date
Priority claimed from GBGB1201566.5A external-priority patent/GB201201566D0/en
Application filed filed Critical
Publication of JP2015505555A publication Critical patent/JP2015505555A/ja
Publication of JP2015505555A5 publication Critical patent/JP2015505555A5/ja
Application granted granted Critical
Publication of JP6199316B2 publication Critical patent/JP6199316B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2014555310A 2012-01-30 2013-01-30 1H−ピロロ[2,3−b]ピリジン誘導体およびキナーゼ阻害剤としてのその使用 Expired - Fee Related JP6199316B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB1201566.5 2012-01-30
GBGB1201566.5A GB201201566D0 (en) 2012-01-30 2012-01-30 New chemical compounds
PCT/GB2013/050212 WO2013114113A1 (en) 2012-01-30 2013-01-30 1h-pyrrolo[2,3-b] pyridine derivatives and their use as kinase inhibitors

Publications (3)

Publication Number Publication Date
JP2015505555A JP2015505555A (ja) 2015-02-23
JP2015505555A5 true JP2015505555A5 (https=) 2015-11-12
JP6199316B2 JP6199316B2 (ja) 2017-09-20

Family

ID=45876325

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2014555310A Expired - Fee Related JP6199316B2 (ja) 2012-01-30 2013-01-30 1H−ピロロ[2,3−b]ピリジン誘導体およびキナーゼ阻害剤としてのその使用

Country Status (21)

Country Link
US (3) US10000481B2 (https=)
EP (1) EP2809670B1 (https=)
JP (1) JP6199316B2 (https=)
CN (4) CN107011341A (https=)
AU (1) AU2013213954B2 (https=)
BR (1) BR112014018795B1 (https=)
CA (1) CA2862940C (https=)
DK (1) DK2809670T3 (https=)
EA (1) EA026657B1 (https=)
ES (1) ES2637340T3 (https=)
GB (1) GB201201566D0 (https=)
HK (1) HK1200447A1 (https=)
HU (1) HUE035332T2 (https=)
IL (1) IL233595B (https=)
IN (1) IN2014DN06104A (https=)
MX (1) MX352927B (https=)
NZ (1) NZ627361A (https=)
PL (1) PL2809670T3 (https=)
PT (1) PT2809670T (https=)
WO (1) WO2013114113A1 (https=)
ZA (1) ZA201405070B (https=)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB201201566D0 (en) * 2012-01-30 2012-03-14 Vernalis R&D Ltd New chemical compounds
SG11201406818VA (en) * 2012-04-23 2014-11-27 Genentech Inc Intermediates and processes for preparing compounds
CN105705499B (zh) * 2013-08-22 2018-10-12 基因泰克公司 用于制备化合物的方法
CN104829609B (zh) * 2014-02-11 2016-08-03 北大方正集团有限公司 取代的吡啶并嘧啶化合物及其制备方法和应用
MA41559A (fr) * 2015-09-08 2017-12-26 Taiho Pharmaceutical Co Ltd Composé de pyrimidine condensé ou un sel de celui-ci
US10032914B2 (en) * 2015-10-20 2018-07-24 Taiwan Semiconductor Manufacturing Co., Ltd. Semiconductor device and manufacturing method thereof
CA3015484C (en) 2016-02-23 2022-11-08 Taiho Pharmaceutical Co., Ltd. Novel condensed pyrimidine compound or salt thereof
EP3674325A4 (en) 2017-08-21 2021-11-03 Taiho Pharmaceutical Co., Ltd. FUSION PROTEIN OF DCTN1 PROTEIN WITH RET PROTEIN
TW202043198A (zh) 2019-01-17 2020-12-01 美商Ifm Due有限公司 用於治療與sting活性相關之病況的化合物及組合物
CN111518096B (zh) 2019-02-02 2022-02-11 江苏威凯尔医药科技有限公司 两面神激酶jak家族抑制剂及其制备和应用
US12428395B2 (en) 2019-08-01 2025-09-30 Sperogenix Therapeutics Limited Heterocyclic compounds as kinase inhibitor and uses thereof
IT202000005527A1 (it) * 2020-03-16 2021-09-16 Univ Degli Studi Di Trento Trattamento terapeutico di cromatinopatie
JP2023540674A (ja) * 2020-07-15 2023-09-26 アイエフエム デュー インコーポレイテッド Sting活性に関連する状態を治療するための化合物および組成物
WO2022015975A1 (en) 2020-07-15 2022-01-20 Ifm Due, Inc. Compounds and compositions for treating conditions associated with sting activity
PY2157405A (es) * 2020-07-15 2022-04-22 Ifm Due Inc Compuestos y composiciones para el tratamiento de afecciones asociadas a la actividad del sting
EP4274824A1 (en) 2021-01-08 2023-11-15 IFM Due, Inc. Heterobicyclic compounds having an urea or analogue and their compositions for treating conditions associated with sting activity
IL310724A (en) 2021-08-10 2024-04-01 Ifm Due Inc COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH STING ACTIVITY
CN118613473A (zh) * 2022-01-12 2024-09-06 艾福姆德尤股份有限公司 用于治疗与sting活性相关的病症的化合物和组合物
CN116554170A (zh) * 2023-04-26 2023-08-08 上海大学 4-氟-7-氮杂吲哚的制备方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US1012976A (en) * 1909-03-25 1911-12-26 Adolf Bordt Adding-machine.
WO2003028724A1 (en) * 2001-10-04 2003-04-10 Smithkline Beecham Corporation Chk1 kinase inhibitors
US7531553B2 (en) * 2003-03-21 2009-05-12 Amgen Inc. Heterocyclic compounds and methods of use
NZ590160A (en) * 2003-11-21 2012-07-27 Array Biopharma Inc AKT protein kinase inhibitors
CA2711614A1 (en) * 2008-01-08 2009-07-16 Array Biopharma Inc. Pyrrolopyridines as kinase inhibitors
DK2294065T3 (da) * 2008-01-22 2014-04-28 Vernalis R&D Ltd Indolyl-pyridonderivater med checkpoint kinase 1 inhibitorisk aktivitet
CL2009001152A1 (es) * 2008-05-13 2009-10-16 Array Biopharma Inc Compuestos derivados de n-(4-(cicloalquilo nitrogenado-1-il)-1h-pirrolo[2,3-b]piridin-3-il)amida, inhibidores de cinasa; proceso de preparacion; composicion farmaceutica; y su uso para el tratamiento de una enfermedad proliferativa.
KR20110015699A (ko) 2008-06-11 2011-02-16 제넨테크, 인크. 디아자카르바졸 및 사용 방법
CN102573994B (zh) * 2009-08-06 2015-06-24 默克专利有限公司 双环脲化合物
US9290499B2 (en) * 2010-05-19 2016-03-22 The University Of North Carolina At Chapel Hill Pyrazolopyrimidine compounds for the treatment of cancer
GB201201566D0 (en) * 2012-01-30 2012-03-14 Vernalis R&D Ltd New chemical compounds

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